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SG11202100727VA - Boronic acid derivatives - Google Patents

Boronic acid derivatives

Info

Publication number
SG11202100727VA
SG11202100727VA SG11202100727VA SG11202100727VA SG11202100727VA SG 11202100727V A SG11202100727V A SG 11202100727VA SG 11202100727V A SG11202100727V A SG 11202100727VA SG 11202100727V A SG11202100727V A SG 11202100727VA SG 11202100727V A SG11202100727V A SG 11202100727VA
Authority
SG
Singapore
Prior art keywords
acid derivatives
boronic acid
boronic
derivatives
acid
Prior art date
Application number
SG11202100727VA
Inventor
Markus Klein
Oliver Schadt
Philipp Haselmayer
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of SG11202100727VA publication Critical patent/SG11202100727VA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
SG11202100727VA 2018-07-26 2019-07-23 Boronic acid derivatives SG11202100727VA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP18185848 2018-07-26
PCT/EP2019/069744 WO2020020858A1 (en) 2018-07-26 2019-07-23 Boronic acid derivatives

Publications (1)

Publication Number Publication Date
SG11202100727VA true SG11202100727VA (en) 2021-02-25

Family

ID=63077806

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11202100727VA SG11202100727VA (en) 2018-07-26 2019-07-23 Boronic acid derivatives

Country Status (15)

Country Link
US (1) US20210317145A1 (en)
EP (1) EP3826723B1 (en)
JP (1) JP2021531310A (en)
KR (1) KR20210038590A (en)
CN (1) CN112469480A (en)
AU (1) AU2019310779A1 (en)
BR (1) BR112021001359A2 (en)
CA (1) CA3107377A1 (en)
DK (1) DK3826723T3 (en)
ES (1) ES2968443T3 (en)
IL (1) IL280376B2 (en)
MX (1) MX2021000214A (en)
SG (1) SG11202100727VA (en)
TW (1) TW202019436A (en)
WO (1) WO2020020858A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114075227B (en) * 2020-08-19 2023-07-04 北京嵩润医药科技有限责任公司 Pyrazole boric acid compound, pharmaceutical composition containing pyrazole boric acid compound and application of pyrazole boric acid compound and pharmaceutical composition
TW202237143A (en) * 2020-12-10 2022-10-01 南韓商Lg化學股份有限公司 Boronic acid compounds
WO2023061445A1 (en) * 2021-10-14 2023-04-20 首药控股(北京)股份有限公司 Boronic acid derivative
WO2023107487A1 (en) * 2021-12-06 2023-06-15 Pretzel Therapeutics, Inc. Lonp1 inhibitor compounds, uses and methods

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103497232A (en) 2008-06-17 2014-01-08 米伦纽姆医药公司 Boronate ester compounds and pharmaceutical compositions thereof
HK1206261A1 (en) 2011-12-22 2016-01-08 Ares Trading S.A. Alpha-amino boronic acid derivatives, selective immunoproteasome inhibitors
CA2866135A1 (en) 2012-03-02 2014-09-06 Dr. Reddy's Laboratories Limited Pharmaceutical compositions comprising boronic acid compounds
SG11201702620SA (en) * 2014-10-01 2017-04-27 Merck Patent Gmbh Boronic acid derivatives
KR20170066506A (en) * 2014-10-01 2017-06-14 메르크 파텐트 게엠베하 Boronic acid derivatives
WO2016050359A1 (en) 2014-10-01 2016-04-07 Merck Patent Gmbh Boronic acid derivatives
US10669289B2 (en) * 2014-10-01 2020-06-02 Merck Patent Gmbh Boronic acid derivatives
CN110540547A (en) * 2018-05-28 2019-12-06 秦艳茹 Synthesis and application of peptide borate compound

Also Published As

Publication number Publication date
ES2968443T3 (en) 2024-05-09
EP3826723A1 (en) 2021-06-02
CA3107377A1 (en) 2020-01-30
WO2020020858A1 (en) 2020-01-30
CN112469480A (en) 2021-03-09
JP2021531310A (en) 2021-11-18
KR20210038590A (en) 2021-04-07
IL280376B1 (en) 2024-04-01
BR112021001359A2 (en) 2021-04-20
DK3826723T3 (en) 2024-01-15
AU2019310779A1 (en) 2021-03-18
US20210317145A1 (en) 2021-10-14
MX2021000214A (en) 2021-03-31
IL280376A (en) 2021-03-01
IL280376B2 (en) 2024-08-01
EP3826723B1 (en) 2023-10-18
TW202019436A (en) 2020-06-01

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