NL8104938A - 1.1-dioxopenicillanoyloxymethyl-6-(d-alfa-amino-alfa-fenylaceetamido)penicillanaat, werkwijze voor de bereiding en toepassing daarvan. - Google Patents

1.1-dioxopenicillanoyloxymethyl-6-(d-alfa-amino-alfa-fenylaceetamido)penicillanaat, werkwijze voor de bereiding en toepassing daarvan. Download PDF

Info

Publication number: NL8104938A
Authority: NL; Netherlands
Prior art keywords: tosylate; compound; preparation; amino; compound according
Prior art date: 1980-10-31

Application number

NL8104938A

Other languages

English (en)

Dutch (nl)

Original Assignee

Leo Pharm Prod Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1980-10-31

Filing date

1981-10-30

Publication date

1982-05-17

1981-10-30 Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd

1982-05-17 Publication of NL8104938A publication Critical patent/NL8104938A/nl

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

NL8104938A 1980-10-31 1981-10-30 1.1-dioxopenicillanoyloxymethyl-6-(d-alfa-amino-alfa-fenylaceetamido)penicillanaat, werkwijze voor de bereiding en toepassing daarvan. NL8104938A (nl)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB8035156		1980-10-31
GB8035156		1980-10-31

Publications (1)

Publication Number	Publication Date
NL8104938A true NL8104938A (nl)	1982-05-17

Family

ID=10517019

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NL8104938A NL8104938A (nl)	1980-10-31	1981-10-30	1.1-dioxopenicillanoyloxymethyl-6-(d-alfa-amino-alfa-fenylaceetamido)penicillanaat, werkwijze voor de bereiding en toepassing daarvan.

Country Status (26)

Country	Link
US (1)	US4831025A (fr)
JP (1)	JPS57126493A (fr)
KR (1)	KR870001982B1 (fr)
AT (1)	AT373893B (fr)
AU (1)	AU543870B2 (fr)
BE (1)	BE890938A (fr)
CA (1)	CA1180696A (fr)
CH (1)	CH647527A5 (fr)
DE (1)	DE3143219A1 (fr)
DK (1)	DK154219C (fr)
ES (1)	ES506751A0 (fr)
FI (1)	FI813331L (fr)
FR (1)	FR2493322B1 (fr)
GB (1)	GB2114969B (fr)
GR (1)	GR75369B (fr)
IE (1)	IE51640B1 (fr)
IL (1)	IL64009A (fr)
IT (1)	IT1193735B (fr)
LU (1)	LU83727A1 (fr)
NL (1)	NL8104938A (fr)
NO (1)	NO813683L (fr)
NZ (1)	NZ198622A (fr)
PH (1)	PH17820A (fr)
PT (1)	PT73913B (fr)
SE (1)	SE452322B (fr)
ZA (1)	ZA817091B (fr)

Families Citing this family (43)

