NL177116C - PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-HISTAMINE ACTIVITY AND SUITABLE ACTIVE BENZYL-PHTHALAZONE ANALOG. - Google Patents
PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-HISTAMINE ACTIVITY AND SUITABLE ACTIVE BENZYL-PHTHALAZONE ANALOG.Info
- Publication number
- NL177116C NL177116C NLAANVRAGE7200400,A NL7200400A NL177116C NL 177116 C NL177116 C NL 177116C NL 7200400 A NL7200400 A NL 7200400A NL 177116 C NL177116 C NL 177116C
- Authority
- NL
- Netherlands
- Prior art keywords
- phthalazone
- analog
- suitable active
- medicinal products
- preparing medicinal
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH101271A CH572914A5 (en) | 1971-01-22 | 1971-01-22 |
Publications (3)
Publication Number | Publication Date |
---|---|
NL7200400A NL7200400A (en) | 1972-07-25 |
NL177116B NL177116B (en) | 1985-03-01 |
NL177116C true NL177116C (en) | 1985-08-01 |
Family
ID=4200381
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NLAANVRAGE7200400,A NL177116C (en) | 1971-01-22 | 1972-01-11 | PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-HISTAMINE ACTIVITY AND SUITABLE ACTIVE BENZYL-PHTHALAZONE ANALOG. |
Country Status (21)
Country | Link |
---|---|
AR (1) | AR197293A1 (en) |
AT (1) | AT313288B (en) |
AU (1) | AU3767472A (en) |
BE (1) | BE778269A (en) |
CA (1) | CA1010041A (en) |
CH (1) | CH572914A5 (en) |
DE (1) | DE2164058C3 (en) |
DK (1) | DK136981B (en) |
ES (1) | ES398949A1 (en) |
FI (1) | FI53704C (en) |
FR (1) | FR2122517B1 (en) |
GB (1) | GB1377231A (en) |
HK (1) | HK62577A (en) |
HU (1) | HU163979B (en) |
IL (1) | IL38496A (en) |
NL (1) | NL177116C (en) |
OA (1) | OA04087A (en) |
PL (1) | PL88930B1 (en) |
SE (1) | SE404604B (en) |
YU (1) | YU35361B (en) |
ZA (1) | ZA718712B (en) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE49205T1 (en) * | 1984-09-14 | 1990-01-15 | Asta Pharma Ag | SUBSTITUTE BENZYLPHTHALAZINONE DERIVATIVES. |
ES2053678T3 (en) * | 1987-11-13 | 1994-08-01 | Asta Medica Ag | PROCEDURE FOR PREPARING AN AZELASTIN CONTENT MEDICATION FOR NASAL AND / OR EYE APPLICATION. |
ATE106883T1 (en) * | 1987-11-13 | 1994-06-15 | Asta Medica Ag | AZELASTINE EMBONATE, PROCESS FOR ITS PRODUCTION AND PHARMACEUTICAL PREPARATIONS CONTAINING AZELASTINE EMBONATE AS THE ACTIVE SUBSTANCE. |
PT88984B (en) * | 1987-11-13 | 1993-01-29 | Asta Medica Ag | METHOD FOR THE PREPARATION OF AZELASTINE EMBONATE AND EARMACEUTICAL COMPOSITIONS CONTAINING AS ACTIVE INGREDIENT |
DE3836579A1 (en) * | 1987-11-13 | 1989-05-24 | Asta Pharma Ag | Azelastine-containing pharmaceutical compositions for use in the nose and/or on the eye |
DE3912292A1 (en) * | 1988-04-20 | 1989-11-09 | Asta Pharma Ag | Azelastine-containing pharmaceuticals with controlled release of active substance |
US5110814A (en) * | 1989-01-11 | 1992-05-05 | Asta Pharma Ag | Azelastine and its salts used to combat psoriasis |
DK0396069T3 (en) * | 1989-05-05 | 1994-07-25 | Asta Medica Ag | Salts of azelastine with improved solubility |
DE4207234A1 (en) * | 1992-03-07 | 1993-09-09 | Asta Medica Ag | NEW AMINOCARBONIC ACID DERIVATIVES WITH ANTIALLERGIC / ANTIASTHMIC EFFECT AND METHOD FOR THE PRODUCTION THEREOF |
DE4345224C2 (en) * | 1993-12-18 | 1999-07-01 | Asta Medica Ag | Process for the preparation of acid addition salts of azelastine and flezelastin |
DE4343409C2 (en) * | 1993-12-18 | 1997-03-20 | Asta Medica Ag | Improved process for the production of hexahydroazepinones and hexahydroazepinols |
GB2389530B (en) | 2002-06-14 | 2007-01-10 | Cipla Ltd | Pharmaceutical compositions |
