SI9300581A - Transdermal therapeutic system with estradiol as activ substance - Google Patents

Transdermal therapeutic system with estradiol as activ substance Download PDF

Info

Publication number: SI9300581A
Authority: SI; Slovenia
Prior art keywords: estradiol; humidity; transdermal therapeutic; therapeutic system; active substance
Prior art date: 1992-11-06

Application number

SI9300581A

Other languages

English (en)

Slovenian (sl)

Inventor

Michael Horstmann

Sylvia Hahn

Reinhold Meconi

Robert-Peter Klein

Original Assignee

Lohmann Therapie Syst Lts

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-11-06

Filing date

1993-11-05

Publication date

1994-06-30

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6472230&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI9300581(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1993-11-05 Application filed by Lohmann Therapie Syst Lts filed Critical Lohmann Therapie Syst Lts

1994-06-30 Publication of SI9300581A publication Critical patent/SI9300581A/sl

Links

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229930182833 estradiol Natural products 0.000 title claims abstract description 31
230000001225 therapeutic effect Effects 0.000 title claims abstract description 16
239000000126 substance Substances 0.000 title claims description 4
239000013543 active substance Substances 0.000 claims abstract description 25
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
- A61K9/7061—Polyacrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7069—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained otherwise than by reactions only involving carbon to carbon unsaturated bonds, e.g. polysiloxane, polyesters, polyurethane, polyethylene oxide
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7092—Transdermal patches having multiple drug layers or reservoirs, e.g. for obtaining a specific release pattern, or for combining different drugs

Landscapes

Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Dermatology (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Steroid Compounds (AREA)

SI9300581A 1992-11-06 1993-11-05 Transdermal therapeutic system with estradiol as activ substance SI9300581A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE4237453A DE4237453C1 (sh)	1992-11-06	1992-11-06

Publications (1)

Publication Number	Publication Date
SI9300581A true SI9300581A (en)	1994-06-30

Family

ID=6472230

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SI9300581A SI9300581A (en)	1992-11-06	1993-11-05	Transdermal therapeutic system with estradiol as activ substance

Country Status (24)

Country	Link
US (1)	US5912008A (sh)
EP (1)	EP0716599B1 (sh)
JP (1)	JP3237016B2 (sh)
KR (1)	KR100306946B1 (sh)
AT (1)	ATE164516T1 (sh)
AU (1)	AU678408B2 (sh)
CA (1)	CA2147172C (sh)
CZ (1)	CZ286907B6 (sh)
DE (2)	DE4237453C1 (sh)
DK (1)	DK0716599T3 (sh)
ES (1)	ES2117152T3 (sh)
FI (1)	FI113339B (sh)
HR (1)	HRP931360B1 (sh)
HU (1)	HU221847B1 (sh)
IL (1)	IL107395A (sh)
MY (1)	MY118171A (sh)
NO (1)	NO311783B1 (sh)
NZ (1)	NZ257137A (sh)
PL (1)	PL174604B1 (sh)
SI (1)	SI9300581A (sh)
SK (1)	SK279911B6 (sh)
WO (1)	WO1994010984A1 (sh)
YU (1)	YU69693A (sh)
ZA (1)	ZA938257B (sh)