* Cited by examiner, † Cited by third party
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US4432987A (en) *	1982-04-23	1984-02-21	Pfizer Inc.	Crystalline benzenesulfonate salts of sultamicillin
PH20068A (en) *	1982-12-06	1986-09-18	Pfizer	Process and intermediates for sultamicillin and analogs
KR910009271B1 (ko) *	1989-06-20	1991-11-08	김영설	1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
ES2161602B1 (es) *	1999-04-08	2003-02-16	Asturpharma S A	Sintesis de 6-(d-alfa-(bencilidenaminofenilacetamido))penicilanato de 1,1-dioxopenicilanoiloximetilo y analogos. nuevos intermedios para la sintesis de sultamicilina.
US6638532B2 (en)	2000-02-24	2003-10-28	Advancis Pharmaceutical Corp.	Tetracycline—doxycycline antibiotic composition
US6991807B2 (en) *	2000-02-24	2006-01-31	Advancis Pharmaceutical, Corp.	Antibiotic composition
US6632453B2 (en)	2000-02-24	2003-10-14	Advancis Pharmaceutical Corp.	Ciprofoxacin-metronidazole antibiotic composition
US6610328B2 (en)	2000-02-24	2003-08-26	Advancis Pharmaceutical Corp.	Amoxicillin-clarithromycin antibiotic composition
AU3984101A (en) *	2000-02-24	2001-09-03	Advanced Pharma Inc	Antibiotic and antifungal compositions
US6663890B2 (en)	2000-02-24	2003-12-16	Advancis Pharmaceutical Corp.	Metronidazole antibiotic product, use and formulation thereof
US6669948B2 (en)	2000-02-24	2003-12-30	Advancis Pharmaceutical Corp.	Antibiotic product, use and formulation thereof
US6544555B2 (en)	2000-02-24	2003-04-08	Advancis Pharmaceutical Corp.	Antibiotic product, use and formulation thereof
US6627222B2 (en)	2000-02-24	2003-09-30	Advancis Pharmaceutical Corp.	Amoxicillin-dicloxacillin antibiotic composition
US6565882B2 (en)	2000-02-24	2003-05-20	Advancis Pharmaceutical Corp	Antibiotic composition with inhibitor
EP1257255A4 (fr) *	2000-02-24	2008-07-30	Advancis Pharmaceutical Corp	Produit therapeutique, son application et sa formulation
US7025989B2 (en) *	2000-02-24	2006-04-11	Advancis Pharmaceutical Corp.	Multiple-delayed released antibiotic product, use and formulation thereof
US6730320B2 (en)	2000-02-24	2004-05-04	Advancis Pharmaceutical Corp.	Tetracycline antibiotic product, use and formulation thereof
US6623758B2 (en)	2000-02-24	2003-09-23	Advancis Pharmaceutical Corp.	Cephalosporin-metronidazole antibiotic composition
US6667042B2 (en)	2000-02-24	2003-12-23	Advancis Pharmaceutical Corp.	Fluroquinilone antibiotic product, use and formulation thereof
US6667057B2 (en)	2000-02-24	2003-12-23	Advancis Pharmaceutical Corp.	Levofloxacin antibiotic product, use and formulation thereof
US6663891B2 (en)	2000-02-24	2003-12-16	Advancis Pharmaceutical Corp.	Erythromyacin antibiotic product, use and formulation thereof
US7157095B2 (en) *	2000-10-13	2007-01-02	Advancis Pharmaceutical Corporation	Multiple-delayed release antifungal product, use and formulation thereof
US6541014B2 (en)	2000-10-13	2003-04-01	Advancis Pharmaceutical Corp.	Antiviral product, use and formulation thereof
US7105174B2 (en) *	2000-10-13	2006-09-12	Advancis Pharmaceutical Corporation	Multiple-delayed release anti-neoplastic product, use and formulation thereof
US7074417B2 (en) *	2000-10-13	2006-07-11	Advancis Pharmaceutical Corporation	Multiple-delayed release anti-viral product, use and formulation thereof
US20020197314A1 (en) *	2001-02-23	2002-12-26	Rudnic Edward M.	Anti-fungal composition
US20040114368A1 (en) *	2002-12-13	2004-06-17	Shyu Shing Jy	Light device having rotatable or movable view
WO2004104022A2 (fr) *	2003-05-16	2004-12-02	The General Hospital Corporation	Compositions contenant un facteur chimio-tactique epithelial pathogene (eicosanoide et hepoxiline a3), leurs inhibiteurs et leurs procedes d'utilisation
JP2006528190A (ja)	2003-07-21	2006-12-14	アドバンシスファーマスーティカルコーポレイション	抗生物質製剤、その使用法及び作成方法
CA2533178C (fr)	2003-07-21	2014-03-11	Advancis Pharmaceutical Corporation	Produit antibiotique, son utilisation et sa formulation
WO2005009364A2 (fr)	2003-07-21	2005-02-03	Advancis Pharmaceutical Corporation	Produit antibiotique, utilisation et formulation associees
US8758820B2 (en)	2003-08-11	2014-06-24	Shionogi Inc.	Robust pellet
US8062672B2 (en)	2003-08-12	2011-11-22	Shionogi Inc.	Antibiotic product, use and formulation thereof
CA2535780A1 (fr)	2003-08-29	2005-03-17	Advancis Pharmaceuticals Corporation	Produit antibiotique, son utilisation et sa formulation
US8460710B2 (en)	2003-09-15	2013-06-11	Shionogi, Inc.	Antibiotic product, use and formulation thereof
WO2006014427A1 (fr)	2004-07-02	2006-02-09	Advancis Pharmaceutical Corporation	Comprimé pour distribution par impulsion
WO2007004239A1 (fr) *	2005-07-06	2007-01-11	Morepen Laboratories Limited	Nouvelle forme polymorphique du tosylate de sultamicilline et procede correspondant
US8357394B2 (en)	2005-12-08	2013-01-22	Shionogi Inc.	Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en)	2006-12-04	2014-07-15	Shionogi Inc.	Modified release amoxicillin products
US8299052B2 (en) *	2006-05-05	2012-10-30	Shionogi Inc.	Pharmaceutical compositions and methods for improved bacterial eradication
EP2874624B8 (fr)	2012-07-17	2019-10-02	Bayer New Zealand Limited	Formulations antibiotiques injectables et leurs procédés d'utilisation
WO2014014364A1 (fr)	2012-07-17	2014-01-23	Bayer New Zealand Limited	Formulations antibiotiques injectables et leurs procédés d'utilisation
US11116737B1 (en)	2020-04-10	2021-09-14	University Of Georgia Research Foundation, Inc.	Methods of using probenecid for treatment of coronavirus infections

