[go: up one dir, main page]

PT89630A - Processo para a preparacao de amidas de aminoacidos com accao psicotropica, e de composicoes farmaceuticas que as contem - Google Patents

Processo para a preparacao de amidas de aminoacidos com accao psicotropica, e de composicoes farmaceuticas que as contem

Info

Publication number
PT89630A
PT89630A PT89630A PT8963089A PT89630A PT 89630 A PT89630 A PT 89630A PT 89630 A PT89630 A PT 89630A PT 8963089 A PT8963089 A PT 8963089A PT 89630 A PT89630 A PT 89630A
Authority
PT
Portugal
Prior art keywords
psychotropic
pharmaceutical compositions
compositions containing
amino acid
preparing amino
Prior art date
Application number
PT89630A
Other languages
English (en)
Inventor
Franz Hock
Hansjorg Urbach
Wolfgang Ruger
Reinhard Becker
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of PT89630A publication Critical patent/PT89630A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02Linear peptides containing at least one abnormal peptide link
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/005Enzyme inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Genetics & Genomics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Molecular Biology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
PT89630A 1988-02-04 1989-02-03 Processo para a preparacao de amidas de aminoacidos com accao psicotropica, e de composicoes farmaceuticas que as contem PT89630A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3803225A DE3803225A1 (de) 1988-02-04 1988-02-04 Aminosaeureamide mit psychotroper wirkung, verfahren zu ihrer herstellung, sie enthaltende mittel und deren verwendung

Publications (1)

Publication Number Publication Date
PT89630A true PT89630A (pt) 1989-10-04

Family

ID=6346557

Family Applications (1)

Application Number Title Priority Date Filing Date
PT89630A PT89630A (pt) 1988-02-04 1989-02-03 Processo para a preparacao de amidas de aminoacidos com accao psicotropica, e de composicoes farmaceuticas que as contem

Country Status (12)

Country Link
EP (1) EP0326974A1 (pt)
JP (1) JPH021444A (pt)
KR (1) KR890013057A (pt)
AU (1) AU2958789A (pt)
DE (1) DE3803225A1 (pt)
DK (1) DK51789A (pt)
FI (1) FI890501A (pt)
HU (1) HU203119B (pt)
IL (1) IL89146A0 (pt)
NO (1) NO890447L (pt)
PT (1) PT89630A (pt)
ZA (1) ZA89815B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2611597B2 (ja) * 1992-01-27 1997-05-21 いすゞ自動車株式会社 ディーゼル機関のシリンダヘッド
DE19605175A1 (de) * 1996-02-13 1997-08-14 Sourovoi Andrej Dr Lipidverbindungen und deren Verwendung
NZ571826A (en) * 2006-04-11 2012-01-12 Novartis Ag HCV/HIV inhibitors and their uses
WO2009122433A2 (en) * 2008-03-13 2009-10-08 Ipca Laboratories Limited A process for preparation of ramipril
US8512690B2 (en) 2009-04-10 2013-08-20 Novartis Ag Derivatised proline containing peptide compounds as protease inhibitors
US8669281B1 (en) 2013-03-14 2014-03-11 Alkermes Pharma Ireland Limited Prodrugs of fumarates and their use in treating various diseases
DK2970101T3 (en) 2013-03-14 2018-08-20 Alkermes Pharma Ireland Ltd PRO-DRUGS OF FUMARATES AND THEIR USE IN TREATING DIFFERENT DISEASES
NZ723269A (en) 2014-02-24 2017-04-28 Alkermes Pharma Ireland Ltd Sulfonamide and sulfinamide prodrugs of fumarates and their use in treating various diseases

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL58849A (en) * 1978-12-11 1983-03-31 Merck & Co Inc Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them
GR75019B (pt) * 1980-09-17 1984-07-12 Univ Miami
DE3174844D1 (en) * 1980-10-23 1986-07-24 Schering Corp Carboxyalkyl dipeptides, processes for their production and pharmaceutical compositions containing them
US4462943A (en) * 1980-11-24 1984-07-31 E. R. Squibb & Sons, Inc. Carboxyalkyl amino acid derivatives of various substituted prolines
EP0079521A1 (en) * 1981-11-09 1983-05-25 Merck & Co. Inc. Process for preparation of carboxyalkyldipeptide derivatives
EP0080822A1 (en) * 1981-11-27 1983-06-08 Beecham Group Plc Anti-hypertensive prolinol-based peptides
EP0115091A1 (en) * 1983-01-27 1984-08-08 ENI-Ente Nazionale Idrocarburi N-carboxyacyl derivatives of cyclic amino acids, useful as antihypertensives
CN86101850A (zh) * 1985-03-22 1987-02-04 森得克斯(美国)有限公司 N,n′-二烷基胍基二肽的制造方法与用途
DE3610391A1 (de) * 1986-03-27 1987-10-08 Hoechst Ag Verbindungen mit nootroper wirkung, diese enthaltende mittel und deren verwendung bei der behandlung und prophylaxe cognitiver dysfunktionen

