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NO20070502L - Azaindoles useful as inhibitors of protein kinases - Google Patents

Azaindoles useful as inhibitors of protein kinases

Info

Publication number
NO20070502L
NO20070502L NO20070502A NO20070502A NO20070502L NO 20070502 L NO20070502 L NO 20070502L NO 20070502 A NO20070502 A NO 20070502A NO 20070502 A NO20070502 A NO 20070502A NO 20070502 L NO20070502 L NO 20070502L
Authority
NO
Norway
Prior art keywords
inhibitors
protein kinases
azaindoles
useful
azaindoles useful
Prior art date
Application number
NO20070502A
Other languages
Norwegian (no)
Inventor
Michael Mortimore
Francoise Pierard
Juan-Miguel Jimenez
Ronald Kengtel
Guy Brenchley
Francesca Mazzei
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US11/098,751 external-priority patent/US7514448B2/en
Priority claimed from PCT/US2005/023429 external-priority patent/WO2006004984A1/en
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of NO20070502L publication Critical patent/NO20070502L/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)

Abstract

Foreliggende oppfinnelse vedrører azaindoler (I) som er nyttige som inhibitorer av proteinkinaser. Oppfinnelsen tilveiebringer også farmasøytisk akseptable sammensetninger omfattende nevnte forbindelser og metoder for å anvende sammensetningene i behandlingen av forskjellige sykdommer, tilstander eller forstyrrelser. Oppfinnelsen tilveiebringer også fremgangsmåter for å fremstille forbindelsene ifølge oppfinnelsen.The present invention relates to azaindoles (I) which are useful as inhibitors of protein kinases. The invention also provides pharmaceutically acceptable compositions comprising said compounds and methods for using the compositions in the treatment of various diseases, conditions or disorders. The invention also provides methods for preparing the compounds of the invention.

NO20070502A 2004-06-30 2007-01-26 Azaindoles useful as inhibitors of protein kinases NO20070502L (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US58438304P 2004-06-30 2004-06-30
US58472104P 2004-07-01 2004-07-01
US11/098,751 US7514448B2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
PCT/US2005/011358 WO2005103050A2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
PCT/US2005/023429 WO2006004984A1 (en) 2004-06-30 2005-06-29 Azaindoles useful as inhibitors of protein kinases

Publications (1)

Publication Number Publication Date
NO20070502L true NO20070502L (en) 2007-01-26

Family

ID=37801682

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20070502A NO20070502L (en) 2004-06-30 2007-01-26 Azaindoles useful as inhibitors of protein kinases

Country Status (4)

Country Link
JP (2) JP5122280B2 (en)
IL (1) IL180303A0 (en)
MX (1) MX2007000092A (en)
NO (1) NO20070502L (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5122280B2 (en) * 2004-06-30 2013-01-16 バーテックス ファーマシューティカルズ インコーポレイテッド Azaindoles useful as inhibitors of protein kinases
RU2007109073A (en) * 2004-08-13 2008-09-20 Дженентек, Инк. (Us) INHIBITORS FOR ATP-DEPENDENT ENZYM ON THE BASIS OF THIAZOL
DE102008038221A1 (en) * 2008-08-18 2010-02-25 Merck Patent Gmbh 7-azaindole derivatives
DE102009058280A1 (en) * 2009-12-14 2011-06-16 Merck Patent Gmbh thiazole
RU2603008C2 (en) 2010-04-16 2016-11-20 Ац Иммуне С.А. New compounds for treating diseases, associated with amyloid or amyloid-like proteins
MX2013000103A (en) * 2010-06-23 2013-06-13 Vertex Pharma Pyrrolo- pyrazine derivatives useful as inhibitors of atr kinase.
DE102011105469A1 (en) * 2011-06-24 2012-12-27 Merck Patent Gmbh 7-azaindole derivatives
JP6225178B2 (en) * 2012-05-31 2017-11-01 フェネックス ファーマシューティカルス アーゲー Carboxamide or sulfonamide substituted thiazoles and related derivatives as modulators of the orphan nuclear receptor RORγ
BR112016017981B1 (en) * 2014-02-04 2023-01-17 Taiho Pharmaceutical Co., Ltd. AZAINDOLA DERIVATIVE COMPOUNDS, JAK3 INHIBITOR, PHARMACEUTICAL COMPOSITION AND AGENT COMPRISING SAID COMPOUNDS, AND USE THEREOF TO TREAT A DISEASE INVOLVING JAK3
WO2023110843A1 (en) * 2021-12-15 2023-06-22 Almirall, S.A. Heterobicyclic derivatives as itk inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6265403B1 (en) * 1999-01-20 2001-07-24 Merck & Co., Inc. Angiogenesis inhibitors
JP2003525291A (en) * 2000-03-01 2003-08-26 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 2,4-disubstituted thiazolyl derivatives
SE0202463D0 (en) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel compounds
JP5019612B2 (en) * 2004-04-02 2012-09-05 バーテックス ファーマシューティカルズ インコーポレイテッド Azaindoles and other protein kinases useful as inhibitors of ROCK
JP5122280B2 (en) * 2004-06-30 2013-01-16 バーテックス ファーマシューティカルズ インコーポレイテッド Azaindoles useful as inhibitors of protein kinases

Also Published As

Publication number Publication date
MX2007000092A (en) 2007-03-07
IL180303A0 (en) 2007-06-03
JP2012012417A (en) 2012-01-19
JP2008513352A (en) 2008-05-01
JP5122280B2 (en) 2013-01-16

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