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RS53129B - Novel compounds 951: a biphenyloxypropanoic acid as crth2 modulator and intermediates - Google Patents

Novel compounds 951: a biphenyloxypropanoic acid as crth2 modulator and intermediates

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Publication number
RS53129B
RS53129B RS20140008A RSP20140008A RS53129B RS 53129 B RS53129 B RS 53129B RS 20140008 A RS20140008 A RS 20140008A RS P20140008 A RSP20140008 A RS P20140008A RS 53129 B RS53129 B RS 53129B
Authority
RS
Serbia
Prior art keywords
acid
biphenyloxypropanoic
intermediates
novel compounds
crth2
Prior art date
Application number
RS20140008A
Other languages
Serbian (sr)
Inventor
Roger Victor Bonnert
Timothy Jon Luker
Anil Patel
Aaron Rigby
Original Assignee
Astrazeneca Ab.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39942682&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS53129(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab. filed Critical Astrazeneca Ab.
Publication of RS53129B publication Critical patent/RS53129B/en

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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
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Abstract

Jedinjenje formule (I):naznačeno time što je smeša (2S)-2-({3'-hloro-4'-[(2,2-dimetilpirolidin-1-il)karbonil]-5-fluorobifenil-2-il}oksi)propanske kiseline i (2R)-2-({3'-hloro-4'-[(2,2-dimetilpirolidin-1-il)karbonil]-5-fluorobifenil-2-il}oksi)propanske kiseline, ili njihovih farmaceutski prihvatljivih solvata ili farmaceutski prihvatljivih soli ili solvata farmaceutski prihvatljivih soli.Prijava sadrži još 19 patentnih zahteva.Compound of Formula (I): wherein the mixture is (2S) -2 - ({3'-chloro-4 '- [(2,2-dimethylpyrrolidin-1-yl) carbonyl] -5-fluorobiphenyl-2-yl} oxy) propanoic acid and (2R) -2 - ({3'-chloro-4 '- [(2,2-dimethylpyrrolidin-1-yl) carbonyl] -5-fluorobiphenyl-2-yl} oxy) propanoic acid, or of their pharmaceutically acceptable solvates or pharmaceutically acceptable salts or solvates of pharmaceutically acceptable salts. The application contains a further 19 claims.

RS20140008A 2007-07-05 2008-07-01 Novel compounds 951: a biphenyloxypropanoic acid as crth2 modulator and intermediates RS53129B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US94801207P 2007-07-05 2007-07-05
PCT/GB2008/050525 WO2009004379A1 (en) 2007-07-05 2008-07-01 Novel compounds 951: a biphenyloxypropanoic acid as crth2 modulator and intermediates

Publications (1)

Publication Number Publication Date
RS53129B true RS53129B (en) 2014-06-30

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RS20140008A RS53129B (en) 2007-07-05 2008-07-01 Novel compounds 951: a biphenyloxypropanoic acid as crth2 modulator and intermediates

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EP (1) EP2173730B1 (en)
JP (1) JP5368438B2 (en)
KR (1) KR20100039326A (en)
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AU (1) AU2008272690B2 (en)
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CA (1) CA2691615A1 (en)
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DK (1) DK2173730T3 (en)
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HR (1) HRP20140004T1 (en)
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NZ (1) NZ582192A (en)
PE (2) PE20121515A1 (en)
PL (1) PL2173730T3 (en)
PT (1) PT2173730E (en)
RS (1) RS53129B (en)
SA (1) SA08290406B1 (en)
SI (1) SI2173730T1 (en)
TW (1) TWI453017B (en)
UA (1) UA100983C2 (en)
UY (1) UY31208A1 (en)
WO (1) WO2009004379A1 (en)
ZA (1) ZA200909226B (en)

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