NO964348D0 - CCK- eller gastrin-modulerende 5-hetrocykliske-1,5-benzodiazepiner - Google Patents

CCK- eller gastrin-modulerende 5-hetrocykliske-1,5-benzodiazepiner

Info

Publication number: NO964348D0
Authority: NO; Norway
Prior art keywords: gastrin; cck; benzodiazepines; modulating; heterocyclic
Prior art date: 1994-04-14

Application number

NO964348A

Other languages

English (en)

Other versions

NO964348L (no

Inventor

Christopher Joseph Aquino

Elisabeth Ellen Sugg

Jerzy Ryszard Szewczyk

Original Assignee

Glaxo Wellcome Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-04-14

Filing date

1996-10-11

Publication date

1996-10-11

1994-04-14 Priority claimed from GB9407433A external-priority patent/GB9407433D0/en

1994-10-14 Priority claimed from GB9420783A external-priority patent/GB9420783D0/en

1996-10-11 Application filed by Glaxo Wellcome Inc filed Critical Glaxo Wellcome Inc

1996-10-11 Publication of NO964348D0 publication Critical patent/NO964348D0/no

1996-12-02 Publication of NO964348L publication Critical patent/NO964348L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Diabetes (AREA)
General Chemical & Material Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Obesity (AREA)
Hematology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Endocrinology (AREA)
Emergency Medicine (AREA)
Child & Adolescent Psychology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

NO964348A 1994-04-14 1996-10-11 CCK- eller gastrin-modulerende 5-hetrocykliske-1,5-benzodiazepiner NO964348L (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GB9407433A GB9407433D0 (en)	1994-04-14	1994-04-14	Heterocyclic derivatives
GB9420783A GB9420783D0 (en)	1994-10-14	1994-10-14	Heterocyclic derivatives
PCT/US1995/004163 WO1995028419A1 (en)	1994-04-14	1995-04-12	Cck or gastrin modulating 5-heterocyclic-1,5-benzodiazepines

Publications (2)

Publication Number	Publication Date
NO964348D0 true NO964348D0 (no)	1996-10-11
NO964348L NO964348L (no)	1996-12-02

Family

ID=26304703

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO964348A NO964348L (no)	1994-04-14	1996-10-11	CCK- eller gastrin-modulerende 5-hetrocykliske-1,5-benzodiazepiner

Country Status (25)

Country	Link
EP (1)	EP0756602B1 (no)
JP (1)	JPH09511223A (no)
KR (1)	KR970702274A (no)
CN (1)	CN1176646A (no)
AT (1)	ATE181737T1 (no)
AU (1)	AU697349B2 (no)
BR (1)	BR9507381A (no)
CA (1)	CA2186900A1 (no)
CZ (1)	CZ286764B6 (no)
DE (1)	DE69510545T2 (no)
DK (1)	DK0756602T3 (no)
ES (1)	ES2135722T3 (no)
FI (1)	FI964045A (no)
GR (1)	GR3031335T3 (no)
HU (1)	HUT76135A (no)
IL (1)	IL113365A (no)
IS (1)	IS4367A (no)
MX (1)	MX9604765A (no)
NO (1)	NO964348L (no)
NZ (1)	NZ283929A (no)
PL (1)	PL180026B1 (no)
RU (1)	RU2152939C1 (no)
SK (1)	SK281433B6 (no)
TW (1)	TW369529B (no)
WO (1)	WO1995028419A1 (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9307833D0 (en) *	1993-04-15	1993-06-02	Glaxo Inc	Modulators of cholecystokinin and gastrin
PE27497A1 (es) *	1994-04-15	1997-08-07	Glaxo Inc	Derivados de 1,5 benzodiazepina
WO1998025911A1 (fr) *	1996-12-10	1998-06-18	Zeria Pharmaceutical Co., Ltd.	Derives de 1,5-benzodiazepine
US7910548B2 (en) *	1997-06-06	2011-03-22	Amylin Pharmaceuticals, Inc.	Methods for treating obesity
EP1123928A4 (en) *	1998-10-20	2005-02-16	Takeda Pharmaceutical	1,5-BENZODIAZEPINE COMPOUNDS, PROCESS FOR PRODUCING THE SAME, AND MEDICAMENT
JP4535350B2 (ja) *	1998-11-17	2010-09-01	クミアイ化学工業株式会社	ピリミジニルベンズイミダゾール誘導体及び農園芸用殺菌剤
ES2311120T3 (es) *	2002-08-27	2009-02-01	Merck Patent Gmbh	Derivados de glicinamida como inhibidores de quinasa-raf.
CN1950374A (zh)	2004-05-25	2007-04-18	辉瑞产品公司	四氮杂苯并[e]甘菊环衍生物及其类似物
SG11201404030YA (en)	2012-01-13	2014-10-30	Nippon Chemiphar Co	P2x4 receptor antagonist
CN109071504B (zh)	2016-02-05	2022-03-08	戴纳立制药公司	受体相互作用蛋白激酶1的抑制剂
PL3552017T3 (pl)	2016-12-09	2022-08-08	Denali Therapeutics Inc.	Związki użyteczne jako inhibitory RIPK1
PH12022550852A1 (en)	2019-10-07	2023-05-03	Kallyope Inc	Gpr119 agonists
MX2024008648A (es)	2022-01-12	2024-09-23	Denali Therapeutics Inc	Formas cristalinas de (s)-5-bencil-n-(5-metil-4-oxo-2,3,4,5-tetrah idropirido [3,2- b][1,4]oxacepin-3-il)-4h-1,2,4-triazol-3-carboxam ida.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2641280B1 (fr) *	1988-12-29	1994-01-21	Roussel Uclaf	Nouveaux derives de la 2,4-dioxo 2,3,4,5-tetrahydro 1h-1,5-benzodiazepine, leur procede de preparation et leur application comme medicaments
GEP20001968B (en) *	1992-01-21	2000-03-05	Glaxo Spa	Arilthio Compounds as Antibacterial and Antiviral Agents
GB9307833D0 (en) *	1993-04-15	1993-06-02	Glaxo Inc	Modulators of cholecystokinin and gastrin

