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SE449995B - 6-perhalogenalkylsulfonyloxipenicillansyraderivat samt forfarande for framstellning derav - Google Patents

6-perhalogenalkylsulfonyloxipenicillansyraderivat samt forfarande for framstellning derav

Info

Publication number
SE449995B
SE449995B SE8003676A SE8003676A SE449995B SE 449995 B SE449995 B SE 449995B SE 8003676 A SE8003676 A SE 8003676A SE 8003676 A SE8003676 A SE 8003676A SE 449995 B SE449995 B SE 449995B
Authority
SE
Sweden
Prior art keywords
acid
ester
group
formula
compound
Prior art date
Application number
SE8003676A
Other languages
English (en)
Swedish (sv)
Other versions
SE8003676L (sv
Inventor
J E G Kemp
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of SE8003676L publication Critical patent/SE8003676L/xx
Publication of SE449995B publication Critical patent/SE449995B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32Esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04Preparation
    • C07D499/10Modification of an amino radical directly attached in position 6
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SE8003676A 1979-05-19 1980-05-16 6-perhalogenalkylsulfonyloxipenicillansyraderivat samt forfarande for framstellning derav SE449995B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7917505 1979-05-19

Publications (2)

Publication Number Publication Date
SE8003676L SE8003676L (sv) 1980-11-20
SE449995B true SE449995B (sv) 1987-06-01

Family

ID=10505288

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8003676A SE449995B (sv) 1979-05-19 1980-05-16 6-perhalogenalkylsulfonyloxipenicillansyraderivat samt forfarande for framstellning derav

Country Status (28)

Country Link
US (1) US4356122A (nl)
JP (1) JPS5941994B2 (nl)
KR (1) KR840000079B1 (nl)
AR (1) AR225038A1 (nl)
AT (1) AT366694B (nl)
AU (1) AU517488B2 (nl)
BE (1) BE883319A (nl)
CA (1) CA1140916A (nl)
CH (1) CH650262A5 (nl)
CS (1) CS214756B2 (nl)
DD (1) DD151310A5 (nl)
DE (1) DE3018847C2 (nl)
DK (1) DK155180A (nl)
ES (1) ES8105737A1 (nl)
FI (1) FI71562C (nl)
FR (1) FR2457293A1 (nl)
GR (1) GR68461B (nl)
IE (1) IE49804B1 (nl)
IL (1) IL60097A (nl)
IT (1) IT1140946B (nl)
LU (1) LU82458A1 (nl)
NL (1) NL180937C (nl)
NO (1) NO801473L (nl)
PH (1) PH15033A (nl)
PL (1) PL224188A1 (nl)
PT (1) PT71253A (nl)
SE (1) SE449995B (nl)
ZA (1) ZA802908B (nl)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA803742B (en) * 1979-07-02 1981-06-24 Beecham Group Ltd Penicillanic acid derivatives, their preparation and use
JPS6034969A (ja) * 1983-08-08 1985-02-22 Toyama Chem Co Ltd 新規なペニシラン酸誘導体およびその塩類
AU2018240467B2 (en) * 2017-03-23 2022-09-15 Neubase Therapeutics, Inc. Peptide nucleic acid (PNA) monomers with an orthogonally protected ester moiety

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5749555B2 (nl) * 1973-04-04 1982-10-22
US4282149A (en) * 1977-03-21 1981-08-04 Massachusetts Institute Of Technology Carbon and oxygen analogs of penicillin
US4265882A (en) * 1977-10-03 1981-05-05 Massachusetts Institute Of Technology Sulphur analogs of penicillins having a nucleophile substituted in the 6 and 7 position, respectively

Also Published As

Publication number Publication date
IT1140946B (it) 1986-10-10
DE3018847A1 (de) 1980-12-11
NL180937C (nl) 1987-05-18
FI71562B (fi) 1986-10-10
KR830002769A (ko) 1983-05-30
CH650262A5 (de) 1985-07-15
PT71253A (en) 1980-06-01
AU5846880A (en) 1980-11-27
IL60097A (en) 1983-02-23
DK155180A (da) 1980-11-20
ZA802908B (en) 1981-05-27
KR840000079B1 (ko) 1984-02-08
LU82458A1 (fr) 1980-10-08
ES491612A0 (es) 1981-05-16
AU517488B2 (en) 1981-08-06
FI801581A (fi) 1980-11-20
GR68461B (nl) 1981-12-30
IT8022104A0 (it) 1980-05-16
FR2457293B1 (nl) 1983-05-20
PL224188A1 (nl) 1981-02-13
IE801024L (en) 1980-11-19
IE49804B1 (en) 1985-12-25
FI71562C (fi) 1987-01-19
JPS5941994B2 (ja) 1984-10-11
JPS55157588A (en) 1980-12-08
DE3018847C2 (de) 1982-09-30
CA1140916A (en) 1983-02-08
BE883319A (fr) 1980-11-14
ATA259780A (de) 1981-09-15
PH15033A (en) 1982-05-20
AT366694B (de) 1982-04-26
NO801473L (no) 1980-11-20
NL8002843A (nl) 1980-11-21
FR2457293A1 (fr) 1980-12-19
CS214756B2 (en) 1982-05-28
ES8105737A1 (es) 1981-05-16
NL180937B (nl) 1986-12-16
SE8003676L (sv) 1980-11-20
DD151310A5 (de) 1981-10-14
AR225038A1 (es) 1982-02-15
US4356122A (en) 1982-10-26
IL60097A0 (en) 1980-07-31

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