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US5906830A (en) *	1995-09-08	1999-05-25	Cygnus, Inc.	Supersaturated transdermal drug delivery systems, and methods for manufacturing the same
DE19600347A1 (de) *	1996-01-08	1997-07-10	Lohmann Therapie Syst Lts	Hauthaftende pharmazeutische Zubereitung, insbesondere TTS zur Abgabe von 17-beta-Estradiol an den menschlichen Organismus
DE19701949A1 (de) *	1997-01-13	1998-07-16	Jenapharm Gmbh	Transdermales therapeutisches System
US5968547A (en)	1997-02-24	1999-10-19	Euro-Celtique, S.A.	Method of providing sustained analgesia with buprenorphine
DE19827732A1 (de) *	1998-06-22	1999-12-23	Rottapharm Bv	Transdermales System vom Matrix-Typ zur Abgabe von Wirkstoffen mit einer hohen Abgaberate von Steroid-Hormonen und die Verwendung eines derartigen Systems zur Hormonersatztherapie
JP4399044B2 (ja) *	1998-10-14	2010-01-13	久光製薬株式会社	吸収促進剤及び該吸収促進剤を有してなる経皮吸収製剤
US6631186B1 (en) *	1999-04-09	2003-10-07	Sbc Technology Resources, Inc.	System and method for implementing and accessing call forwarding services
DE19925613A1 (de) *	1999-06-04	2000-12-07	Lohmann Therapie Syst Lts	Verbundlaminat und Verfahren zu seiner Herstellung
ITRM20060440A1 (it) *	2006-08-10	2008-02-11	Carmine Antropoli	Uso della nifedipina per il trattamento antirughe
US20100087768A1 (en) *	2008-10-02	2010-04-08	Forlano Paula	Transdermal drug delivery system for liquid active ingredient
DE102010026903A1 (de)	2010-07-12	2012-01-12	Amw Gmbh	Transdermales therapeutisches System mit Avocadoöl oder Palmöl als Hilfsstoff
WO2013006613A1 (en)	2011-07-05	2013-01-10	Novan, Inc.	Methods of manufacturing topical compositions and apparatus for same
BR112014000178A2 (pt) *	2011-07-05	2017-02-07	Novan Inc	composições tópicas
DE102012000369A1 (de)	2012-01-11	2013-07-11	Alfred E. Tiefenbacher (Gmbh & Co. Kg)	Transdermales therapeutisches System mit Cholinesterase-Hemmer
US9855211B2 (en)	2013-02-28	2018-01-02	Novan, Inc.	Topical compositions and methods of using the same
CA2954061C (en)	2014-07-11	2023-01-24	Novan, Inc.	Topical antiviral compositions and methods of using the same
US10322082B2 (en)	2014-07-11	2019-06-18	Novan, Inc.	Topical antiviral compositions and methods of using the same
EP3442502A4 (en)	2016-04-13	2019-11-06	Novan, Inc.	COMPOSITIONS, SYSTEMS, KITS AND METHODS FOR TREATING INFECTIONS
DE102017127433A1 (de)	2017-11-21	2019-05-23	Lts Lohmann Therapie-Systeme Ag	TTS auf Basis von klebenden Weichmacher-Polymer-Matrices

