NO932325L - NEW BENZODIAZEPINE DERIVATIVES - Google Patents
NEW BENZODIAZEPINE DERIVATIVESInfo
- Publication number
- NO932325L NO932325L NO93932325A NO932325A NO932325L NO 932325 L NO932325 L NO 932325L NO 93932325 A NO93932325 A NO 93932325A NO 932325 A NO932325 A NO 932325A NO 932325 L NO932325 L NO 932325L
- Authority
- NO
- Norway
- Prior art keywords
- membered
- receptor
- cck
- substituted aryl
- new benzodiazepine
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Nytt benzodiazepinderivat representert ved generell formel (I) et farmasøytisk akseptabelt salt derav, et farmasøytisk preparat derav, og en fremgangsmåte for frem- stilling av dette. I formel (I) betegner R1 eventuelt substituert aryl, 5-leddet monosyklisk gruppe, 6-leddet monosyklisk gruppe eller aromatisk, heterosyklisk gruppe om- fattende 5-leddede og 6-leddede ringer; og R2 betegner eventuelt sub- stituert aryl. Forbindelsen (I) har en CCK-B-reseptorantagonisme og en virkning til å inhibere pentagastrin- stimulert magesekresjon og er således anvendbar ved behandling og forhind- ring av sykdommer hvori en CCK-B- reseptor og en gastrinreseptor deltar,A new benzodiazepine derivative represented by general formula (I) represents a pharmaceutically acceptable salt thereof, a pharmaceutical preparation thereof, and a process for its preparation. In formula (I), R 1 optionally represents substituted aryl, 5-membered monocyclic group, 6-membered monocyclic group or aromatic heterocyclic group comprising 5-membered and 6-membered rings; and R2 represents optionally substituted aryl. Compound (I) has a CCK-B receptor antagonism and an effect to inhibit pentagastrin-stimulated gastric secretion and is thus useful in the treatment and prevention of diseases in which a CCK-B receptor and a gastrin receptor participate.
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP41826390 | 1990-12-25 | ||
| JP11121691 | 1991-02-20 | ||
| JP28205691 | 1991-10-02 | ||
| PCT/JP1991/001720 WO1992011246A1 (en) | 1990-12-25 | 1991-12-17 | Novel benzodiazepine derivative |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO932325L true NO932325L (en) | 1993-06-24 |
| NO932325D0 NO932325D0 (en) | 1993-06-24 |
Family
ID=27467860
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO932325A NO932325D0 (en) | 1990-12-25 | 1993-06-24 | NEW BENZODIAZEPINE DERIVATIVES |
Country Status (1)
| Country | Link |
|---|---|
| NO (1) | NO932325D0 (en) |
-
1993
- 1993-06-24 NO NO932325A patent/NO932325D0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO932325D0 (en) | 1993-06-24 |
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