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR1532222A (fr) *	1963-10-28	1968-07-12	Bristol Myers Co	Procédé de préparation de dérivés de la pénicilline
IE49880B1 (en) *	1979-02-13	1986-01-08	Leo Pharm Prod Ltd	Penicillin derivatives
ZA80796B (en) *	1979-02-13	1981-02-25	Leo Pharm Prod Ltd	Chemical compounds
US4244951A (en) *	1979-05-16	1981-01-13	Pfizer Inc.	Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
IE51516B1 (en) *	1980-10-06	1987-01-07	Leo Pharm Prod Ltd	1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate

1981
- 1981-10-06 IL IL64009A patent/IL64009A/xx not_active IP Right Cessation
- 1981-10-08 IE IE2361/81A patent/IE51640B1/en not_active IP Right Cessation
- 1981-10-13 NZ NZ198622A patent/NZ198622A/en unknown
- 1981-10-14 GB GB08131010A patent/GB2114969B/en not_active Expired
- 1981-10-14 ZA ZA817091A patent/ZA817091B/xx unknown
- 1981-10-15 AU AU76365/81A patent/AU543870B2/en not_active Expired
- 1981-10-19 PH PH26362A patent/PH17820A/en unknown
- 1981-10-20 AT AT0447781A patent/AT373893B/de not_active IP Right Cessation
- 1981-10-23 FI FI813331A patent/FI813331L/fi not_active Application Discontinuation
- 1981-10-23 IT IT68383/81A patent/IT1193735B/it active
- 1981-10-26 CA CA000388756A patent/CA1180696A/fr not_active Expired
- 1981-10-27 DK DK472181A patent/DK154219C/da not_active IP Right Cessation
- 1981-10-29 SE SE8106404A patent/SE452322B/sv not_active IP Right Cessation
- 1981-10-29 GR GR66381A patent/GR75369B/el unknown
- 1981-10-30 BE BE0/206403A patent/BE890938A/fr not_active IP Right Cessation
- 1981-10-30 NL NL8104938A patent/NL8104938A/nl active Search and Examination
- 1981-10-30 JP JP56175559A patent/JPS57126493A/ja active Granted
- 1981-10-30 CH CH6947/81A patent/CH647527A5/de not_active IP Right Cessation
- 1981-10-30 KR KR1019810004171A patent/KR870001982B1/ko active
- 1981-10-30 ES ES506751A patent/ES506751A0/es active Granted
- 1981-10-30 NO NO813683A patent/NO813683L/no unknown
- 1981-10-30 PT PT73913A patent/PT73913B/pt unknown
- 1981-10-30 FR FR8120476A patent/FR2493322B1/fr not_active Expired
- 1981-10-30 LU LU83727A patent/LU83727A1/fr unknown
- 1981-10-30 DE DE19813143219 patent/DE3143219A1/de active Granted
1987
- 1987-03-13 US US07/024,858 patent/US4831025A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
AU543870B2 (en)	1985-05-09
AU7636581A (en)	1982-05-06
CH647527A5 (de)	1985-01-31
PH17820A (en)	1985-01-07
BE890938A (fr)	1982-04-30
KR830007671A (ko)	1983-11-04
IE812361L (en)	1982-04-30
GB2114969A (en)	1983-09-01
ES8206531A1 (es)	1982-08-16
IL64009A (en)	1984-09-30
DK154219B (da)	1988-10-24
DE3143219C2 (fr)	1990-05-17
ATA447781A (de)	1983-07-15
ZA817091B (en)	1982-10-27
AT373893B (de)	1984-02-27
US4831025A (en)	1989-05-16
NO813683L (no)	1982-05-03
IT1193735B (it)	1988-08-24
DK472181A (da)	1982-05-01
PT73913B (en)	1984-05-29
FI813331L (fi)	1982-05-01
GR75369B (fr)	1984-07-13
PT73913A (en)	1981-11-01
NZ198622A (en)	1985-07-12
KR870001982B1 (ko)	1987-10-24
IT8168383A0 (it)	1981-10-23
JPS57126493A (en)	1982-08-06
JPH027957B2 (fr)	1990-02-21
LU83727A1 (fr)	1982-05-07
DK154219C (da)	1989-03-20
FR2493322B1 (fr)	1986-06-13
SE452322B (sv)	1987-11-23
IL64009A0 (en)	1982-01-31
FR2493322A1 (fr)	1982-05-07
CA1180696A (fr)	1985-01-08
DE3143219A1 (de)	1982-08-12
IE51640B1 (en)	1987-01-21
ES506751A0 (es)	1982-08-16
SE8106404L (sv)	1982-05-01
GB2114969B (en)	1985-02-20

