NO20035728D0 - Pyrrolopyrimidiner som proteinkinaseinhibitorer - Google Patents

Pyrrolopyrimidiner som proteinkinaseinhibitorer

Info

Publication number: NO20035728D0
Authority: NO; Norway
Prior art keywords: pyrrolopyrimidines; protein kinase; kinase inhibitors; inhibitors; protein
Prior art date: 2001-06-23

Application number

NO20035728A

Other languages

English (en)

Other versions

NO20035728L (no

Inventor

Paul Joseph Cox

Tahir Nadeem Majid

Shelley Amendola

Stephanie Daniele Deprets

Chris Edlin

Brian Leslie Pedgrift

Frank Halley

Michael Edwards

Bernard Baudoin

Lain Mcfarlane Mclay

Davis John Aldous

Original Assignee

Aventis Pharma Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-06-23

Filing date

2003-12-19

Publication date

2003-12-19

2001-06-23 Priority claimed from GBGB0115393.1A external-priority patent/GB0115393D0/en

2003-12-19 Application filed by Aventis Pharma Ltd filed Critical Aventis Pharma Ltd

2003-12-19 Publication of NO20035728D0 publication Critical patent/NO20035728D0/no

2004-02-23 Publication of NO20035728L publication Critical patent/NO20035728L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Immunology (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Otolaryngology (AREA)
Physical Education & Sports Medicine (AREA)
Cardiology (AREA)
Orthopedic Medicine & Surgery (AREA)
Heart & Thoracic Surgery (AREA)
Ophthalmology & Optometry (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Plural Heterocyclic Compounds (AREA)

NO20035728A 2001-06-23 2003-12-19 Pyrrolopyrimidiner som proteinkinaseinhibitorer NO20035728L (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GBGB0115393.1A GB0115393D0 (en)	2001-06-23	2001-06-23	Chemical compounds
US30167801P	2001-06-28	2001-06-28
PCT/GB2002/002835 WO2003000695A1 (en)	2001-06-23	2002-06-21	Pyrrolopyrimidines as protein kinase inhibitors

Publications (2)

Publication Number	Publication Date
NO20035728D0 true NO20035728D0 (no)	2003-12-19
NO20035728L NO20035728L (no)	2004-02-23

Family

ID=26246238

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20035728A NO20035728L (no)	2001-06-23	2003-12-19	Pyrrolopyrimidiner som proteinkinaseinhibitorer

Country Status (12)

