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NO991534L - Farmas°ytiske forbindelser som omfatter polyaminer substituert med elektronaffinitetsgrupper - Google Patents

Farmas°ytiske forbindelser som omfatter polyaminer substituert med elektronaffinitetsgrupper

Info

Publication number
NO991534L
NO991534L NO991534A NO991534A NO991534L NO 991534 L NO991534 L NO 991534L NO 991534 A NO991534 A NO 991534A NO 991534 A NO991534 A NO 991534A NO 991534 L NO991534 L NO 991534L
Authority
NO
Norway
Prior art keywords
electron affinity
affinity groups
pharmaceutical compounds
group
compound
Prior art date
Application number
NO991534A
Other languages
English (en)
Other versions
NO991534D0 (no
Inventor
Li-Xi Yang
Kurt G Hofer
Original Assignee
Univ Florida
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Florida filed Critical Univ Florida
Publication of NO991534D0 publication Critical patent/NO991534D0/no
Publication of NO991534L publication Critical patent/NO991534L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/91—Nitro radicals
    • C07D233/92—Nitro radicals attached in position 4 or 5
    • C07D233/95—Nitro radicals attached in position 4 or 5 with hydrocarbon radicals, substituted by nitrogen atoms, attached to other ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/20—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic unsaturated carbon skeleton
    • C07C211/22—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic unsaturated carbon skeleton containing at least two amino groups bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0086—Platinum compounds
    • C07F15/0093—Platinum compounds without a metal-carbon linkage

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

En forbindelse eller et salt derav som omfatter et polyamin som inneholder minst 2 elektronaffinitets- grupper, er tilveiebrakt. Ved en fore- trukket utførelsesform har polyaminfor- bindelsen formelen (1) B\ /R NAN R'' V (1) hvor A er en avstandsdel; R1, R2, R3 og R* er uavhengig av hverandre hydrogen, hydrokarbon, heterosubstituert hydro- karbon, heteroaryl, heterosubstituert heteroaryl eller en elektronaffinitets- gruppe som inneholder substituent; og forbindelsen inneholder minst en ter- tiær amingruppe som har tre substitu- enter som hver uavhengig av hverandre inneholder minst en elektronaffinitets- gruppe eller hydrofil gruppe.
NO991534A 1996-09-30 1999-03-29 Farmas°ytiske forbindelser som omfatter polyaminer substituert med elektronaffinitetsgrupper NO991534L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/722,396 US6060604A (en) 1995-03-31 1996-09-30 Pharmaceutical compounds comprising polyamines substituted with electron-affinic groups
PCT/US1997/017408 WO1998014190A1 (en) 1996-09-30 1997-09-29 Pharmaceutical compounds comprising polyamines substituted with electron-affinic groups

Publications (2)

Publication Number Publication Date
NO991534D0 NO991534D0 (no) 1999-03-29
NO991534L true NO991534L (no) 1999-03-29

Family

ID=24901655

Family Applications (1)

Application Number Title Priority Date Filing Date
NO991534A NO991534L (no) 1996-09-30 1999-03-29 Farmas°ytiske forbindelser som omfatter polyaminer substituert med elektronaffinitetsgrupper

Country Status (10)

Country Link
US (3) US6060604A (no)
EP (1) EP0956016A4 (no)
JP (1) JP2001501932A (no)
KR (1) KR20000048682A (no)
CN (1) CN1232395A (no)
AU (1) AU725206B2 (no)
BR (1) BR9713241A (no)
CA (1) CA2265558A1 (no)
NO (1) NO991534L (no)
WO (1) WO1998014190A1 (no)

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US6423707B1 (en) 2000-08-28 2002-07-23 California Pacific Medical Center Nitroimidazole ester analogues and therapeutic applications
US6723755B2 (en) 2002-06-12 2004-04-20 Piotr Chomczynski Method of treating rosacea
US7459502B2 (en) * 2003-11-03 2008-12-02 Ilypsa, Inc. Pharmaceutical compositions comprising crosslinked polyamine polymers
US7335795B2 (en) 2004-03-22 2008-02-26 Ilypsa, Inc. Crosslinked amine polymers
US7767768B2 (en) * 2003-11-03 2010-08-03 Ilypsa, Inc. Crosslinked amine polymers
US7449605B2 (en) * 2003-11-03 2008-11-11 Ilypsa, Inc. Crosslinked amine polymers
US7608674B2 (en) * 2003-11-03 2009-10-27 Ilypsa, Inc. Pharmaceutical compositions comprising cross-linked small molecule amine polymers
US7385012B2 (en) * 2003-11-03 2008-06-10 Ilypsa, Inc. Polyamine polymers
US7812057B2 (en) * 2004-08-25 2010-10-12 Molecular Research Center, Inc. Cosmetic compositions
US7875602B2 (en) * 2005-10-21 2011-01-25 Sutter West Bay Hospitals Camptothecin derivatives as chemoradiosensitizing agents
WO2014117021A2 (en) * 2013-01-25 2014-07-31 Xcell Biosciences, Inc. Methods, compositions, kits, and systems for selective enrichment of target cells

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Also Published As

Publication number Publication date
US6057453A (en) 2000-05-02
AU725206B2 (en) 2000-10-05
US6060604A (en) 2000-05-09
BR9713241A (pt) 2000-04-04
WO1998014190A1 (en) 1998-04-09
NO991534D0 (no) 1999-03-29
CA2265558A1 (en) 1998-04-09
KR20000048682A (ko) 2000-07-25
AU4655497A (en) 1998-04-24
JP2001501932A (ja) 2001-02-13
EP0956016A1 (en) 1999-11-17
US6255495B1 (en) 2001-07-03
CN1232395A (zh) 1999-10-20
EP0956016A4 (en) 2001-11-14

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