PT98645A - Processo para a preparacao de 3-(1,2-benzisoxazol-3-il-)-4-piridinaminas e seus derivados - Google Patents

Processo para a preparacao de 3-(1,2-benzisoxazol-3-il-)-4-piridinaminas e seus derivados

Info

Publication number: PT98645A
Authority: PT; Portugal
Prior art keywords: pyridinamines; benzisoxazol; hydrogen; derivatives; loweralkyl
Prior art date: 1990-08-13

Application number

PT98645A

Other languages

English (en)

Other versions

PT98645B (pt

Inventor

Joseph Thomas Klein

Richard C Effland

Original Assignee

Hoechst Roussel Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-08-13

Filing date

1991-08-12

Publication date

1992-06-30

1991-08-12 Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma

1992-06-30 Publication of PT98645A publication Critical patent/PT98645A/pt

1999-01-29 Publication of PT98645B publication Critical patent/PT98645B/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

PT98645A 1990-08-13 1991-08-12 Processo para a preparacao de 3-(1,2-benzisoxazol-3-il-)-4-piridinaminas e seus derivados PT98645B (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US07/566,932 US5055476A (en)	1990-08-13	1990-08-13	3-(1,2-benzisoxazol-3-yl)-4-pyridinamines and derivatives

Publications (2)

Publication Number	Publication Date
PT98645A true PT98645A (pt)	1992-06-30
PT98645B PT98645B (pt)	1999-01-29

Family

ID=24265033

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT98645A PT98645B (pt)	1990-08-13	1991-08-12	Processo para a preparacao de 3-(1,2-benzisoxazol-3-il-)-4-piridinaminas e seus derivados

Country Status (24)

Country	Link
US (1)	US5055476A (pt)
EP (1)	EP0471297B1 (pt)
JP (1)	JP3057829B2 (pt)
KR (1)	KR100191386B1 (pt)
AT (1)	ATE130004T1 (pt)
AU (1)	AU633791B2 (pt)
CA (1)	CA2048959C (pt)
CZ (1)	CZ280568B6 (pt)
DE (1)	DE69114405T2 (pt)
DK (1)	DK0471297T3 (pt)
ES (1)	ES2079531T3 (pt)
FI (1)	FI103970B1 (pt)
GR (1)	GR3018184T3 (pt)
HU (1)	HU213201B (pt)
IE (1)	IE70597B1 (pt)
IL (1)	IL99166A (pt)
MX (1)	MX9100639A (pt)
NO (1)	NO179519C (pt)
NZ (1)	NZ239326A (pt)
PT (1)	PT98645B (pt)
RU (1)	RU2012561C1 (pt)
TW (1)	TW202446B (pt)
YU (1)	YU140991A (pt)
ZA (1)	ZA916342B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5308826A (en) *	1993-04-22	1994-05-03	Zeneca Limited	Herbicidal 4-substituted pyridyl-3-carbinols
US5595958A (en) *	1994-05-02	1997-01-21	Zeneca Limited	3-substituted pyridine compounds and derivatives thereof
WO1995029898A1 (en) *	1994-05-02	1995-11-09	Zeneca Limited	Herbicidal hydroxybenzyl-substituted heteroaryl compounds and derivatives thereof
KR20150144817A (ko)	2011-06-10	2015-12-28	메르크 파텐트 게엠베하	Btk 억제 활성을 갖는 피리미딘 및 피리딘 화합물의 조성물 및 제조방법
RU2626650C2 (ru) *	2015-08-31	2017-07-31	Федеральное государственное бюджетное образовательное учреждение высшего образования "Пермский государственный национальный исследовательский университет"	2-Арил-2,4-дигидрокси-2,5-дигидро-3-гетерил-5-оксо-1Н-пиррол-1-ил-4-метилбелзолсульфаниламиды, обладающие анальгетической активностью
EP4429465A1 (en)	2021-11-10	2024-09-18	Symrise AG	Compositions comprising trpm8 agonistic cooling agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4355037A (en) *	1981-11-12	1982-10-19	Hoechst-Roussel Pharmaceuticals	3-(4-Piperidyl)-1,2-benzisoxales
IL66866A (en) *	1982-04-09	1987-08-31	Hoechst Roussel Pharma	1-(3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl)-4-(substituted)-piperazines and-piperidines,a process for the preparation thereof,and pharmaceutical compositions containing them
CA1335289C (en) *	1987-10-26	1995-04-18	Fujio Antoku	Piperidinyl benzisoxazole derivatives, their production and pharmaceutical use
MY107955A (en) *	1990-07-27	1996-07-15	Ici Plc	Fungicides.

