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NO173827C - Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazokinoxaliner - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazokinoxaliner

Info

Publication number
NO173827C
NO173827C NO894474A NO894474A NO173827C NO 173827 C NO173827 C NO 173827C NO 894474 A NO894474 A NO 894474A NO 894474 A NO894474 A NO 894474A NO 173827 C NO173827 C NO 173827C
Authority
NO
Norway
Prior art keywords
imidazoquinoxalins
preparation
therapeutically active
analogous procedures
novel
Prior art date
Application number
NO894474A
Other languages
English (en)
Other versions
NO173827B (no
NO894474D0 (no
NO894474L (no
Inventor
Frank Waetjen
Holger Claus Hansen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of NO894474D0 publication Critical patent/NO894474D0/no
Publication of NO894474L publication Critical patent/NO894474L/no
Publication of NO173827B publication Critical patent/NO173827B/no
Publication of NO173827C publication Critical patent/NO173827C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO894474A 1988-11-10 1989-11-09 Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazokinoxaliner NO173827C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK626288A DK626288D0 (da) 1988-11-10 1988-11-10 Kemisk proces til fremstilling af imidazoquinoxaliner og mellemprodukter til brug i processen

Publications (4)

Publication Number Publication Date
NO894474D0 NO894474D0 (no) 1989-11-09
NO894474L NO894474L (no) 1990-05-11
NO173827B NO173827B (no) 1993-11-01
NO173827C true NO173827C (no) 1994-02-09

Family

ID=8148369

Family Applications (1)

Application Number Title Priority Date Filing Date
NO894474A NO173827C (no) 1988-11-10 1989-11-09 Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazokinoxaliner

Country Status (17)

Country Link
US (1) US4999353A (no)
EP (1) EP0368652B1 (no)
JP (1) JPH02178285A (no)
AT (1) ATE119162T1 (no)
AU (1) AU622941B2 (no)
CA (1) CA2002624A1 (no)
DE (1) DE68921418T2 (no)
DK (1) DK626288D0 (no)
ES (1) ES2068903T3 (no)
FI (1) FI92931C (no)
GR (1) GR3015718T3 (no)
IE (1) IE68939B1 (no)
IL (1) IL92055A (no)
NO (1) NO173827C (no)
NZ (1) NZ231321A (no)
PT (1) PT92279B (no)
ZA (1) ZA898051B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK588489D0 (da) * 1989-11-22 1989-11-22 Ferrosan As Heterocykliske forbindelser, deres fremstilling og anvendelse
JP3147902B2 (ja) * 1991-06-14 2001-03-19 ファルマシア・アンド・アップジョン・カンパニー イミダゾ〔1,5−a〕キノキサリン
WO1993012113A1 (en) * 1991-12-17 1993-06-24 The Upjohn Company 3-SUBSTITUTED IMIDAZO (1,5-a) AND IMIDAZO (1,5-a)-TRIAZOLO (1,5-c) QUINOXALINES AND QUINAZOLINES WITH CNS ACTIVITY
DE4228095A1 (de) * 1992-08-24 1994-03-03 Asta Medica Ag Neue 4,5-Dihydro-4-oxo-pyrrolo[1,2-a]chinoxaline und entsprechende Aza-analoga und Verfahren zu deren Herstellung
FR2696466B1 (fr) * 1992-10-02 1994-11-25 Rhone Poulenc Rorer Sa Dérivés de 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, leur préparation et les médicaments les contenant.
US5792766A (en) * 1996-03-13 1998-08-11 Neurogen Corporation Imidazo 1,5-c! quinazolines; a new class of GABA brain receptor ligands
JP4042925B2 (ja) * 1996-11-20 2008-02-06 シスメックス株式会社 幼若白血球の分類計数法
US20040180898A1 (en) * 2003-03-03 2004-09-16 Bang-Chi Chen Processes for preparing imidazoquinoxalinones, heterocyclic-substituted imidazopyrazinones, imidazoquinoxalines and heterocyclic-substituted imidazopyrazines
JP6964343B2 (ja) 2015-11-20 2021-11-10 フォーマ セラピューティクス,インコーポレイテッド ユビキチン特異的プロテアーゼ1阻害剤としてのプリノン

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4440929A (en) * 1981-07-16 1984-04-03 Usv Pharmaceutical Corporation Imidazoquinoxaline compounds
DK476885D0 (da) * 1985-10-17 1985-10-17 Ferrosan As Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf
ATE80392T1 (de) * 1985-10-17 1992-09-15 Novo Nordisk As Oxadiazolylacetonitrile, ihre herstellung und anwendung.
DK155524C (da) * 1987-03-18 1989-09-11 Ferrosan As Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse
DK160876C (da) * 1987-12-08 1991-10-14 Novo Nordisk As Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar
IL90315A0 (en) * 1988-06-01 1989-12-15 Ferrosan As Imidazoquinoxaline compounds,their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
DK626288D0 (da) 1988-11-10
IL92055A0 (en) 1990-07-12
NZ231321A (en) 1991-10-25
NO173827B (no) 1993-11-01
FI92931B (fi) 1994-10-14
ZA898051B (en) 1990-08-29
ES2068903T3 (es) 1995-05-01
US4999353A (en) 1991-03-12
JPH02178285A (ja) 1990-07-11
FI895257A0 (fi) 1989-11-06
IL92055A (en) 1994-01-25
IE68939B1 (en) 1996-07-24
CA2002624A1 (en) 1990-05-10
FI92931C (fi) 1995-01-25
NO894474D0 (no) 1989-11-09
EP0368652B1 (en) 1995-03-01
PT92279B (pt) 1995-08-09
NO894474L (no) 1990-05-11
ATE119162T1 (de) 1995-03-15
AU4439389A (en) 1990-05-17
EP0368652A1 (en) 1990-05-16
DE68921418D1 (de) 1995-04-06
AU622941B2 (en) 1992-04-30
DE68921418T2 (de) 1995-07-13
PT92279A (pt) 1990-05-31
IE893374L (en) 1990-05-10
GR3015718T3 (en) 1995-07-31

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