[go: up one dir, main page]

SE8207092D0 - Forfarande for framstellning av optiskt aktiva penemer - Google Patents

Forfarande for framstellning av optiskt aktiva penemer

Info

Publication number
SE8207092D0
SE8207092D0 SE8207092A SE8207092A SE8207092D0 SE 8207092 D0 SE8207092 D0 SE 8207092D0 SE 8207092 A SE8207092 A SE 8207092A SE 8207092 A SE8207092 A SE 8207092A SE 8207092 D0 SE8207092 D0 SE 8207092D0
Authority
SE
Sweden
Prior art keywords
procedure
optically active
unsubstituted
hydrogen
formula
Prior art date
Application number
SE8207092A
Other languages
English (en)
Other versions
SE458684B (sv
SE8207092L (sv
Inventor
M Alpegiani
C Battistini
A Bedeschi
G Franceschi
M Foglio
F Zarini
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of SE8207092D0 publication Critical patent/SE8207092D0/sv
Publication of SE8207092L publication Critical patent/SE8207092L/sv
Publication of SE458684B publication Critical patent/SE458684B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/18Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804Compounds having Si-O-C linkages
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/568Four-membered rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
SE8207092A 1981-12-11 1982-12-10 Foerfarande foer framstaellning av azetidin-2-oner vilka anvaends som mellanprodukter foer framstaellning av penemer SE458684B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8137513 1981-12-11

Publications (3)

Publication Number Publication Date
SE8207092D0 true SE8207092D0 (sv) 1982-12-10
SE8207092L SE8207092L (sv) 1983-06-12
SE458684B SE458684B (sv) 1989-04-24

Family

ID=10526562

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8207092A SE458684B (sv) 1981-12-11 1982-12-10 Foerfarande foer framstaellning av azetidin-2-oner vilka anvaends som mellanprodukter foer framstaellning av penemer

Country Status (21)

Country Link
US (1) US4508649A (sv)
JP (2) JPS58126888A (sv)
AT (1) AT379399B (sv)
AU (1) AU556854B2 (sv)
BE (1) BE895322A (sv)
CA (1) CA1215705A (sv)
CH (1) CH655504B (sv)
DE (1) DE3245270C2 (sv)
DK (1) DK160311C (sv)
FI (1) FI76347C (sv)
FR (2) FR2518098B1 (sv)
GB (1) GB2111496B (sv)
GR (1) GR77078B (sv)
HU (1) HU187807B (sv)
IE (1) IE54513B1 (sv)
IL (1) IL67434A (sv)
IT (1) IT1206106B (sv)
NL (2) NL8204720A (sv)
SE (1) SE458684B (sv)
SU (1) SU1389680A3 (sv)
ZA (1) ZA829063B (sv)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO831160L (no) * 1982-04-08 1983-10-10 Erba Farmitalia Fremstilling av substituerte penem-derivater
GB8300295D0 (en) * 1983-01-06 1983-02-09 Erba Farmitalia Penem esters
GB8321677D0 (en) * 1983-08-11 1983-09-14 Erba Farmitalia Preparation of penems
JPS62501556A (ja) * 1984-07-13 1987-06-25 メルシャン株式会社 新規2↓−オキソアゼチジン類、その製造方法および応用
GB8713515D0 (en) * 1987-06-10 1987-07-15 Erba Farmitalia Methoxymethyl compounds
GB8818789D0 (en) * 1988-08-08 1988-09-07 Erba Carlo Spa Crystalline(5r 6s)-2-carbamoyloxymethyl-6-((1r)-hydroxyethyl)-2-penem-carboxylic acid & pharmaceutical formulation
EP0371875B1 (en) * 1988-11-29 1994-12-28 Takasago International Corporation Process for preparing 4-acetoxyazetidinones
US5204460A (en) * 1988-11-29 1993-04-20 Takasago International Corporation Ruthenium catalyzed process for preparing 4-acetoxyazetidinones
EP0597401A3 (en) * 1992-11-11 1995-07-26 Takeda Chemical Industries Ltd Preparation of penemes.

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4348320A (en) * 1976-11-19 1982-09-07 Merck & Co., Inc. Substituted azetidiones
EP0042026B1 (de) * 1978-02-02 1986-01-08 Ciba-Geigy Ag 3,4-Disubstituierte Azetidin-2-onverbindungen und Verfahren zu ihrer Herstellung
AT365594B (de) * 1978-11-24 1982-01-25 Erba Farmitalia Verfahren zur herstellung von neuen 7-oxo-4-thia1-aza-bicyclo-(3,2,0)heptanderivaten
EP0013067A1 (en) * 1978-12-22 1980-07-09 Beecham Group Plc Bicyclic beta-lactam antibacterial agents, their use in pharmaceutical compositions, processes for their preparation and intermediates for use in such processes
GB2037277B (en) * 1978-12-22 1983-05-05 Beecham Group Ltd -lactam antibacterial agents their use in pharmaceutical compositions processes for their preparation and intermediates for use in such processes
AT368506B (de) * 1979-02-24 1982-10-25 Erba Farmitalia Verfahren zur herstellung von neuen penemcarbonsaeuren und deren salzen
US4269771A (en) * 1979-04-06 1981-05-26 Farmitalia Carlo Erba Total synthesis of 7-oxo-4-thia-1-azabicyclo-[3,2,0]-heptane-2-carboxyl derivatives useful as β-lactamase inhibitors and antibacterial agents
JPS55153789A (en) * 1979-04-11 1980-11-29 Sankyo Co Ltd Penem-3-carboxylic acid derivative and its preparation
US4482565A (en) * 1980-02-22 1984-11-13 Farmitalia Carlo Erba S.P.A. β-Lactam-containing antibacterial agents and β-lactamase inhibitors
GB2079744A (en) * 1980-07-04 1982-01-27 Erba Farmitalia 6-Alkyl-2-functionalized penems