1995
- 1995-04-12 CN CN95193582A patent/CN1176646A/zh active Pending
- 1995-04-12 DE DE69510545T patent/DE69510545T2/de not_active Expired - Fee Related
- 1995-04-12 NZ NZ283929A patent/NZ283929A/en unknown
- 1995-04-12 TW TW084103539A patent/TW369529B/zh active
- 1995-04-12 DK DK95915540T patent/DK0756602T3/da active
- 1995-04-12 SK SK1300-96A patent/SK281433B6/sk unknown
- 1995-04-12 AU AU22390/95A patent/AU697349B2/en not_active Ceased
- 1995-04-12 CZ CZ19962972A patent/CZ286764B6/cs not_active IP Right Cessation
- 1995-04-12 RU RU96121555/04A patent/RU2152939C1/ru active
- 1995-04-12 JP JP7516406A patent/JPH09511223A/ja active Pending
- 1995-04-12 ES ES95915540T patent/ES2135722T3/es not_active Expired - Lifetime
- 1995-04-12 CA CA002186900A patent/CA2186900A1/en not_active Abandoned
- 1995-04-12 BR BR9507381A patent/BR9507381A/pt unknown
- 1995-04-12 EP EP95915540A patent/EP0756602B1/en not_active Expired - Lifetime
- 1995-04-12 WO PCT/US1995/004163 patent/WO1995028419A1/en active IP Right Grant
- 1995-04-12 HU HU9602835A patent/HUT76135A/hu unknown
- 1995-04-12 MX MX9604765A patent/MX9604765A/es unknown
- 1995-04-12 AT AT95915540T patent/ATE181737T1/de not_active IP Right Cessation
- 1995-04-12 KR KR1019960705732A patent/KR970702274A/ko not_active Application Discontinuation
- 1995-04-12 PL PL95316870A patent/PL180026B1/pl unknown
- 1995-04-13 IL IL11336595A patent/IL113365A/xx not_active IP Right Cessation
1996
- 1996-09-30 IS IS4367A patent/IS4367A/is unknown
- 1996-10-09 FI FI964045A patent/FI964045A/fi unknown
- 1996-10-11 NO NO964348A patent/NO964348L/no not_active Application Discontinuation
1999
- 1999-09-28 GR GR990402437T patent/GR3031335T3/el unknown

