NO161497C - Analogifremgangsmaate for fremstilling av terapeutisk aktive 9a-aza-9a-homoerytromycin-derivater. - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive 9a-aza-9a-homoerytromycin-derivater.

Info

Publication number: NO161497C
Authority: NO; Norway
Prior art keywords: homoerytromycin; aza; derivatives; preparation; therapeutic active
Prior art date: 1984-04-13

Application number

NO851466A

Other languages

English (en)

Other versions

NO851466L (no

NO161497B (no

Inventor

James Robert Hauske

Arthur Adam Nagel

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-04-13

Filing date

1985-04-12

Publication date

1989-08-23

1984-04-13 Priority claimed from US06/600,252 external-priority patent/US4512982A/en

1985-04-12 Application filed by Pfizer filed Critical Pfizer

1985-10-14 Publication of NO851466L publication Critical patent/NO851466L/no

1989-05-16 Publication of NO161497B publication Critical patent/NO161497B/no

1989-08-23 Publication of NO161497C publication Critical patent/NO161497C/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Health & Medical Sciences (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

NO851466A 1984-04-13 1985-04-12 Analogifremgangsmaate for fremstilling av terapeutisk aktive 9a-aza-9a-homoerytromycin-derivater. NO161497C (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US06/600,252 US4512982A (en)	1984-04-13	1984-04-13	9α-Aza-9α-homoerythromycin compounds, pharmaceutical composition and therapeutic method
US06/616,529 US4518590A (en)	1984-04-13	1984-06-04	9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method

Publications (3)

Publication Number	Publication Date
NO851466L NO851466L (no)	1985-10-14
NO161497B NO161497B (no)	1989-05-16
NO161497C true NO161497C (no)	1989-08-23

Family

ID=27083554

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO851466A NO161497C (no)	1984-04-13	1985-04-12	Analogifremgangsmaate for fremstilling av terapeutisk aktive 9a-aza-9a-homoerytromycin-derivater.

Country Status (19)

Country	Link
US (1)	US4518590A (no)
EP (1)	EP0159856B1 (no)
KR (1)	KR860002111B1 (no)
AU (1)	AU549235B2 (no)
CA (1)	CA1234805A (no)
DE (1)	DE3565267D1 (no)
DK (1)	DK164785A (no)
EG (1)	EG17459A (no)
ES (3)	ES8607335A1 (no)
FI (1)	FI851449L (no)
GR (1)	GR850900B (no)
HU (1)	HU195668B (no)
IE (1)	IE57739B1 (no)
IL (1)	IL74865A (no)
NO (1)	NO161497C (no)
NZ (1)	NZ211769A (no)
PH (1)	PH21185A (no)
PT (1)	PT80270B (no)
YU (3)	YU62385A (no)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5075289A (en) *	1988-06-07	1991-12-24	Abbott Laboratories	9-r-azacyclic erythromycin antibiotics
US4904644A (en) *	1988-08-03	1990-02-27	Schering Corporation	Antimicrobial compound isolated from Actinomadura fulva subsp indica
EP0503932B1 (en)	1991-03-15	1998-12-02	Merck & Co. Inc.	9-Deoxo-9(z)-hydroxy-iminoerythromycin A and O-derivatives thereof
US5912331A (en) *	1991-03-15	1999-06-15	Merck & Co., Inc.	Process for the preparation of 9-deoxo-9(Z)-hydroxyiminoerythromycin A
US5985844A (en) *	1992-03-26	1999-11-16	Merck & Co., Inc.	Homoerythromycin A derivatives modified at the 4"-and 8A-positions
AU663089B2 (en) *	1991-04-09	1995-09-28	Abbott Laboratories	Macrocyclic lactam prokinetic agents
US5189159A (en) *	1992-04-02	1993-02-23	Merck & Co., Inc.	8a-AZA-8a-homoerythromycin cyclic iminoethers
US5523399A (en) *	1991-12-27	1996-06-04	Taisho Pharmaceutical Co., Ltd.	5-O-desosaminylerythronolide derivatives
US5215980A (en) *	1992-01-17	1993-06-01	Merck & Co., Inc.	10-AZA-9-deoxo-11-deoxy-erythromycin A and derivatives thereof
US5210235A (en) *	1992-08-26	1993-05-11	Merck & Co., Inc.	Methods of elaborating erythromycin fragments into amine-containing fragments of azalide antibiotics
US5332807A (en) *	1993-04-14	1994-07-26	Merck & Co., Inc.	Process of producing 8A- and 9A-azalide antibiotics
WO1994026758A1 (en) *	1993-05-19	1994-11-24	Pfizer Inc.	Intermediate for azithromycin
US5441939A (en) *	1994-03-04	1995-08-15	Pfizer Inc.	3"-desmethoxy derivatives of erythromycin and azithromycin
FR2739620B1 (fr) *	1995-10-09	1997-12-19	Roussel Uclaf	Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
USRE38426E1 (en) *	1995-10-09	2004-02-10	Aventis Pharma S.A.	5-O-deosaminyl 6-O-methyl erythronolide A derivatives, preparation method therefor and use thereof for preparing biologically active materials
ATE306491T1 (de) *	2000-08-23	2005-10-15	Wockhardt Ltd	Verfahren zur herstellung von wasserfreiem azithromycin
JP4104463B2 (ja)	2001-04-27	2008-06-18	ファイザー・プロダクツ・インク	４’’−置換された−９−デオキソ−９ａ−アザ−９ａ−ホモエリスロマイシン誘導体を製造するための方法
WO2003070173A2 (en)	2002-02-15	2003-08-28	Sympore Gmbh	Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
AU2003211113B2 (en)	2002-02-15	2007-08-09	Merckle Gmbh	Antibiotic conjugates
US20050171342A1 (en)	2002-02-15	2005-08-04	Michael Burnet	Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
GB0310992D0 (en) *	2003-05-13	2003-06-18	Glaxo Group Ltd	Novel compounds
US7468428B2 (en) *	2004-03-17	2008-12-23	App Pharmaceuticals, Llc	Lyophilized azithromycin formulation
US20060116336A1 (en) *	2004-03-17	2006-06-01	American Pharmaceutical Partners, Inc.	Lyophilized azithromycin formulation