Country	Link
US (1)	US7259154B2 (no)
KR (1)	KR100875380B1 (no)
AP (1)	AP2003002929A0 (no)
BG (1)	BG108453A (no)
CO (1)	CO5540313A2 (no)
CR (1)	CR7193A (no)
HK (1)	HK1068134A1 (no)
HR (1)	HRP20031049A2 (no)
IL (2)	IL159506A0 (no)
MA (1)	MA27129A1 (no)
MX (1)	MXPA03011998A (no)
NO (1)	NO20035728L (no)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TWI329105B (en)	2002-02-01	2010-08-21	Rigel Pharmaceuticals Inc	2,4-pyrimidinediamine compounds and their uses
MXPA05001096A (es)	2002-07-29	2005-11-23	Rigel Pharmaceuticals Inc	Metodos para tratamiento o prevencion de enfermedades autoinmunes con compuestos de 2,4-diamino-pirimidina.
CA2533377C (en) *	2003-07-30	2012-11-27	Rigel Pharmaceuticals, Inc.	Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds
US7465726B2 (en)	2004-08-02	2008-12-16	Osi Pharmaceuticals, Inc.	Substituted pyrrolo[2.3-B]pyridines
FR2878849B1 (fr) *	2004-12-06	2008-09-12	Aventis Pharma Sa	Indoles substitues, compositions les contenant, procede de fabrication et utilisation
JP2008543855A (ja)	2005-06-13	2008-12-04	ライジェルファーマシューティカルズ，インコーポレイテッド	変形性骨疾患を処置するための方法および組成物
DE602005000514T2 (de) *	2005-06-17	2007-10-25	Magneti Marelli Powertrain S.P.A.	Brennstoffeinspritzventil
PT1913000E (pt)	2005-07-29	2012-02-28	Pfizer Prod Inc	Derivados de pirrolo[2,3-d]pirimidina, suas substâncias intermédias e processo de síntese
US20070219183A1 (en) *	2006-03-17	2007-09-20	Wyeth	Dihydropyrazolo[1,5-A]pyrimidine and dihydroimidazo[1,5-A]pyrimidine derivatives and methods of use thereof
JP2011511005A (ja) *	2008-02-04	2011-04-07	オーエスアイ・フアーマスーテイカルズ・インコーポレーテツド	２−アミノピリジン系キナーゼ阻害薬
AR070317A1 (es) *	2008-02-06	2010-03-31	Osi Pharm Inc	Furo (3,2-c) piridina y tieno (3,2-c) piridinas
EP2356116A1 (en) *	2008-11-20	2011-08-17	OSI Pharmaceuticals, Inc.	Substituted pyrroloý2,3-b¨-pyridines and-pyrazines
AR081039A1 (es)	2010-05-14	2012-05-30	Osi Pharmaceuticals Llc	Inhibidores biciclicos fusionados de quinasa
EP2569315A1 (en)	2010-05-14	2013-03-20	OSI Pharmaceuticals, LLC	Fused bicyclic kinase inhibitors
JP2014513687A (ja)	2011-05-10	2014-06-05	メルク・シャープ・アンド・ドーム・コーポレーション	Ｓｙｋ阻害薬としてのピリジルアミノピリジン
JP2014513686A (ja)	2011-05-10	2014-06-05	メルク・シャープ・アンド・ドーム・コーポレーション	Ｓｙｋ阻害薬としてのアミノピリミジン
US9145391B2 (en)	2011-05-10	2015-09-29	Merck Sharp & Dohme Corp.	Bipyridylaminopyridines as Syk inhibitors
US9216173B2 (en)	2011-10-05	2015-12-22	Merck Sharp & Dohme Corp.	2-Pyridyl carboxamide-containing spleen tyrosine kinase (SYK) inhibitors
WO2013052391A1 (en)	2011-10-05	2013-04-11	Merck Sharp & Dohme Corp.	PHENYL CARBOXAMIDE-CONTAINING SPLEEN TYROSINE KINASE (Syk) INHIBITORS
WO2013052393A1 (en)	2011-10-05	2013-04-11	Merck Sharp & Dohme Corp.	3-PYRIDYL CARBOXAMIDE-CONTAINING SPLEEN TYROSINE KINASE (Syk) INHIBITORS
US9242984B2 (en)	2012-06-20	2016-01-26	Merck Sharp & Dohme Corp.	Pyrazolyl derivatives as Syk inhibitors
EP2863913B1 (en)	2012-06-20	2018-09-12	Merck Sharp & Dohme Corp.	Imidazolyl analogs as syk inhibitors
EP2863915B1 (en)	2012-06-22	2017-12-06	Merck Sharp & Dohme Corp.	SUBSTITUTED DIAZINE AND TRIAZINE SPLEEN TYROSINE KINASE (Syk) INHIBITORS
WO2013192098A1 (en)	2012-06-22	2013-12-27	Merck Sharp & Dohme Corp.	SUBSTITUTED PYRIDINE SPLEEN TYROSINE KINASE (Syk) INHIBITORS
EP2884982B1 (en)	2012-08-20	2017-09-20	Merck Sharp & Dohme Corp.	SUBSTITUTED PHENYL SPLEEN TYROSINE KINASE (Syk) INHIBITORS
US9586931B2 (en)	2012-09-28	2017-03-07	Merck Sharp & Dohme Corp.	Triazolyl derivatives as Syk inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PT888349E (pt)	1996-01-23	2002-10-31	Novartis Ag	Pirrolopirimidinas e processos para a sua preparacao
HUP0001507A3 (en)	1997-03-19	2002-01-28	Abbott Gmbh & Co Kg	Pyrrolo [2,3-d] pyrimidine derivatives, process for their preparation, their use and pharmaceutical compositions containing them
PA8474101A1 (es)	1998-06-19	2000-09-29	Pfizer Prod Inc	Compuestos de pirrolo [2,3-d] pirimidina
ES2208433T3 (es)	1999-12-10	2004-06-16	Pfizer Products Inc.	Compuestos de pirrolo(2,3-d)pirimidina como inhibidores de proteina quinasas.