PL2377557T3 (en) | 2004-11-24 | 2017-05-31 | Meda Pharmaceuticals Inc. | Compositions comprising azelastine and methods of use thereof |
US20070020330A1 (en) | 2004-11-24 | 2007-01-25 | Medpointe Healthcare Inc. | Compositions comprising azelastine and methods of use thereof |
US8758816B2 (en) | 2004-11-24 | 2014-06-24 | Meda Pharmaceuticals Inc. | Compositions comprising azelastine and methods of use thereof |
WO2007122156A1 (en) * | 2006-04-20 | 2007-11-01 | Glaxo Group Limited | 2-substituted 4-benzylphthalazinone derivatives as histamine h1 and h3 antagonists |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1046625B (en) * | 1957-08-15 | 1958-12-18 | Hydrierwerk Rodleben Veb | Process for the production of basic substituted phthalazones |
GB1100911A (en) * | 1963-08-20 | 1968-01-24 | Benger Lab Ltd | Phthalazine derivatives |
DK119061B (en) * | 1966-10-28 | 1970-11-09 | Hydrierwerk Rodleben Veb | Process for the preparation of basic substituted phthalazones or salts or quaternary ammonium compounds thereof. |
-
1971
- 1971-01-22 CH CH101271A patent/CH572914A5/xx not_active IP Right Cessation
- 1971-12-23 DE DE2164058A patent/DE2164058C3/en not_active Expired
- 1971-12-30 ZA ZA718712A patent/ZA718712B/en unknown
-
1972
- 1972-01-03 IL IL38496A patent/IL38496A/en unknown
- 1972-01-06 AU AU37674/72A patent/AU3767472A/en not_active Expired
- 1972-01-11 NL NLAANVRAGE7200400,A patent/NL177116C/en not_active IP Right Cessation
- 1972-01-12 GB GB143372A patent/GB1377231A/en not_active Expired
- 1972-01-13 AT AT25672A patent/AT313288B/en active
- 1972-01-17 YU YU112/72A patent/YU35361B/en unknown
- 1972-01-18 ES ES398949A patent/ES398949A1/en not_active Expired
- 1972-01-18 CA CA132,681A patent/CA1010041A/en not_active Expired
- 1972-01-19 FR FR7201729A patent/FR2122517B1/fr not_active Expired
- 1972-01-19 AR AR240139A patent/AR197293A1/en active
- 1972-01-20 PL PL1972153002A patent/PL88930B1/pl unknown
- 1972-01-20 BE BE778269A patent/BE778269A/en not_active IP Right Cessation
- 1972-01-21 SE SE7200722A patent/SE404604B/en unknown
- 1972-01-21 HU HUAA695A patent/HU163979B/hu unknown
- 1972-01-21 DK DK30272AA patent/DK136981B/en unknown
- 1972-01-21 FI FI160/72A patent/FI53704C/en active
- 1972-05-15 OA OA54568A patent/OA04087A/en unknown
-
1977
- 1977-12-22 HK HK625/77A patent/HK62577A/en unknown
Also Published As
Publication number | Publication date |
---|---|
AT313288B (en) | 1974-02-11 |
YU35361B (en) | 1980-12-31 |
BE778269A (en) | 1972-07-19 |
DE2164058B2 (en) | 1980-10-23 |
FI53704B (en) | 1978-03-31 |
IL38496A0 (en) | 1972-03-28 |
CA1010041A (en) | 1977-05-10 |
AR197293A1 (en) | 1974-03-29 |
NL7200400A (en) | 1972-07-25 |
HK62577A (en) | 1977-12-30 |
FR2122517B1 (en) | 1975-08-01 |
DE2164058A1 (en) | 1972-07-27 |
HU163979B (en) | 1973-12-28 |
SE404604B (en) | 1978-10-16 |
DK136981B (en) | 1977-12-27 |
ZA718712B (en) | 1972-09-27 |
ES398949A1 (en) | 1975-06-01 |
CH572914A5 (en) | 1976-02-27 |
PL88930B1 (en) | 1976-10-30 |
IL38496A (en) | 1975-05-22 |
FI53704C (en) | 1978-07-10 |
AU3767472A (en) | 1973-07-12 |
SU440838A3 (en) | 1974-08-25 |
DE2164058C3 (en) | 1981-08-13 |
DK136981C (en) | 1978-06-05 |
YU11272A (en) | 1980-06-30 |
FR2122517A1 (en) | 1972-09-01 |
GB1377231A (en) | 1974-12-11 |
OA04087A (en) | 1979-10-30 |
NL177116B (en) | 1985-03-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
BB | A search report has been drawn up | ||
BC | A request for examination has been filed | ||
A85 | Still pending on 85-01-01 | ||
V4 | Discontinued because of reaching the maximum lifetime of a patent |