1990
- 1990-08-13 US US07/566,932 patent/US5055476A/en not_active Expired - Fee Related
1991
- 1991-08-03 TW TW080106082A patent/TW202446B/zh active
- 1991-08-08 EP EP91113335A patent/EP0471297B1/en not_active Expired - Lifetime
- 1991-08-08 DE DE69114405T patent/DE69114405T2/de not_active Expired - Fee Related
- 1991-08-08 DK DK91113335.3T patent/DK0471297T3/da active
- 1991-08-08 ES ES91113335T patent/ES2079531T3/es not_active Expired - Lifetime
- 1991-08-08 AT AT91113335T patent/ATE130004T1/de not_active IP Right Cessation
- 1991-08-09 FI FI913800A patent/FI103970B1/fi active
- 1991-08-09 NZ NZ239326A patent/NZ239326A/en unknown
- 1991-08-12 MX MX9100639A patent/MX9100639A/es not_active IP Right Cessation
- 1991-08-12 IE IE285191A patent/IE70597B1/en not_active IP Right Cessation
- 1991-08-12 JP JP3201713A patent/JP3057829B2/ja not_active Expired - Fee Related
- 1991-08-12 CZ CS912489A patent/CZ280568B6/cs not_active IP Right Cessation
- 1991-08-12 PT PT98645A patent/PT98645B/pt not_active IP Right Cessation
- 1991-08-12 CA CA002048959A patent/CA2048959C/en not_active Expired - Fee Related
- 1991-08-12 AU AU81765/91A patent/AU633791B2/en not_active Ceased
- 1991-08-12 RU SU915001260A patent/RU2012561C1/ru active
- 1991-08-12 ZA ZA916342A patent/ZA916342B/xx unknown
- 1991-08-12 IL IL9916691A patent/IL99166A/en not_active IP Right Cessation
- 1991-08-12 NO NO913142A patent/NO179519C/no unknown
- 1991-08-12 HU HU912673A patent/HU213201B/hu not_active IP Right Cessation
- 1991-08-13 KR KR1019910013939A patent/KR100191386B1/ko not_active IP Right Cessation
- 1991-08-14 YU YU140991A patent/YU140991A/sh unknown
1995
- 1995-11-22 GR GR950403309T patent/GR3018184T3/el unknown

Also Published As

Publication number	Publication date
MX9100639A (es)	1992-04-01
JP3057829B2 (ja)	2000-07-04
IE70597B1 (en)	1996-12-11
FI103970B (fi)	1999-10-29
HU213201B (en)	1997-03-28
ES2079531T3 (es)	1996-01-16
DE69114405T2 (de)	1996-05-02
KR100191386B1 (ko)	1999-06-15
NO179519B (no)	1996-07-15
IL99166A0 (en)	1992-07-15
TW202446B (pt)	1993-03-21
CA2048959C (en)	2003-07-29
AU633791B2 (en)	1993-02-04
CA2048959A1 (en)	1992-02-14
NO913142D0 (no)	1991-08-12
CS248991A3 (en)	1992-03-18
NO913142L (no)	1992-02-14
FI913800A (fi)	1992-02-14
HUT61755A (en)	1993-03-01
JPH05112562A (ja)	1993-05-07
ZA916342B (en)	1992-04-29
US5055476A (en)	1991-10-08
NZ239326A (en)	1994-04-27
NO179519C (no)	1996-10-23
IL99166A (en)	1995-12-08
DK0471297T3 (da)	1996-03-04
PT98645B (pt)	1999-01-29
EP0471297A1 (en)	1992-02-19
CZ280568B6 (cs)	1996-02-14
FI103970B1 (fi)	1999-10-29
RU2012561C1 (ru)	1994-05-15
FI913800A0 (fi)	1991-08-09
YU140991A (sh)	1995-01-31
KR920004383A (ko)	1992-03-27
GR3018184T3 (en)	1996-02-29
DE69114405D1 (de)	1995-12-14
IE912851A1 (en)	1992-02-26
ATE130004T1 (de)	1995-11-15
EP0471297B1 (en)	1995-11-08
HU912673D0 (en)	1992-01-28
AU8176591A (en)	1992-02-20

Publication	Publication Date	Title
GR3030798T3 (en)	1999-11-30	2-(Piperidin-4-yl, pyridin-4-yl and tetrahydropyridin-4-yl)benzofuran-7-ol and carbamate derivatives, their preparation and their use as acetylcholinesterase inhibitors.
PT98645A (pt)	1992-06-30	Processo para a preparacao de 3-(1,2-benzisoxazol-3-il-)-4-piridinaminas e seus derivados
PT92234A (pt)	1990-05-31	Processo para a preparacao de 1,2,3,4-tetraidro-1,9-acridinodiaminas
AU640590B2 (en)	1993-08-26	3-(1h-indazol-3-yl)-4-pyridinamines
BR9200475A (pt)	1992-10-20	Composto e processo para a sua preparacao,composicao farmaceutica e uso do dito composto
ES2079530T3 (es)	1996-01-16	1-(piridinilalquil)-1h-indoles, -indolinas y compuestos analogos relacionados.

Legal Events

Date	Code	Title	Description
1992-06-30	BB1A	Laying open of patent application	Effective date: 19920225
1999-01-29	FG3A	Patent granted, date of granting	Effective date: 19981022
2005-06-30	MM3A	Annulment or lapse	Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20050422

Date

Code

Title

Description

1992-06-30

BB1A

Laying open of patent application

Effective date: 19920225

1999-01-29

FG3A

Patent granted, date of granting

Effective date: 19981022

2005-06-30

MM3A

Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20050422