NO893270L - PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TETRAHYDROPYRIDINE ACETIC ACID DERIVATIVES. - Google Patents
PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TETRAHYDROPYRIDINE ACETIC ACID DERIVATIVES.Info
- Publication number
- NO893270L NO893270L NO89893270A NO893270A NO893270L NO 893270 L NO893270 L NO 893270L NO 89893270 A NO89893270 A NO 89893270A NO 893270 A NO893270 A NO 893270A NO 893270 L NO893270 L NO 893270L
- Authority
- NO
- Norway
- Prior art keywords
- procedure
- preparation
- acetic acid
- acid derivatives
- therapeutic active
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
- C07D217/04—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/12—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
- C07D217/14—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
- C07D217/16—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Indole Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE3827727A DE3827727A1 (en) | 1988-08-16 | 1988-08-16 | ANALYZED TETRAHYDROPYRIDINE IGNESE DERIVATIVES, METHOD FOR THE PRODUCTION AND USE OF SUCH CONNECTIONS FOR CARDIRO PROTECTION |
Publications (2)
Publication Number | Publication Date |
---|---|
NO893270D0 NO893270D0 (en) | 1989-08-15 |
NO893270L true NO893270L (en) | 1990-02-19 |
Family
ID=6360928
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO89893270A NO893270L (en) | 1988-08-16 | 1989-08-15 | PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TETRAHYDROPYRIDINE ACETIC ACID DERIVATIVES. |
Country Status (16)
Country | Link |
---|---|
EP (1) | EP0358957A1 (en) |
JP (1) | JPH02160767A (en) |
KR (1) | KR900003129A (en) |
AU (1) | AU637767B2 (en) |
DD (3) | DD285595A5 (en) |
DE (1) | DE3827727A1 (en) |
DK (1) | DK399789A (en) |
FI (1) | FI893832A (en) |
HU (1) | HU208434B (en) |
IL (1) | IL91301A0 (en) |
NO (1) | NO893270L (en) |
PH (1) | PH27356A (en) |
PL (1) | PL161521B1 (en) |
PT (1) | PT91451A (en) |
YU (1) | YU160189A (en) |
ZA (1) | ZA896205B (en) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5162336A (en) * | 1990-06-21 | 1992-11-10 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Tetrahydro-pyrido-indoles as cholecystokinin and gastrin antagonists |
DE4041482A1 (en) * | 1990-12-22 | 1992-06-25 | Boehringer Ingelheim Kg | NEW PHARMACEUTICAL USE OF CARBOCYCLIC AND HETEROCYCLICALLY ANNELATED DIHYDROPYRIDINE |
DE4104257A1 (en) * | 1991-02-13 | 1992-08-20 | Boehringer Ingelheim Kg | USE OF ANALYZED TETRAHYDROPYRIDINE IGNESE DERIVATIVES FOR THE TREATMENT OF NEUROLOGICAL ILLNESSES |
US5674878A (en) * | 1992-06-22 | 1997-10-07 | Boehringer Ingelheim Kg | Anellated dihydropyridines and the use thereof for the production of pharmaceutical preparations |
KR100291706B1 (en) * | 1992-06-22 | 2001-10-24 | 베링거 인겔하임 카게 | Closed dihydropyridine, preparation method thereof and pharmaceutical composition comprising the same |
EP0620222A3 (en) * | 1993-04-14 | 1995-04-12 | Lilly Co Eli | Tetrahydro-beta-carbolines. |
