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NO904022D0 - Fremgangsmaate for fremstilling av nye n-aryl- og n-heteroarylamid- og -urinstoffderivater. - Google Patents

Fremgangsmaate for fremstilling av nye n-aryl- og n-heteroarylamid- og -urinstoffderivater.

Info

Publication number
NO904022D0
NO904022D0 NO904022A NO904022A NO904022D0 NO 904022 D0 NO904022 D0 NO 904022D0 NO 904022 A NO904022 A NO 904022A NO 904022 A NO904022 A NO 904022A NO 904022 D0 NO904022 D0 NO 904022D0
Authority
NO
Norway
Prior art keywords
heteroarylamide
aryl
procedure
preparation
new
Prior art date
Application number
NO904022A
Other languages
English (en)
Other versions
NO904022L (no
Inventor
Peter A Mccarthy
Frederick J Walker
Ernest Hamanaka
George Chang
Thien Truong
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO904022D0 publication Critical patent/NO904022D0/no
Publication of NO904022L publication Critical patent/NO904022L/no

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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/18—Halogen atoms or nitro radicals
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Plural Heterocyclic Compounds (AREA)
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NO90904022A 1989-09-15 1990-09-14 Fremgangsmaate for fremstilling av nye n-aryl- og n-heteroarylamid- og -urinstoffderivater. NO904022L (no)

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PCT/US1989/004033 WO1991004027A1 (en) 1989-09-15 1989-09-15 New n-aryl and n-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme a: cholesterol acyl transferase (acat)

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EP0418071A3 (en) 1992-03-25
CN1050183A (zh) 1991-03-27
ATE177082T1 (de) 1999-03-15
IL110321A0 (en) 1994-10-21
IL110324A0 (en) 1994-10-21
IL95610A0 (en) 1991-06-30
ES2071033T3 (es) 1995-06-16
AU652345B2 (en) 1994-08-25
JPH0825974B2 (ja) 1996-03-13
CA2025301C (en) 2001-10-16
EP0609960A1 (en) 1994-08-10
EP0418071A2 (en) 1991-03-20
DE69018908D1 (de) 1995-06-01
HU9302945D0 (en) 1993-12-28
DK0609960T3 (da) 1999-09-27
DE69018908T2 (de) 1995-08-24
KR910006233A (ko) 1991-04-27
ES2127878T3 (es) 1999-05-01
NO904022L (no) 1991-03-18
FI904537A0 (fi) 1990-09-14
MX22406A (es) 1994-01-31
PL291470A1 (en) 1992-07-13
PT95310B (pt) 1997-06-30
PL165357B1 (pl) 1994-12-30
FI111362B (fi) 2003-07-15
DE69032981T2 (de) 1999-07-08
KR930011303B1 (ko) 1993-11-29
PT95310A (pt) 1991-05-22
EP0418071B1 (en) 1995-04-26
AU6255390A (en) 1991-04-18
EG19358A (en) 1994-12-30
IE66324B1 (en) 1995-12-27
HUT70027A (en) 1995-09-28
DD298092A5 (de) 1992-02-06
EP0609960B1 (en) 1999-03-03
IE903336A1 (en) 1991-04-10
ATE121730T1 (de) 1995-05-15
PL291471A1 (en) 1992-06-26
WO1991004027A1 (en) 1991-04-04
CA2025301A1 (en) 1991-03-16
GR3029826T3 (en) 1999-06-30
PL291472A1 (en) 1992-07-13
ZA907346B (en) 1992-05-27
JPH03120243A (ja) 1991-05-22
PL165370B1 (pl) 1994-12-30
DE69032981D1 (de) 1999-04-08
DK0418071T3 (da) 1995-09-04
NZ235323A (en) 1993-02-25
IL95610A (en) 1994-12-29

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