Publication	Publication Date	Title
NL8104938A (nl)	1982-05-17	1.1-dioxopenicillanoyloxymethyl-6-(d-alfa-amino-alfa-fenylaceetamido)penicillanaat, werkwijze voor de bereiding en toepassing daarvan.
JP2021105030A (ja)	2021-07-26	ニコチンアミドリボシドの結晶形
KR930002509B1 (ko)	1993-04-03	결정성 칼슘 슈도모네이트 제법
HU190603B (en)	1986-09-29	Process for the production of /6r7r/-3-carbomoil-oxy-methyl-7- /1z/-2-2/fur-2-il/methoxy-imino-acet-amido/-cef-3-em-4-carboxylic acid-ester of new form
HRP20000669A2 (en)	2001-08-31	Novel crystalline forms of an antiviral benzimidazole compound
KR100191989B1 (ko)	1999-06-15	신규한 결정형의 무수7-((1알파,5알파,6알파)-6-아미노-3-아자비사이클로(3.1.0)헥스-3-일)-6-플루오로-1-(2,4-디플루오로페닐)-1,4-디하이드로-4-옥소-1,8-나프티리딘-3-카복실산 메탄설폰산 염
HU206348B (en)	1992-10-28	Process for producing cristalline beta-lactame-hydrate and pharmaceutical compositions containing them
JPH02178281A (ja)	1990-07-11	β―ラクタム抗生物質の水和物
DE3139554C2 (fr)	1990-04-26
US3822256A (en)	1974-07-02	Crystalline monohydrates of sodium and potassium cephalexin
JPS5962584A (ja)	1984-04-10	コクシジユ−ム症に対して活性なキナゾリノン誘導体
CN105683162A (zh)	2016-06-15	N-(4-氯-2-羟基-3((3s)-3-哌啶基磺酰基)苯基)-n’-(3-氟-2-甲基苯基)脲的氢溴酸盐
EP0162394A2 (fr)	1985-11-27	Céphalosporines et procédé pour leur préparation
NL8200607A (nl)	1982-09-16	2-amino-3(halogeenbenzoyl)-methylfenylazijnzuren, en zouten daarvan.
GB2084572A (en)	1982-04-15	1,1-Dioxopenicillanoyloxymethyl 6-(D- alpha -amino- alpha -phenylacetamido)penicillanate napsylate
EP0439353B1 (fr)	1996-04-24	Hydrochlorure cristallin d'un nouvel antibiotique bêta-lactame et procédé de préparation
US3956279A (en)	1976-05-11	Crystalline pivaloyloxymethyl d(-)-α-aminobenzylpenicillinate
JPH0414679B2 (fr)	1992-03-13
US3928591A (en)	1975-12-23	7-(D-{60 -amino-1,4-cyclohexadien-1-ylacetamido)desacetoxycephalosporanic acid dihydrate compositions
JPS6145625B2 (fr)	1986-10-08
PL80147B1 (en)	1975-08-30	Zinc complexes of quaternary pyridine derivatives[gb1219998a]

Legal Events

Date	Code	Title
1985-01-01	A85	Still pending on 85-01-01
1988-10-03	BA	A request for search or an international-type search has been filed
1988-10-03	BB	A search report has been drawn up
1989-02-01	BC	A request for examination has been filed
2000-11-01	BN	A decision not to publish the application has become irrevocable