2002
- 2002-06-21 MX MXPA03011998A patent/MXPA03011998A/es active IP Right Grant
- 2002-06-21 AP APAP/P/2003/002929A patent/AP2003002929A0/en unknown
- 2002-06-21 KR KR1020037016809A patent/KR100875380B1/ko not_active IP Right Cessation
- 2002-06-21 IL IL15950602A patent/IL159506A0/xx unknown
2003
- 2003-12-10 CR CR7193A patent/CR7193A/es unknown
- 2003-12-15 BG BG108453A patent/BG108453A/bg unknown
- 2003-12-16 MA MA27444A patent/MA27129A1/fr unknown
- 2003-12-17 HR HR20031049A patent/HRP20031049A2/hr not_active Application Discontinuation
- 2003-12-19 NO NO20035728A patent/NO20035728L/no not_active Application Discontinuation
- 2003-12-22 CO CO03111600A patent/CO5540313A2/es not_active Application Discontinuation
- 2003-12-22 IL IL159506A patent/IL159506A/en not_active IP Right Cessation
- 2003-12-23 US US10/744,478 patent/US7259154B2/en not_active Expired - Fee Related
2005
- 2005-01-10 HK HK05100184A patent/HK1068134A1/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
CO5540313A2 (es)	2005-07-29
KR100875380B1 (ko)	2008-12-23
AP2003002929A0 (en)	2003-12-31
IL159506A0 (en)	2004-06-01
KR20040019317A (ko)	2004-03-05
IL159506A (en)	2011-12-29
MA27129A1 (fr)	2005-01-03
BG108453A (bg)	2004-12-30
HRP20031049A2 (en)	2004-06-30
CR7193A (es)	2004-11-23
NO20035728L (no)	2004-02-23
HK1068134A1 (en)	2005-04-22
US7259154B2 (en)	2007-08-21
US20040142947A1 (en)	2004-07-22
MXPA03011998A (es)	2005-07-01

Publication	Publication Date	Title
NO20041887L (no)	2004-05-07	Benzomidazoler anvendelige som proteinkinase-inhibitorer
NO20035728L (no)	2004-02-23	Pyrrolopyrimidiner som proteinkinaseinhibitorer
EE200400003A (et)	2004-02-16	Pürrolopürimidiinid kui valgukinaasi inhibiitorid
NO20011356D0 (no)	2001-03-16	Pyrrolopyrimidiner som proteinkinase-inhibitorer
NO20032704L (no)	2003-08-21	Pyrazolforbindelser nyttige som proteinkinaseinhibitorer
NO20031191D0 (no)	2003-03-14	Pyrazolforbindelser nyttige som proteinkinaseinhibitorer
DK1337527T3 (da)	2010-01-04	Indolylmaleinimidderivater som proteinkinase C-inhibitorer
AU2003254053A8 (en)	2004-02-09	Pyrazolopyrimidines as protein kinase inhibitors
NO20021239L (no)	2002-03-13	Pteridinoner som kinase-inhibitorer
NO20023828L (no)	2002-09-30	Pyrimidin-4-on derivater som LDL-PLA2 inhibitorer
ATE505471T1 (de)	2011-04-15	Azaindol-kinaseinhibitoren
ID30460A (id)	2001-12-06	Inhibitor-inhibitor protein siklik tirosin kinase
DE60234125D1 (de)	2009-12-03	E inhibitoren
NO20023713D0 (no)	2002-08-06	2-benzotiazolyl-urea-derivater samt anvendelse derav som proteinkinaseinhibitorer
NO20011574D0 (no)	2001-03-28	Substituerte 3-cyanokinoliner som proteintyrosin-kinsase- inhibitorer
DK1140840T3 (da)	2006-07-31	omega-carboxyaryl-substituerede diphenylurinstoffer som raf-kinase-inhibitorer
ATE255114T1 (de)	2003-12-15	Tricyclische proteinkinasehemmer
DK1317448T4 (da)	2011-05-30	Pyrazolforbindelser anvendelige som proteinkinaseinhibitorer
NO20015301D0 (no)	2001-10-30	Liv-In Boenheter
ATA8102001A (de)	2002-05-15	Sitzmöbel
ITBA20010050A0 (it)	2001-10-12	Arpione
SE0104413D0 (sv)	2001-12-21	New protein

Legal Events

Date	Code	Title	Description
2010-09-27	FC2A	Withdrawal, rejection or dismissal of laid open patent application