DE4343641A1 (en) * | 1993-12-21 | 1995-06-29 | Boehringer Ingelheim Kg | Anellated dihydropyridines and their use for the preparation of pharmaceutical preparations |
DE4343683A1 (en) * | 1993-12-21 | 1995-06-22 | Boehringer Ingelheim Kg | Anellated dihydropyridines and their use for the preparation of pharmaceutical preparations |
DE59409595D1 (en) * | 1993-12-21 | 2000-12-28 | Boehringer Ingelheim Pharma | FELLED DIHYDROPYRIDINE AND THEIR USE FOR THE PRODUCTION OF PHARMACEUTICAL PREPARATIONS |
EP1159273A1 (en) | 1999-03-02 | 2001-12-05 | Boehringer Ingelheim Pharmaceuticals Inc. | Compounds useful as reversible inhibitors of cathepsin s |
US6420364B1 (en) | 1999-09-13 | 2002-07-16 | Boehringer Ingelheim Pharmaceuticals, Inc. | Compound useful as reversible inhibitors of cysteine proteases |
EP1458714A1 (en) * | 2001-12-19 | 2004-09-22 | H. Lundbeck A/S | 3,4-dihydro-1h-isoquinoloin-2-yl-derivatives |
GB2422828A (en) * | 2005-02-03 | 2006-08-09 | Hunter Fleming Ltd | Tricyclic cytoprotective compounds comprising an indole residue |
US8710245B2 (en) | 2009-12-04 | 2014-04-29 | Psychogenics Inc. | Multicyclic compounds and methods of use thereof |
CN116514761A (en) | 2016-07-29 | 2023-08-01 | 赛诺维信制药公司 | Compounds, compositions and uses thereof |
KR20190065246A (en) | 2016-07-29 | 2019-06-11 | 선오비온 파마슈티컬스 인코포레이티드 | Compounds and compositions and uses thereof |
IL268694B2 (en) | 2017-02-16 | 2023-10-01 | Sunovion Pharmaceuticals Inc | Treatment of schizophrenia |
JP7191085B2 (en) | 2017-08-02 | 2022-12-16 | サノビオン ファーマシューティカルズ インク | Isochroman compounds and uses thereof |
CN112135827B (en) | 2018-02-16 | 2024-01-12 | 赛诺维信制药公司 | Salts, crystal forms and preparation methods thereof |
EP3938045A1 (en) | 2019-03-14 | 2022-01-19 | Sunovion Pharmaceuticals Inc. | Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof |
MX2022012833A (en) | 2020-04-14 | 2022-11-07 | Sunovion Pharmaceuticals Inc | (s)-(4,5-dihydro-7h-thieno[2,3-c]pyran-7-yl)-n-methylmethanamine for treating neurological and psychiatric disorders. |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3021331A (en) * | 1959-07-20 | 1962-02-13 | Pfizer & Co C | Azabenzopyridocolines |
DE2361390A1 (en) * | 1973-12-10 | 1975-06-19 | Merck Patent Gmbh | ISOCHINOLINE DERIVATIVES AND THE PROCESS FOR THEIR PRODUCTION |
HU174697B (en) * | 1976-12-30 | 1980-03-28 | Chinoin Gyogyszer Es Vegyeszet | Process for producing new 6,7-dimethoxy-1,2,3,4-tetrahydro-1-isoquinolin-acetamide derivatives |
FR2447921A1 (en) * | 1979-02-05 | 1980-08-29 | Synthelabo | IMIDAZO AND PYRIMIDO-PYRIDO-INDOLES AND THEIR APPLICATION IN THERAPEUTICS |
FR2455044A1 (en) * | 1979-04-26 | 1980-11-21 | Synthelabo | PYRIDO-INDOLES AND THEIR APPLICATION IN THERAPEUTICS |
DE3013906A1 (en) * | 1980-04-11 | 1981-10-15 | C.H. Boehringer Sohn, 6507 Ingelheim | SUBSTITUTED (ALPHA) -AMINOCARBONYL-L-BENZYL-3,4-DIHYDRO-ISOCHINOLINE, METHOD FOR THE PRODUCTION AND USE THEREOF |