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4150220A (en) *	1977-02-04	1979-04-17	Pfizer Inc.	Semi-synthetic 4"-erythromycin A derivatives
SE445223B (sv) *	1977-02-04	1986-06-09	Pfizer	Sett att framstella 4"-amino-erytomylin-a-derivat
US4180654A (en) *	1978-01-03	1979-12-25	Pfizer Inc.	4"-Deoxy-4"-acylamido derivatives of oleandomycin, erythromycin and erythromycin carbonate
YU43116B (en) *	1979-04-02	1989-04-30	Pliva Pharm & Chem Works	Process for preparing 11-aza-4-o-cladinosyl-6-o-desosaminyl-15-ethyl-7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl-oxacyclopentadecane-2-one(11-aza-10-deox
YU43006B (en) *	1981-03-06	1989-02-28	Pliva Pharm & Chem Works	Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof
US4474768A (en) *	1982-07-19	1984-10-02	Pfizer Inc.	N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
US4465674A (en) *	1983-09-06	1984-08-14	Pfizer Inc.	Azahomoerythromycin D derivative and intermediates therefor

1984
- 1984-06-04 US US06/616,529 patent/US4518590A/en not_active Expired - Lifetime
1985
- 1985-04-09 GR GR850900A patent/GR850900B/el not_active IP Right Cessation
- 1985-04-10 IL IL74865A patent/IL74865A/xx not_active IP Right Cessation
- 1985-04-10 DE DE8585302507T patent/DE3565267D1/de not_active Expired
- 1985-04-10 EP EP85302507A patent/EP0159856B1/en not_active Expired
- 1985-04-11 ES ES542134A patent/ES8607335A1/es not_active Expired
- 1985-04-11 FI FI851449A patent/FI851449L/fi not_active Application Discontinuation
- 1985-04-11 EG EG239/85A patent/EG17459A/xx active
- 1985-04-11 IE IE912/85A patent/IE57739B1/en not_active IP Right Cessation
- 1985-04-11 PT PT80270A patent/PT80270B/pt not_active IP Right Cessation
- 1985-04-11 PH PH32123A patent/PH21185A/en unknown
- 1985-04-11 CA CA000478792A patent/CA1234805A/en not_active Expired
- 1985-04-12 YU YU00623/85A patent/YU62385A/xx unknown
- 1985-04-12 HU HU851370A patent/HU195668B/hu not_active IP Right Cessation
- 1985-04-12 NZ NZ211769A patent/NZ211769A/en unknown
- 1985-04-12 NO NO851466A patent/NO161497C/no not_active IP Right Cessation
- 1985-04-12 AU AU41070/85A patent/AU549235B2/en not_active Ceased
- 1985-04-12 DK DK164785A patent/DK164785A/da not_active IP Right Cessation
- 1985-04-12 KR KR1019850002453A patent/KR860002111B1/ko not_active IP Right Cessation
1986
- 1986-01-31 ES ES551503A patent/ES8704965A1/es not_active Expired
- 1986-01-31 ES ES551502A patent/ES8705458A1/es not_active Expired
1987
- 1987-07-06 YU YU01268/87A patent/YU126887A/xx unknown
- 1987-07-06 YU YU01267/87A patent/YU126787A/xx unknown

Also Published As

Publication number	Publication date
YU126787A (en)	1988-02-29
HU195668B (en)	1988-06-28
EP0159856B1 (en)	1988-09-28
IE57739B1 (en)	1993-03-24
FI851449L (fi)	1985-10-14
IL74865A (en)	1987-12-31
IE850912L (en)	1985-10-13
HUT37629A (en)	1986-01-23
EP0159856A2 (en)	1985-10-30
PH21185A (en)	1987-08-12
US4518590A (en)	1985-05-21
ES8704965A1 (es)	1987-04-16
IL74865A0 (en)	1985-07-31
DK164785D0 (da)	1985-04-12
ES551502A0 (es)	1987-05-01
NO851466L (no)	1985-10-14
DE3565267D1 (en)	1988-11-03
AU549235B2 (en)	1986-01-23
FI851449A0 (fi)	1985-04-11
KR850007435A (ko)	1985-12-04
EP0159856A3 (en)	1986-03-19
DK164785A (da)	1985-12-10
KR860002111B1 (ko)	1986-11-26
CA1234805A (en)	1988-04-05
YU126887A (en)	1988-02-29
PT80270A (en)	1985-05-01
ES542134A0 (es)	1986-06-16
PT80270B (pt)	1987-10-20
ES8607335A1 (es)	1986-06-16
GR850900B (no)	1985-11-25
ES551503A0 (es)	1987-04-16
NZ211769A (en)	1987-10-30
AU4107085A (en)	1985-10-17
YU62385A (en)	1988-02-29
NO161497B (no)	1989-05-16
ES8705458A1 (es)	1987-05-01
EG17459A (en)	1992-12-30

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Legal Events

Date	Code	Title	Description
2004-12-27	MM1K	Lapsed by not paying the annual fees