[go: up one dir, main page]

PE20120421A1 - Composicion farmaceutica que comprende aleglitazar - Google Patents

Composicion farmaceutica que comprende aleglitazar

Info

Publication number
PE20120421A1
PE20120421A1 PE2011001309A PE2011001309A PE20120421A1 PE 20120421 A1 PE20120421 A1 PE 20120421A1 PE 2011001309 A PE2011001309 A PE 2011001309A PE 2011001309 A PE2011001309 A PE 2011001309A PE 20120421 A1 PE20120421 A1 PE 20120421A1
Authority
PE
Peru
Prior art keywords
pharmaceutical composition
composition obtained
composition
happiness
includes happiness
Prior art date
Application number
PE2011001309A
Other languages
English (en)
Inventor
Alexander Glomme
Paul Wojtera
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of PE20120421A1 publication Critical patent/PE20120421A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biophysics (AREA)
  • Cardiology (AREA)
  • Molecular Biology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

SE REFIERE A UN PROCESO QUE COMPRENDE: A) PULVERIZAR UNA SOLUCION ACUOSA TAMPONADA CON TAMPON FOSFATO QUE CONTIENE 0.01 MG A 0.9 MG DE ALEGLITAZAR, UN AGLUTINANTE TAL COMO 0.1- 20MG DE POVIDONA Y UN TENSOACTIVO TAL COMO 0.1-2 MG DE LAURILSULFATO SOBRE UN DILUYENTE TAL COMO AZUCAR, CELULOSA MICROCRISTALINA, LACTOSA O ALMIDON Y UN DESINTEGRANTE TAL COMO 0.5-20 MG DE CROSCARMELOSA SODICA; B) MEZCLAR LA COMPOSICION OBTENIDA EN EL PASO (A) CON UN LUBRICANTE TAL COMO 0.5-3MG DE ESTEARATO DE MAGNESIO; C) COMPRIMIR LA COMPOSICION OBTENIDA EN EL PASO (B) PARA LA OBTENCION DE UNA TABLETA. DICHA COMPOSICION ES UTIL PARA EL TRATAMIENTO O PROFILAXIS DE LA DIABETES TIPO II O DE ENFERMEDADES CARDIOVASCULARES
PE2011001309A 2009-01-23 2010-01-13 Composicion farmaceutica que comprende aleglitazar PE20120421A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP09151254 2009-01-23

Publications (1)

Publication Number Publication Date
PE20120421A1 true PE20120421A1 (es) 2012-05-04

Family

ID=42112184

Family Applications (2)

Application Number Title Priority Date Filing Date
PE2016000386A PE20160746A1 (es) 2009-01-23 2010-01-13 Composicion farmaceutica que comprende aleglitazar
PE2011001309A PE20120421A1 (es) 2009-01-23 2010-01-13 Composicion farmaceutica que comprende aleglitazar

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PE2016000386A PE20160746A1 (es) 2009-01-23 2010-01-13 Composicion farmaceutica que comprende aleglitazar

Country Status (25)