Also Published As

Publication number Publication date
DK51789A (da) 1989-08-05
DE3803225A1 (de) 1989-08-17
JPH021444A (ja) 1990-01-05
EP0326974A1 (de) 1989-08-09
AU2958789A (en) 1989-08-10
IL89146A0 (en) 1989-09-10
ZA89815B (en) 1989-09-27
DK51789D0 (da) 1989-02-03
HU203119B (en) 1991-05-28
KR890013057A (ko) 1989-09-21
HUT50847A (en) 1990-03-28
NO890447D0 (no) 1989-02-03
FI890501A (fi) 1989-08-05
NO890447L (no) 1989-08-07
FI890501A0 (fi) 1989-02-02

Similar Documents

Publication Publication Date Title
PT90836A (pt) Processo para a preparacao de derivados de aminoacidos e de composicoes farmaceuticas que os contem
PT89899A (pt) Processo para a preparacao de novos derivados de aminoacidos e de composicoes farmaceuticas que os contem
PT89094A (pt) Processo para a preparacao de 1-aril-3-quinolina-e 1-aril-3-isoquinolina-carboxamidas e de composicoes farmaceuticas que as contem
PT89009A (pt) Processo para a preparacao de novos derivados de fluorocitidina e composicoes farmaceuticas que os contem
PT83013B (pt) Processo para a preparacao de hidroxialquilxantinas terciarias, e de composicoes farmaceuticas que as contem
PT83143B (pt) Processo para a preparacao de 1,4-dihidro-piridinas 2-substituidas com tiometilo e de composicoes farmaceuticas que as contem
PT88914A (pt) Processo para a preparacao de polipeptidos e de composicoes farmaceuticas que os contem
PT89655B (pt) Processo para a preparacao de novas lactamas substituidas e de composicoes farmaceuticas que as contem
PT84681B (pt) Processo para a preparacao de carboxamidas heterociclicas e de composicoes farmaceuticas que as contem
PT88679A (pt) Processo para a preparacao de derivados de aminoacidos e de composicoes farmaceuticas que os contem
PT98365A (pt) Processo para a preparacao de novos derivados de oxalilo e de composicoes farmaceuticas que os contem
PT84064B (pt) Processo para a preparacao de novos derivados de aminoacidos e de composicoes farmaceuticas que os contem
PT90142A (pt) Processo para a preparacao de novos imidazois substituidos em 2,3 e 4 e de 1,2,4-triazois substituido4 em 3,4 e 5 bem como de composicoes farmaceuticas que os contem
PT84358B (pt) Processo para a preparacao de naftotiazepinonas e de composicoes farmaceuticas que as contem
PT83495B (pt) Processo para a preparacao de difenilpiperidinas n-substituidas e de composicoes farmaceuticas que as contem
PT83239B (pt) Processo para a preparacao de derivados de aminoacidos e de composicoes farmaceuticas que os contem
PT82984B (pt) Processo para a preparacao de derivados de poli-4-aminopirrole-2-carboxamido e de composicoes farmaceuticas que os contem
PT90415A (pt) Processo para a preparacao de sais de adicao de acido de taurina ou glicina amidada e de composicoes farmaceuticas que os contem
PT88335A (pt) Processo para a preparacao de derivados do acido 1,4-dihidro-4-oxo-3-quinolinocarboxilico e de composicoes farmaceuticas que os contem
PT89630A (pt) Processo para a preparacao de amidas de aminoacidos com accao psicotropica, e de composicoes farmaceuticas que as contem
PT89501B (pt) Processo para a preparacao de novos gliceridos de amino-acidos e de composicoes farmaceuticas que os contem
PT91803A (pt) Processo para a preparacao de novos derivados da 2'-halogenometilideno-, 2'-etenilideno- e 2'-etinil-adenosina e de composicoes farmaceuticas que os contem
PT90904A (pt) Processo para a preparacao de derivados de 3-oxo-propanonitrilo triciclicos e de composicoes farmaceuticas que os contem
PT98816A (pt) Processo para a preparacao de tienodiazepinas e de composicoes farmaceuticas que as contem
PT87090A (pt) Processo para a preparacao de derivados de imidazopiridinas e de composicoes farmaceuticas que os contem

Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19931012