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PA8600601A1 - Ligandos de receptores de cannabinoides y sus usos - Google Patents

Ligandos de receptores de cannabinoides y sus usos

Info

Publication number
PA8600601A1
PA8600601A1 PA20048600601A PA8600601A PA8600601A1 PA 8600601 A1 PA8600601 A1 PA 8600601A1 PA 20048600601 A PA20048600601 A PA 20048600601A PA 8600601 A PA8600601 A PA 8600601A PA 8600601 A1 PA8600601 A1 PA 8600601A1
Authority
PA
Panama
Prior art keywords
cannabinoid
receiver links
links
receiver
cannabinoid receptors
Prior art date
Application number
PA20048600601A
Other languages
English (en)
Inventor
Robert Lee Dow
Philip Albert Carpino
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of PA8600601A1 publication Critical patent/PA8600601A1/es

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34—Tobacco-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Nutrition Science (AREA)
  • Reproductive Health (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Gynecology & Obstetrics (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)

Abstract

EN LA PRESENTE, SE DESCRIBEN COMPUESTOS DE FORMULA (I) Y (II) QUE ACTUAN COMO LIGANDOS DE RECEPTORES DE CANNABINOIDES, Y SUS USOS EN EL TRATAMIENTO DE ENFERMEDADES CONECTADAS CON LA MEDIACION DE RECEPTORES DE CANNABINOIDES EN ANIMALES.
PA20048600601A 2003-04-23 2004-04-20 Ligandos de receptores de cannabinoides y sus usos PA8600601A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US46490803P 2003-04-23 2003-04-23

Publications (1)

Publication Number Publication Date
PA8600601A1 true PA8600601A1 (es) 2005-05-24

Family

ID=33310977

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20048600601A PA8600601A1 (es) 2003-04-23 2004-04-20 Ligandos de receptores de cannabinoides y sus usos

Country Status (31)

Country Link
US (1) US20040214856A1 (es)
EP (1) EP1622903B1 (es)
JP (1) JP2006524225A (es)
KR (1) KR20060006048A (es)
CN (1) CN1809566A (es)
AP (1) AP2005003427A0 (es)
AR (1) AR044037A1 (es)
AT (1) ATE409700T1 (es)
AU (1) AU2004232552A1 (es)
BR (1) BRPI0409791A (es)
CA (1) CA2521538A1 (es)
CL (1) CL2004000827A1 (es)
CO (1) CO5640084A2 (es)
DE (1) DE602004016839D1 (es)
EA (1) EA200501504A1 (es)
EC (1) ECSP056117A (es)
ES (1) ES2309517T3 (es)
GT (1) GT200400076A (es)
IS (1) IS8054A (es)
MA (1) MA27766A1 (es)
MX (1) MXPA05011454A (es)
NL (1) NL1026027C2 (es)
NO (1) NO20055516L (es)
OA (1) OA13047A (es)
PA (1) PA8600601A1 (es)
PE (1) PE20050419A1 (es)
TN (1) TNSN05272A1 (es)
TW (1) TW200510419A (es)
UY (1) UY28276A1 (es)
WO (1) WO2004094421A1 (es)
ZA (1) ZA200508568B (es)

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IS8054A (is) 2005-09-29
ATE409700T1 (de) 2008-10-15
EA200501504A1 (ru) 2006-04-28
TW200510419A (en) 2005-03-16
CO5640084A2 (es) 2006-05-31
BRPI0409791A (pt) 2006-05-30
MA27766A1 (fr) 2006-02-01
AR044037A1 (es) 2005-08-24
EP1622903A1 (en) 2006-02-08
ECSP056117A (es) 2006-03-01
CL2004000827A1 (es) 2005-03-04
GT200400076A (es) 2004-12-16
WO2004094421A1 (en) 2004-11-04
ZA200508568B (en) 2007-04-25
NL1026027A1 (nl) 2004-10-27
US20040214856A1 (en) 2004-10-28
ES2309517T3 (es) 2008-12-16
EP1622903B1 (en) 2008-10-01
CA2521538A1 (en) 2004-11-04
TNSN05272A1 (fr) 2007-07-10
KR20060006048A (ko) 2006-01-18
OA13047A (en) 2006-11-10
UY28276A1 (es) 2004-11-30
NL1026027C2 (nl) 2005-07-05
MXPA05011454A (es) 2005-12-12
AU2004232552A1 (en) 2004-11-04
NO20055516L (no) 2005-11-22
JP2006524225A (ja) 2006-10-26
DE602004016839D1 (de) 2008-11-13
CN1809566A (zh) 2006-07-26
PE20050419A1 (es) 2005-06-18
AP2005003427A0 (en) 2005-12-31

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