Also Published As

Publication number Publication date
FR2518098B1 (fr) 1986-02-21
GB2111496B (en) 1985-05-09
AT379399B (de) 1985-12-27
FR2518098A1 (fr) 1983-06-17
HU187807B (en) 1986-02-28
FI76347C (sv) 1988-10-10
ATA443582A (de) 1985-05-15
NL8204720A (nl) 1983-07-01
DE3245270A1 (de) 1983-06-23
IT1206106B (it) 1989-04-14
FI824192A0 (fi) 1982-12-07
JPS61178987A (ja) 1986-08-11
NL8600460A (nl) 1986-06-02
DE3245270C2 (de) 1997-05-15
IL67434A (en) 1986-07-31
FI76347B (fi) 1988-06-30
JPS58126888A (ja) 1983-07-28
SE458684B (sv) 1989-04-24
GR77078B (sv) 1984-09-06
DK551182A (da) 1983-06-12
BE895322A (fr) 1983-06-10
SE8207092L (sv) 1983-06-12
GB2111496A (en) 1983-07-06
CH655504B (sv) 1986-04-30
AU9115682A (en) 1983-06-16
IE822917L (en) 1983-06-11
SU1389680A3 (ru) 1988-04-15
DK160311C (da) 1991-07-29
ZA829063B (en) 1983-09-28
AU556854B2 (en) 1986-11-20
JPH045033B2 (sv) 1992-01-30
DK160311B (da) 1991-02-25
IT8224650A0 (it) 1982-12-09
FR2567888B1 (fr) 1987-04-17
FI824192L (fi) 1983-06-12
IE54513B1 (en) 1989-11-08
CA1215705A (en) 1986-12-23
US4508649A (en) 1985-04-02
FR2567888A1 (fr) 1986-01-24
IL67434A0 (en) 1983-05-15
JPH0146516B2 (sv) 1989-10-09

Similar Documents

Publication Publication Date Title
ATE33838T1 (de) Thiazolidinderivate, ihre herstellung und diese enthaltende zusammensetzungen.
DE3167757D1 (en) Dibenz(b,f)(1,4)oxazepine derivatives, process for preparing the same, and pharmaceutical compositions comprising the same
NO163566C (no) 1,5-benzothiazepinderivater som er anvendelige som utgangsmaterialer ved fremstilling av nye, terapeutisk aktive 8-klor-1,5-benzothiazepinderivater.
NO943093L (no) Fremgangsmåte for fremstilling av clavulansyre
CA2043071A1 (en) Heterocyclic compounds
NZ194284A (en) Piperidine and pyrrolidine derivatives and pharmaceutical compositions
HU906402D0 (en) Process for producing tricyclic carbapeneme derivatives an pharmaceutical preparatives containing these compounds as active substance
IE831203L (en) Penicillanic acid dioxide prodrug
ATE224T1 (de) 1,2-dihydro-chinolin-2-on-derivate, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel.
FI933903A0 (fi) Substituerade cyklohexanderivat, foerfarande foer framstaellning daerav och anvaendning av foereningar foer behandling av sjukdomar
DE69022294D1 (de) N-Heteroaryl-purin-6-amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel.
SE8207092L (sv) Forfarande for framstellning av optiskt aktiva penemer
DE69115526D1 (de) 2,4-Pyrimidindionderivate und diese enthaltende Arzneimittel
ATE50448T1 (de) 5-alkyl-1-phenyl-2-piperazinoalkylpyrazolin-3-o - verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel.
ATE3149T1 (de) Isatinderivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen.
SE7703000L (sv) Forfarande for framstellning av karbostyrilderivat
AU574198B2 (en) Penem derivatives
ATE37368T1 (de) Benzothiazolon-derivate, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische zusammensetzungen.
AU658175B2 (en) Use of 2-iminothiazolidin-4-one derivatives as novel pharmaceutical active ingredients
ATE14120T1 (de) Sulfimine, deren salze und deren herstellung sowie diese verbindungen enthaltende arzneimittel.
CA2053705A1 (en) Piperazine derivatives
ATE5408T1 (de) Cephalosporine, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel.
SE7910387L (sv) 7alfa-metoxicefalosporinderivat och forfarande for framstellning derav
FI824479L (fi) Foerfarande och mellanprodukt foer framstaellning av farmakologiskt verksamma (1,2)-anellerade 1,4-bensodiazepinfoereningar
ATE81126T1 (de) Benzopyrrolidinon-derivate, verfahren zu ihrer herstellung und arzneimittel, die sie enthalten.

Legal Events

Date Code Title Description
NAL Patent in force

Ref document number: 8207092-1

Format of ref document f/p: F

NUG Patent has lapsed