Country Link
US (2) US20100190835A1 (es)
EP (1) EP2389166B1 (es)
JP (1) JP5619027B2 (es)
KR (2) KR20140002812A (es)
CN (1) CN102292074B (es)
AR (1) AR075041A1 (es)
AU (1) AU2010206249B2 (es)
BR (1) BRPI1007237B1 (es)
CA (1) CA2748896C (es)
CL (1) CL2011001777A1 (es)
CY (1) CY1113641T1 (es)
DK (1) DK2389166T3 (es)
ES (1) ES2397558T3 (es)
HR (1) HRP20130108T1 (es)
IL (1) IL213671A (es)
MX (1) MX2011007381A (es)
PE (2) PE20160746A1 (es)
PL (1) PL2389166T3 (es)
PT (1) PT2389166E (es)
RU (1) RU2537224C2 (es)
SG (1) SG173058A1 (es)
SI (1) SI2389166T1 (es)
TW (1) TWI406861B (es)
WO (1) WO2010084066A1 (es)
ZA (1) ZA201104670B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013181384A1 (en) 2012-05-31 2013-12-05 Ratiopharm Gmbh Solid state forms of aleglitazar sodium
WO2014016369A1 (en) 2012-07-27 2014-01-30 Ratiopharm Gmbh Pharmaceutical formulation comprising aleglitazar and complexing agent
WO2014016370A1 (en) * 2012-07-27 2014-01-30 Ratiopharm Gmbh Amorphous aleglitazar
WO2014016371A1 (en) 2012-07-27 2014-01-30 Ratiopharm Gmbh Micronized aleglitazar
KR20150054829A (ko) * 2012-09-12 2015-05-20 에프. 호프만-라 로슈 아게 (S)-2-메톡시-3-{4-[2-(5-메틸-2-페닐-옥사졸-4-일)-에톡시]-벤조[b]티오펜-7-일}-프로피온산 및 이의 염의 고체 형태
KR102569636B1 (ko) * 2016-08-10 2023-08-23 에프. 호프만-라 로슈 아게 Akt 단백질 키나아제 저해제를 포함하는 약학 조성물
CN114404375B (zh) * 2022-01-21 2023-06-27 武汉九珑人福药业有限责任公司 一种叶酸固体制剂及其原料组合物、制备方法和应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2772615B1 (fr) * 1997-12-23 2002-06-14 Lipha Comprime multicouche pour la liberation instantanee puis prolongee de substances actives
PL208074B1 (pl) * 2001-05-15 2011-03-31 Hoffmann La Roche Pochodne oksazolu, sposób ich wytwarzania, środek farmaceutyczny i zastosowanie pochodnych oksazolu
GB0303600D0 (en) * 2003-02-17 2003-03-19 Glaxo Group Ltd Novel therapeutic method and compositions
US7262303B2 (en) * 2003-09-29 2007-08-28 Hoffman-La Roche Inc. Process for the production of chiral propionic acid derivatives
US20060051413A1 (en) * 2004-09-08 2006-03-09 Chow Sing S M Method of enhancing absorptions of transmucosal administration formulations
RU2007129642A (ru) * 2005-02-25 2009-03-27 Ф.Хоффманн-Ля Рош Аг (Ch) Таблетки с улучшенным распределением лекарственного вещества
US20060270722A1 (en) * 2005-05-31 2006-11-30 Thornberry Nancy A Combination of a dipeptidyl peptidase-IV inhibitor and a dual PPAR agonist for the treatment of diabetes and obesity
FR2894477A1 (fr) * 2005-12-13 2007-06-15 Galderma Res & Dev Utilisation du naveglitazar pour la preparation d'une composition pharmaceutique destinee au traitement des affections dermatologiques
US20100210692A1 (en) * 2007-03-28 2010-08-19 Farmer Stephen R Methods of treatment using sirt modulators and compositions containing sirt1 modulators

Also Published As

Publication number Publication date
IL213671A0 (en) 2011-07-31
MX2011007381A (es) 2011-08-12
JP2012515741A (ja) 2012-07-12
CL2011001777A1 (es) 2012-02-24
RU2537224C2 (ru) 2014-12-27
AR075041A1 (es) 2011-03-02
CA2748896C (en) 2017-01-03
RU2011134964A (ru) 2013-02-27
ZA201104670B (en) 2012-03-28
PL2389166T3 (pl) 2013-04-30
JP5619027B2 (ja) 2014-11-05
CY1113641T1 (el) 2016-06-22
EP2389166B1 (en) 2012-11-21
BRPI1007237B1 (pt) 2019-05-28
AU2010206249A1 (en) 2011-06-30
BRPI1007237A2 (pt) 2016-02-16
SI2389166T1 (sl) 2013-02-28
CN102292074B (zh) 2013-08-21
US20100190835A1 (en) 2010-07-29
WO2010084066A1 (en) 2010-07-29
DK2389166T3 (da) 2012-12-17
KR20140002812A (ko) 2014-01-08
TW201035089A (en) 2010-10-01
SG173058A1 (en) 2011-08-29
PT2389166E (pt) 2013-01-08
CA2748896A1 (en) 2010-07-29
US20130072529A1 (en) 2013-03-21
EP2389166A1 (en) 2011-11-30
IL213671A (en) 2015-11-30
ES2397558T3 (es) 2013-03-07
HRP20130108T1 (hr) 2013-03-31
AU2010206249B2 (en) 2015-07-09
CN102292074A (zh) 2011-12-21
KR20110105798A (ko) 2011-09-27
TWI406861B (zh) 2013-09-01
PE20160746A1 (es) 2016-08-01

