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NO152607C - OUTSTANDING MATERIALS FOR USE IN THE PREPARATION OF THERAPEUTIC ACTIVE PYRIMIDINE DERIVATIVES - Google Patents

OUTSTANDING MATERIALS FOR USE IN THE PREPARATION OF THERAPEUTIC ACTIVE PYRIMIDINE DERIVATIVES

Info

Publication number
NO152607C
NO152607C NO801378A NO801378A NO152607C NO 152607 C NO152607 C NO 152607C NO 801378 A NO801378 A NO 801378A NO 801378 A NO801378 A NO 801378A NO 152607 C NO152607 C NO 152607C
Authority
NO
Norway
Prior art keywords
preparation
pyrimidine derivatives
therapeutic active
active pyrimidine
outstanding materials
Prior art date
Application number
NO801378A
Other languages
Norwegian (no)
Other versions
NO152607B (en
NO801378L (en
Inventor
Istvan Hermecz
Tibor Breining
Lelle Vasvari
Agnes Horvath
Zoltan Meszaros
Istvan Bitter
Jozsef Koekoesi
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of NO801378L publication Critical patent/NO801378L/en
Publication of NO152607B publication Critical patent/NO152607B/en
Publication of NO152607C publication Critical patent/NO152607C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09BORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
    • C09B62/00Reactive dyes, i.e. dyes which form covalent bonds with the substrates or which polymerise with themselves

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
NO801378A 1979-05-11 1980-05-09 OUTSTANDING MATERIALS FOR USE IN THE PREPARATION OF THERAPEUTIC ACTIVE PYRIMIDINE DERIVATIVES NO152607C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU79CI1932A HU179443B (en) 1979-05-11 1979-05-11 Process for producing substituted geminal dihalogeno-derivatives of pyrido-square bracket-1,2-a-square closed-pyrimidines,pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines and pyrimido-square bracket-1,2,-a-square bracket closed-asepines

Publications (3)

Publication Number Publication Date
NO801378L NO801378L (en) 1980-11-12
NO152607B NO152607B (en) 1985-07-15
NO152607C true NO152607C (en) 1985-10-23

Family

ID=10994747

Family Applications (1)

Application Number Title Priority Date Filing Date
NO801378A NO152607C (en) 1979-05-11 1980-05-09 OUTSTANDING MATERIALS FOR USE IN THE PREPARATION OF THERAPEUTIC ACTIVE PYRIMIDINE DERIVATIVES

Country Status (24)

Country Link
JP (1) JPS5615286A (en)
AT (1) AT377261B (en)
BE (1) BE883217A (en)
CA (1) CA1141379A (en)
CH (1) CH646971A5 (en)
CS (1) CS241025B2 (en)
DD (1) DD150605A5 (en)
DE (1) DE3017564A1 (en)
DK (1) DK204680A (en)
ES (1) ES491896A0 (en)
FI (1) FI68825C (en)
FR (1) FR2456101A1 (en)
GB (1) GB2051048B (en)
GR (1) GR68518B (en)
HU (1) HU179443B (en)
IL (1) IL59967A (en)
IT (1) IT1133085B (en)
LU (1) LU82437A1 (en)
NL (1) NL8002678A (en)
NO (1) NO152607C (en)
PL (1) PL124035B1 (en)
PT (1) PT71213A (en)
SE (1) SE441747B (en)
SU (1) SU1151210A3 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU178453B (en) * 1979-05-11 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydrazino-4-oxo-6,7,8,9-tetrahydro-4h-p-pyrido-square bracket-1,2-a-square bracket closed-pyrimidine derivatives
US4395549A (en) 1981-10-02 1983-07-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
US5158952A (en) * 1988-11-07 1992-10-27 Janssen Pharmaceutica N.V. 3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use
UA72189C2 (en) 1997-11-17 2005-02-15 Янссен Фармацевтика Н.В. Aqueous suspensions of 9-hydroxy-risperidone fatty acid esters provided in submicron form

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT299212B (en) * 1966-11-02 1972-06-12 Chinoin Gyogyszer Es Vegyeszet Process for the preparation of new homopyrimidazole derivatives and their salts
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity

Also Published As

Publication number Publication date
FI68825B (en) 1985-07-31
FR2456101B1 (en) 1985-04-05
SE8003479L (en) 1980-11-12
CH646971A5 (en) 1984-12-28
PL124035B1 (en) 1982-12-31
GR68518B (en) 1982-01-11
GB2051048B (en) 1983-01-19
JPS5615286A (en) 1981-02-14
CS325880A2 (en) 1985-06-13
PT71213A (en) 1980-06-01
FI801512A (en) 1980-11-12
NO152607B (en) 1985-07-15
SU1151210A3 (en) 1985-04-15
PL224163A1 (en) 1981-02-13
FI68825C (en) 1985-11-11
BE883217A (en) 1980-09-01
ES8102570A1 (en) 1981-02-16
IT8067719A0 (en) 1980-05-09
SE441747B (en) 1985-11-04
DK204680A (en) 1980-11-12
GB2051048A (en) 1981-01-14
LU82437A1 (en) 1980-07-31
AT377261B (en) 1985-02-25
CS241025B2 (en) 1986-03-13
DE3017564A1 (en) 1980-11-13
HU179443B (en) 1982-10-28
ES491896A0 (en) 1981-02-16
DD150605A5 (en) 1981-09-09
NO801378L (en) 1980-11-12
IT1133085B (en) 1986-07-09
IL59967A (en) 1984-05-31
ATA247580A (en) 1984-07-15
CA1141379A (en) 1983-02-15
NL8002678A (en) 1980-11-13
IL59967A0 (en) 1980-07-31
FR2456101A1 (en) 1980-12-05

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