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1992
- 1992-11-06 DE DE4237453A patent/DE4237453C1/de not_active Revoked
1993
- 1993-10-21 MY MYPI93002178A patent/MY118171A/en unknown
- 1993-10-25 IL IL10739593A patent/IL107395A/xx not_active IP Right Cessation
- 1993-10-27 HU HU9501318A patent/HU221847B1/hu active IP Right Grant
- 1993-10-27 JP JP51165094A patent/JP3237016B2/ja not_active Expired - Lifetime
- 1993-10-27 PL PL93308532A patent/PL174604B1/pl unknown
- 1993-10-27 CA CA002147172A patent/CA2147172C/en not_active Expired - Lifetime
- 1993-10-27 AU AU53386/94A patent/AU678408B2/en not_active Expired
- 1993-10-27 DK DK93923559T patent/DK0716599T3/da active
- 1993-10-27 DE DE59308360T patent/DE59308360D1/de not_active Expired - Lifetime
- 1993-10-27 WO PCT/EP1993/002971 patent/WO1994010984A1/de active IP Right Grant
- 1993-10-27 NZ NZ257137A patent/NZ257137A/en not_active IP Right Cessation
- 1993-10-27 AT AT93923559T patent/ATE164516T1/de active
- 1993-10-27 CZ CZ19951162A patent/CZ286907B6/cs not_active IP Right Cessation
- 1993-10-27 EP EP93923559A patent/EP0716599B1/de not_active Expired - Lifetime
- 1993-10-27 ES ES93923559T patent/ES2117152T3/es not_active Expired - Lifetime
- 1993-10-27 SK SK580-95A patent/SK279911B6/sk not_active IP Right Cessation
- 1993-10-27 KR KR1019950701791A patent/KR100306946B1/ko not_active Expired - Lifetime
- 1993-11-03 YU YU69693A patent/YU69693A/sh unknown
- 1993-11-04 HR HRP4237453.7A patent/HRP931360B1/xx not_active IP Right Cessation
- 1993-11-05 ZA ZA938257A patent/ZA938257B/xx unknown
- 1993-11-05 SI SI9300581A patent/SI9300581A/sl unknown
1995
- 1995-05-03 FI FI952115A patent/FI113339B/fi not_active IP Right Cessation
- 1995-05-05 NO NO19951765A patent/NO311783B1/no not_active IP Right Cessation
1997
- 1997-06-16 US US08/876,427 patent/US5912008A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
SK279911B6 (sk)	1999-05-07
NO311783B1 (no)	2002-01-28
KR100306946B1 (ko)	2002-04-24
PL308532A1 (en)	1995-08-21
AU678408B2 (en)	1997-05-29
IL107395A (en)	1997-08-14
US5912008A (en)	1999-06-15
JP3237016B2 (ja)	2001-12-10
JPH08502987A (ja)	1996-04-02
IL107395A0 (en)	1994-01-25
WO1994010984A1 (de)	1994-05-26
DK0716599T3 (da)	1999-01-11
SK58095A3 (en)	1995-11-08
HU9501318D0 (en)	1995-06-28
CA2147172A1 (en)	1994-05-26
DE4237453C1 (sh)	1993-08-19
ES2117152T3 (es)	1998-08-01
EP0716599A1 (de)	1996-06-19
ZA938257B (en)	1994-06-08
MY118171A (en)	2004-09-30
CZ286907B6 (en)	2000-08-16
FI952115L (fi)	1995-05-03
NZ257137A (en)	1996-09-25
AU5338694A (en)	1994-06-08
HRP931360B1 (en)	1999-12-31
YU69693A (sh)	1997-07-31
DE59308360D1 (de)	1998-05-07
EP0716599B1 (de)	1998-04-01
NO951765D0 (no)	1995-05-05
HRP931360A2 (en)	1995-02-28
ATE164516T1 (de)	1998-04-15
NO951765L (no)	1995-05-05
KR950703940A (ko)	1995-11-17
FI952115A0 (fi)	1995-05-03
FI113339B (fi)	2004-04-15
HU221847B1 (hu)	2003-02-28
CA2147172C (en)	2003-12-23
PL174604B1 (pl)	1998-08-31
CZ116295A3 (en)	1995-12-13
HUT71681A (en)	1996-01-29

Publication	Publication Date	Title
SI9300581A (en)	1994-06-30	Transdermal therapeutic system with estradiol as activ substance
AU649732B2 (en)	1994-06-02	Transdermal device
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CA2229184C (en)	2001-07-24	Supersaturated transdermal drug delivery systems, and methods for manufacturing the same
KR101171814B1 (ko)	2012-08-13	펜타닐 함유 점착성 제제
PT697860E (pt)	2001-03-30	Sistema teraputico transdermico que contem estradiol
PL163297B1 (pl)	1994-03-31	Sposób wytwarzania poprzezskórnego ukladu terapeutycznego PL PL PL
SI9300387A (en)	1994-03-31	Transdermale therapeutic system containing active 17-beta estradiol (dry acid)
KR100473677B1 (ko)	2005-03-07	물리적 특성이 향상된 폴리아크릴레이트 매트릭스를 구비한 경피 또는 국소 플래스터 시스템
CZ289313B6 (cs)	2001-12-12	Transdermální terapeutický systém ve formě náplasti
PL201222B1 (pl)	2009-03-31	Preparat transdermalny lazoksyfenu, urządzenie do podawania lazoksyfenu, oraz zastosowanie lazoksyfenu
US20090220580A1 (en)	2009-09-03	Percutaneous Absorption Formulation
US6733785B1 (en)	2004-05-11	Moisture-sensitive preparation of percutaneous absorption type
SI9300589A (en)	1994-06-30	Transdermal therapeutic system for administration of fisostigmin and procedure for its preparation
US5827245A (en)	1998-10-27	Transdermal therapeutic system comprising the active subtance 17-β-Estradiol (Anhydrous)
JP3242324B2 (ja)	2001-12-25	ニトログリセリン経皮吸収型製剤
WO1993000057A1 (en)	1993-01-07	Transdermal nicotine absorption dosage unit and process
PL180943B1 (pl)	2001-05-31	Transdermalny system terapeutyczny zawierający estradiol i sposób wytwarzania tego systemu terapeutycznego