Similar Documents

Publication Publication Date Title
PE20120421A1 (es) Composicion farmaceutica que comprende aleglitazar
ES2524771T3 (es) Composiciones farmacéuticas que comprenden levetiracetam y procedimientos para su preparación
PE20070698A1 (es) Comprimido de disgregacion rapida intraoral que contiene hidrocloruro de ambroxol
HN2011001446A (es) Compuesto utiles para inhibir chk1
ECSP10010160A (es) Composiciones farmaceuticas de accion doble basadas en super-estructuras de antagonista/bloqueador del receptor de angiotensina (arb) e inhibidor de endopeptidasa neutra (nep)
CL2008003827A1 (es) Composicion para tabletas de desintegracion oral que comprende al menos una droga ( temazepam), 0,5-3% de un polimero aglutinanete para odt, un alcohol de azucar y/o sacarido, y un desintegrante; metodo para prepararla; util para tratar una enfermedad o condicion como un trastorno del sueño en pacientes con disfagia..
PE20061345A1 (es) Composicion farmaceutica que comprende sorafenib
PE20090015A1 (es) Preparacion solida
CL2012000793A1 (es) Composicion farmaceutica que comprende 1-cloro-4-(3-d-glucopiranos-il)-2-[4-((s)-tetrahidrofuran-3-iloxi)-bencil]benceno, clorhidrato de metformina y uno o mas excipientes farmaceuticos.
BRPI0922796A2 (pt) Comprimido farmacêutico para administração por via oral e método de fabricação do mesmo
IN2015DN02907A (es)
DOP2011000047A (es) Agentes terapeuticos 414
CR10992A (es) Preparacion solida que comprende alogliptina y pioglitazona
RU2014138035A (ru) Твердая фармацевтическая композиция, содержащая 1-(3-(2-(1-бензотиофен-5-ил)этокси)пропил)азетидин-3-ол или его соль
PE20220751A1 (es) Composiciones solidas que comprenden un agonista del glp-1, un inhibidor del sglt2 y una sal del acido n-(8-(2-hidroxibenzoil)amino)caprilico
PE20080376A1 (es) Formulaciones de comprimidos de liberacion inmediata de un antagonista del receptor de trombina derivado de fluorofenilpiridina
BR112012027794A2 (pt) tablete entérico
MX387086B (es) Preparacion compuesta, que contiene derivado novedoso de acido 3-(4-(benciloxi)fenil)hex-4-inoico y otro ingrediente activo, para prevenir o tratar enfermedades metabolicas
CR11398A (es) Compuesto inhibidor de glicogeno fosforilasa y composicion farmaceutica del mismo.
CL2011002650A1 (es) Composicion que comprende n-(4-(2-furil)-5-(tetrahidropiran-4-ilcarbonil)tiazol-2-il)-2-metilpiridin-5-carboxamida y l-dopa; uso del compuesto para el tratamiento de un trastorno del movimiento secundario de la terapia con l-dopa; uso del compuesto y l-dopa y/o para el tratamiento y/o profilaxis de la enfermedad de parkinson.
RU2008135718A (ru) Композиции клопидогреля бисульфата
ES2721649T3 (es) Comprimidos de N-acetilcisteína tragables
PE20061390A1 (es) Formulaciones de acido hidroxamico suberoilanilida y procedimientos para la produccion de las mismas
PE20060768A1 (es) Composicion farmaceutica que comprende hidroclorotiazida y telmisartano
BRPI0713371A2 (pt) método para a produção de um produto medicamentoso contendo olmesartan medoxomil, e, produto medicamentoso contendo olmesartan medoxomil

Legal Events

Date Code Title Description
FC Refusal