DE3229215A1 (en) * | 1982-08-05 | 1984-02-09 | Basf Ag, 6700 Ludwigshafen | 1- (HALOGENALKYL) -1,2,3,4-TETRAHYDRO-SS-CARBOLINE, THEIR PRODUCTION AND USE |
DE3309596A1 (en) * | 1982-08-05 | 1984-04-05 | Basf Ag, 6700 Ludwigshafen | 2-SUBSTITUTED 1- (3'-AMINOALKYL) -1,2,3,4-TETRAHYDRO-SS-CARBOLINE, THEIR PRODUCTION AND USE AS MEDICINAL PRODUCT |
DE3621413A1 (en) * | 1986-06-26 | 1988-01-07 | Boehringer Ingelheim Kg | USE OF CARBOCYCLIC AND HETEROCYCLICALLY FURNISHED DIHYDROPYRIDINE AS A CARDIOPROTECTIVE AGENT AND NEW HETEROCYCLIC AND CARBOCYCLICALLY FURNISHED DIHYDROPYRIDINE, METHOD FOR THE PRODUCTION THEREOF AND ITS ADDITIONAL PRODUCTS |
IL86131A0 (en) * | 1987-04-24 | 1988-11-15 | Boehringer Ingelheim Kg | Benzo-and thieno-3,4-dihydropyridine derivatives,their preparation and pharmaceutical compositions containing them |
-
1988
- 1988-08-16 DE DE3827727A patent/DE3827727A1/en not_active Ceased
-
1989
- 1989-08-11 EP EP89114943A patent/EP0358957A1/en not_active Withdrawn
- 1989-08-14 IL IL91301A patent/IL91301A0/en unknown
- 1989-08-14 PT PT91451A patent/PT91451A/en not_active Application Discontinuation
- 1989-08-14 KR KR1019890011572A patent/KR900003129A/en not_active Application Discontinuation
- 1989-08-15 JP JP1210567A patent/JPH02160767A/en active Pending
- 1989-08-15 ZA ZA896205A patent/ZA896205B/en unknown
- 1989-08-15 HU HU894200A patent/HU208434B/en not_active IP Right Cessation
- 1989-08-15 NO NO89893270A patent/NO893270L/en unknown
- 1989-08-15 DK DK399789A patent/DK399789A/en not_active Application Discontinuation
- 1989-08-15 YU YU160189A patent/YU160189A/en unknown
- 1989-08-15 FI FI893832A patent/FI893832A/en not_active Application Discontinuation
- 1989-08-16 DD DD89331836A patent/DD285595A5/en not_active IP Right Cessation
- 1989-08-16 PL PL89281066A patent/PL161521B1/en unknown
- 1989-08-16 DD DD89343927A patent/DD297640A5/en not_active IP Right Cessation
- 1989-08-16 DD DD89343928A patent/DD295379A5/en not_active IP Right Cessation
- 1989-08-16 AU AU39925/89A patent/AU637767B2/en not_active Withdrawn - After Issue
- 1989-08-16 PH PH39103A patent/PH27356A/en unknown
Also Published As
Publication number | Publication date |
---|---|
DD295379A5 (en) | 1991-10-31 |
DE3827727A1 (en) | 1990-02-22 |
AU637767B2 (en) | 1993-06-10 |
AU3992589A (en) | 1990-02-22 |
DD285595A5 (en) | 1990-12-19 |
DK399789D0 (en) | 1989-08-15 |
DD297640A5 (en) | 1992-01-16 |
HU208434B (en) | 1993-10-28 |
ZA896205B (en) | 1991-04-24 |
NO893270D0 (en) | 1989-08-15 |
DK399789A (en) | 1990-02-17 |
YU160189A (en) | 1992-09-07 |
IL91301A0 (en) | 1990-03-19 |
HUT51277A (en) | 1990-04-28 |
PH27356A (en) | 1993-06-22 |
KR900003129A (en) | 1990-03-23 |
PT91451A (en) | 1990-03-08 |
PL161521B1 (en) | 1993-07-30 |
FI893832A0 (en) | 1989-08-15 |
FI893832A (en) | 1990-02-17 |
JPH02160767A (en) | 1990-06-20 |
EP0358957A1 (en) | 1990-03-21 |
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