RU2004121986A - Промежуточные соединения для получения ингибиторов гликогенфосфорилазы - Google Patents
Промежуточные соединения для получения ингибиторов гликогенфосфорилазы Download PDFInfo
- Publication number
- RU2004121986A RU2004121986A RU2004121986/04A RU2004121986A RU2004121986A RU 2004121986 A RU2004121986 A RU 2004121986A RU 2004121986/04 A RU2004121986/04 A RU 2004121986/04A RU 2004121986 A RU2004121986 A RU 2004121986A RU 2004121986 A RU2004121986 A RU 2004121986A
- Authority
- RU
- Russia
- Prior art keywords
- preparation
- intermediate compounds
- glycogen phosphorylase
- phosphorylase inhibitors
- inhibitors
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title claims 3
- 102000007390 Glycogen Phosphorylase Human genes 0.000 title 1
- 108010046163 Glycogen Phosphorylase Proteins 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- PIWZAEFTGNOGME-XGBAPZKQSA-N CC1(C)O[C@@H](CN(C2)C([C@@H](C(Cc3ccccc3)NC(c3cc4cc(Cl)ccc4[nH]3)=O)O)=O)[C@@H]2O1 Chemical compound CC1(C)O[C@@H](CN(C2)C([C@@H](C(Cc3ccccc3)NC(c3cc4cc(Cl)ccc4[nH]3)=O)O)=O)[C@@H]2O1 PIWZAEFTGNOGME-XGBAPZKQSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Claims (2)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US34964702P | 2002-01-18 | 2002-01-18 | |
US60/349,647 | 2002-01-18 |
Publications (1)
Publication Number | Publication Date |
---|---|
RU2004121986A true RU2004121986A (ru) | 2005-11-20 |
Family
ID=23373348
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU2004121986/04A RU2004121986A (ru) | 2002-01-18 | 2003-01-06 | Промежуточные соединения для получения ингибиторов гликогенфосфорилазы |
Country Status (16)
Country | Link |
---|---|
US (1) | US6696574B2 (ru) |
EP (1) | EP1470128A1 (ru) |
JP (1) | JP2005514460A (ru) |
KR (1) | KR20040072730A (ru) |
CN (1) | CN1592749A (ru) |
AU (1) | AU2003200853A1 (ru) |
BR (1) | BR0307006A (ru) |
CA (1) | CA2472205A1 (ru) |
HU (1) | HUP0500513A3 (ru) |
IL (1) | IL161507A0 (ru) |
MX (1) | MXPA04006937A (ru) |
PL (1) | PL371408A1 (ru) |
RU (1) | RU2004121986A (ru) |
TW (1) | TW200302220A (ru) |
WO (1) | WO2003059910A1 (ru) |
ZA (1) | ZA200402621B (ru) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20090298745A1 (en) * | 2004-12-02 | 2009-12-03 | Gerard Hugh Thomas | Treatment of Diabetes with Glycogen Phosphorylase Inhibitors |
PE20080251A1 (es) | 2006-05-04 | 2008-04-25 | Boehringer Ingelheim Int | Usos de inhibidores de dpp iv |
JP5959075B2 (ja) * | 2011-05-31 | 2016-08-02 | セラヴァンス バイオファーマ アール&ディー アイピー, エルエルシー | ネプリライシン阻害剤 |
CN103626845B (zh) * | 2013-09-30 | 2015-11-11 | 承德医学院 | 作为糖原磷酸化酶抑制剂的芳基并吡咯-2-甲酰胺二肽衍生物、其制备方法及医药用途 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2342471C (en) * | 1995-06-06 | 2002-10-29 | Judith L. Treadway | Heterocyclecarbonylmethyl amine intermediates |
CA2223625C (en) * | 1995-06-06 | 2003-06-03 | Pfizer Inc. | Substituted n-(indole-2-carbonyl-) amides and derivatives as glycogen phosphorylase inhibitors |
US6277877B1 (en) * | 2000-08-15 | 2001-08-21 | Pfizer, Inc. | Substituted n-(indole-2-carbonyl)glycinamides and derivates as glycogen phosphorylase inhibitors |
-
2003
- 2003-01-06 WO PCT/IB2003/000034 patent/WO2003059910A1/en not_active Application Discontinuation
- 2003-01-06 JP JP2003560013A patent/JP2005514460A/ja active Pending
- 2003-01-06 CN CNA038015455A patent/CN1592749A/zh active Pending
- 2003-01-06 HU HU0500513A patent/HUP0500513A3/hu unknown
- 2003-01-06 AU AU2003200853A patent/AU2003200853A1/en not_active Abandoned
- 2003-01-06 RU RU2004121986/04A patent/RU2004121986A/ru not_active Application Discontinuation
- 2003-01-06 EP EP03700024A patent/EP1470128A1/en not_active Withdrawn
- 2003-01-06 BR BR0307006-9A patent/BR0307006A/pt not_active Application Discontinuation
- 2003-01-06 IL IL16150703A patent/IL161507A0/xx unknown
- 2003-01-06 KR KR10-2004-7011084A patent/KR20040072730A/ko not_active Ceased
- 2003-01-06 PL PL03371408A patent/PL371408A1/xx not_active Application Discontinuation
- 2003-01-06 MX MXPA04006937A patent/MXPA04006937A/es unknown
- 2003-01-06 CA CA002472205A patent/CA2472205A1/en not_active Abandoned
- 2003-01-13 TW TW092100616A patent/TW200302220A/zh unknown
- 2003-01-16 US US10/345,661 patent/US6696574B2/en not_active Expired - Fee Related
-
2004
- 2004-04-02 ZA ZA200402621A patent/ZA200402621B/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP1470128A1 (en) | 2004-10-27 |
KR20040072730A (ko) | 2004-08-18 |
ZA200402621B (en) | 2005-05-27 |
BR0307006A (pt) | 2004-11-03 |
US20030187051A1 (en) | 2003-10-02 |
WO2003059910A1 (en) | 2003-07-24 |
HUP0500513A2 (hu) | 2005-11-28 |
AU2003200853A1 (en) | 2003-07-30 |
HUP0500513A3 (en) | 2006-07-28 |
IL161507A0 (en) | 2004-09-27 |
TW200302220A (en) | 2003-08-01 |
US6696574B2 (en) | 2004-02-24 |
JP2005514460A (ja) | 2005-05-19 |
PL371408A1 (en) | 2005-06-13 |
CA2472205A1 (en) | 2003-07-24 |
CN1592749A (zh) | 2005-03-09 |
MXPA04006937A (es) | 2004-12-06 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA94 | Acknowledgement of application withdrawn (non-payment of fees) |
Effective date: 20060517 |