Also Published As

Publication number	Publication date
HUT76135A (en)	1997-06-30
CA2186900A1 (en)	1995-10-26
JPH09511223A (ja)	1997-11-11
CN1176646A (zh)	1998-03-18
FI964045A0 (fi)	1996-10-09
FI964045A (fi)	1996-10-09
NZ283929A (en)	1998-02-26
PL180026B1 (pl)	2000-12-29
EP0756602A1 (en)	1997-02-05
IL113365A (en)	1999-11-30
WO1995028419A1 (en)	1995-10-26
GR3031335T3 (en)	1999-12-31
DK0756602T3 (da)	2000-01-31
CZ297296A3 (en)	1997-09-17
IS4367A (is)	1996-09-30
ES2135722T3 (es)	1999-11-01
HU9602835D0 (en)	1996-12-30
SK281433B6 (sk)	2001-03-12
AU2239095A (en)	1995-11-10
AU697349B2 (en)	1998-10-01
DE69510545D1 (de)	1999-08-05
PL316870A1 (en)	1997-02-17
CZ286764B6 (en)	2000-06-14
SK130096A3 (en)	1997-08-06
NO964348L (no)	1996-12-02
RU2152939C1 (ru)	2000-07-20
IL113365A0 (en)	1995-07-31
DE69510545T2 (de)	2000-01-13
MX9604765A (es)	1998-05-31
KR970702274A (ko)	1997-05-13
TW369529B (en)	1999-09-11
ATE181737T1 (de)	1999-07-15
BR9507381A (pt)	1997-09-23
EP0756602B1 (en)	1999-06-30

Publication	Publication Date	Title
ES2138691T3 (es)	2000-01-16	Procedimiento para la obtencion de derivados de n-acil-5-fluorocitidina.
GB9514473D0 (en)	1995-09-13	Chemical compounds
NO904802L (no)	1991-05-07	Fremgangsmaate for fremstilling av aromatiske aminforbindelser.
MX9204661A (es)	1994-02-28	Compuestos intermedios derivados de eter y procedimiento para su preparacion.
NO904595L (no)	1991-08-06	Fremgangsmaate for potensiering av den analgetiske effekt av curcuminoider.
AR010062A1 (es)	2000-05-17	Nuevos benzamidaldehidos y su utilizacion
IT1285770B1 (it)	1998-06-18	Composti corticoidei
AR004498A1 (es)	1998-12-16	Compuestos de aminofosfonato y composiciones farmaceuticas que los contienen, el uso de los mismos, y un procedimiento para su preparacion
NO904075D0 (no)	1990-09-18	Fremgangsmaate for oksydativ kobling av metan.
DK0756602T3 (da)	2000-01-31	CCK- eller gastrin-modulerende 5-heterocyclo-1,5-benzodiazepiner
NO911122D0 (no)	1991-03-20	Fremgangsmaate for fremstilling av antihyperkolesterolemiske midler.
EE9900450A (et)	2000-04-17	Tetrahüdropüridoühendid, neid sisaldav ravim ja nende kasutamine
ATE110365T1 (de)	1994-09-15	2-alkyl-4-arylmethylaminochinoline, ihre verwendung und daraus hergestellte arzneimittel.
MX9204342A (es)	1994-03-31	Indoles.
ES8601908A1 (es)	1985-11-16	Procedimiento para la preparacion de nuevas 5,11-dihidro-6h-dibenzo (b,e)azepin-6-onas sustituidas
TR199701202T1 (xx)	1998-03-21	Yeni hidroksimik asit t�revleri.
UY24915A1 (es)	2000-12-29	Derivados de benzoxazindiona, aplicación de los mismos y medicamentos que los contienen
AR021616A1 (es)	2002-07-31	Cicloheptenos sustituidos, procedimiento para su preparacion y uso de los mismos.
ATE176477T1 (de)	1999-02-15	Neue phospholipidderivate
MX9701764A (es)	1997-06-28	Derivados de imidoacidos.
SE9602416D0 (sv)	1996-06-18	New forms of an organic salt of N'N-diacetylcystine
DE59810106D1 (de)	2003-12-11	Substituierte 2,4-diamino-1,3,5-triazine
TR199701011A2 (xx)	1998-04-21	1-karba-(detia)-sefalosforin t�revleri.
RU2076517C1 (ru)	1997-03-27	Пищевой краситель
ECSP972052A (es)	1998-02-13	Quinoxalinadionas

Legal Events

Date	Code	Title	Description
2003-01-20	FC2A	Withdrawal, rejection or dismissal of laid open patent application