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NO991056D0 - Rene enantiomere basiske aryl-cykloalkyl-hydroksykarboksylsyreestere, fremgangsmÕte for deres fremstilling og anvendelse derav i medikamenter - Google Patents

Rene enantiomere basiske aryl-cykloalkyl-hydroksykarboksylsyreestere, fremgangsmÕte for deres fremstilling og anvendelse derav i medikamenter

Info

Publication number
NO991056D0
NO991056D0 NO991056A NO991056A NO991056D0 NO 991056 D0 NO991056 D0 NO 991056D0 NO 991056 A NO991056 A NO 991056A NO 991056 A NO991056 A NO 991056A NO 991056 D0 NO991056 D0 NO 991056D0
Authority
NO
Norway
Prior art keywords
cycloalkyl
hydroxycarboxylic acid
medicaments
preparation
acid esters
Prior art date
Application number
NO991056A
Other languages
English (en)
Other versions
NO314354B1 (no
NO991056L (no
Inventor
Guenter Lambrecht
Michael Elgert
Sittah Czeche
Magali Waelbroeck
Original Assignee
Noe Christian R
Mutschler Ernst
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Noe Christian R, Mutschler Ernst filed Critical Noe Christian R
Publication of NO991056D0 publication Critical patent/NO991056D0/no
Publication of NO991056L publication Critical patent/NO991056L/no
Publication of NO314354B1 publication Critical patent/NO314354B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/12—Oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/42—Oxygen atoms attached in position 3 or 5

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO19991056A 1996-11-11 1999-03-03 Enantiomerrene estere, fremgangsmåte for deres fremstilling og deres anvendelse i legemidler NO314354B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AT197396 1996-11-11
PCT/AT1997/000245 WO1998021183A1 (de) 1996-11-11 1997-11-11 Enantiomerenreine, basische aryl-cycloalkyl-hydroxycarbonsäureester, verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln

Publications (3)

Publication Number Publication Date
NO991056D0 true NO991056D0 (no) 1999-03-03
NO991056L NO991056L (no) 1999-05-11
NO314354B1 NO314354B1 (no) 2003-03-10

Family

ID=3525062

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19991056A NO314354B1 (no) 1996-11-11 1999-03-03 Enantiomerrene estere, fremgangsmåte for deres fremstilling og deres anvendelse i legemidler

Country Status (19)

Country Link
US (1) US6307060B1 (no)
EP (3) EP0937041B1 (no)
JP (1) JP2001504459A (no)
CN (1) CN100391942C (no)
AT (1) ATE238280T1 (no)
AU (1) AU745331B2 (no)
CA (1) CA2271276C (no)
DE (1) DE59709927D1 (no)
DK (2) DK0937041T3 (no)
ES (2) ES2407135T3 (no)
HK (1) HK1061023A1 (no)
HU (1) HU228273B1 (no)
NO (1) NO314354B1 (no)
NZ (1) NZ336202A (no)
PL (1) PL195520B1 (no)
PT (2) PT937041E (no)
RU (1) RU2238936C2 (no)
SI (2) SI1371645T1 (no)
WO (1) WO1998021183A1 (no)

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AR044851A1 (es) 2003-06-24 2005-10-05 Novartis Ag Compuestos heterociclicos, antagonistas del receptor m3 muscarinico
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GB0428416D0 (en) * 2004-12-24 2005-02-02 Novartis Ag Organic compounds
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PL1863476T3 (pl) * 2005-03-16 2016-07-29 Meda Pharma Gmbh & Co Kg Skojarzenie środków antycholinergicznych i antagonistów receptora leukotrienowego do leczenia chorób układu oddechowego
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JP5873013B2 (ja) * 2009-05-29 2016-03-01 パール セラピューティクス，インコーポレイテッド ２つ以上の活性剤を呼吸器送達するための組成物、方法および系
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EP2580194A1 (en) * 2010-06-14 2013-04-17 Chiesi Farmaceutici S.p.A. Process for the preparation of glycopyrronium chloride
JOP20120023B1 (ar) 2011-02-04 2022-03-14 Novartis Ag صياغات مساحيق جافة من جسيمات تحتوي على واحد أو اثنين من المواد الفعالة لعلاج امراض ممرات الهواء الانسدادية او الالتهابية
CN102627595A (zh) * 2012-03-09 2012-08-08 徐奎 一种制备格隆溴铵的方法
KR102232806B1 (ko) 2013-02-28 2021-03-29 더미라, 인코포레이티드 글리코피롤레이트 염
US9006462B2 (en) 2013-02-28 2015-04-14 Dermira, Inc. Glycopyrrolate salts
US8558008B2 (en) 2013-02-28 2013-10-15 Dermira, Inc. Crystalline glycopyrrolate tosylate
JP6232079B2 (ja) 2013-03-14 2017-11-15 ノバルティス アーゲー スプレーブレンディングによるスプレー乾燥製剤の脱アモルファス化
US9452139B2 (en) 2013-03-14 2016-09-27 Novartis Ag Respirable agglomerates of porous carrier particles and micronized drug
CN104586841A (zh) * 2013-10-30 2015-05-06 中国药科大学 (3r,2’r)-格隆溴铵作为m3毒蕈碱性受体拮抗剂在制药中的用途
US9926270B2 (en) 2014-08-20 2018-03-27 Dermira, Inc. Process for production of glycopyrronium tosylate
ES2700597T3 (es) * 2014-12-24 2019-02-18 Lesvi Laboratorios Sl Proceso para la preparación de (3RS) -3 - [(2SR) - (2-ciclopentil-2-hidroxi-2-fenilacetil) oxi] -1,1-dimetilpirrolidinio
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Also Published As

Publication number Publication date
NO314354B1 (no) 2003-03-10
US6307060B1 (en) 2001-10-23
PL332595A1 (en) 1999-09-27
CA2271276C (en) 2009-01-13
PT1371645E (pt) 2013-05-21
ES2407135T3 (es) 2013-06-11
SI0937041T1 (en) 2003-10-31
DE59709927D1 (de) 2003-05-28
JP2001504459A (ja) 2001-04-03
DK1371645T3 (da) 2013-06-03
RU2238936C2 (ru) 2004-10-27
CA2271276A1 (en) 1998-05-22
DK0937041T3 (da) 2003-08-11
NZ336202A (en) 2000-10-27
NO991056L (no) 1999-05-11
EP1371645B1 (de) 2013-02-20
HU228273B1 (en) 2013-02-28
CN1237159A (zh) 1999-12-01
HUP9903791A3 (en) 2001-10-29
EP0937041B1 (de) 2003-04-23
ATE238280T1 (de) 2003-05-15
CN100391942C (zh) 2008-06-04
PL195520B1 (pl) 2007-09-28
EP1371645A1 (de) 2003-12-17
PT937041E (pt) 2003-09-30
SI1371645T1 (sl) 2013-07-31
AU4856097A (en) 1998-06-03
AU745331B2 (en) 2002-03-21
WO1998021183A1 (de) 1998-05-22
HUP9903791A2 (hu) 2000-03-28
EP1369414A1 (de) 2003-12-10
ES2195121T3 (es) 2003-12-01
HK1061023A1 (no) 2004-09-03
EP0937041A1 (de) 1999-08-25

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