[go: up one dir, main page]

NL177116C - PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-HISTAMINE ACTIVITY AND SUITABLE ACTIVE BENZYL-PHTHALAZONE ANALOG. - Google Patents

PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-HISTAMINE ACTIVITY AND SUITABLE ACTIVE BENZYL-PHTHALAZONE ANALOG.

Info

Publication number
NL177116C
NL177116C NLAANVRAGE7200400,A NL7200400A NL177116C NL 177116 C NL177116 C NL 177116C NL 7200400 A NL7200400 A NL 7200400A NL 177116 C NL177116 C NL 177116C
Authority
NL
Netherlands
Prior art keywords
phthalazone
analog
suitable active
medicinal products
preparing medicinal
Prior art date
Application number
NLAANVRAGE7200400,A
Other languages
Dutch (nl)
Other versions
NL7200400A (en
NL177116B (en
Original Assignee
Asta Werke Ag Chem Fab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asta Werke Ag Chem Fab filed Critical Asta Werke Ag Chem Fab
Publication of NL7200400A publication Critical patent/NL7200400A/xx
Publication of NL177116B publication Critical patent/NL177116B/en
Application granted granted Critical
Publication of NL177116C publication Critical patent/NL177116C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NLAANVRAGE7200400,A 1971-01-22 1972-01-11 PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-HISTAMINE ACTIVITY AND SUITABLE ACTIVE BENZYL-PHTHALAZONE ANALOG. NL177116C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH101271A CH572914A5 (en) 1971-01-22 1971-01-22

Publications (3)

Publication Number Publication Date
NL7200400A NL7200400A (en) 1972-07-25
NL177116B NL177116B (en) 1985-03-01
NL177116C true NL177116C (en) 1985-08-01

Family

ID=4200381

Family Applications (1)

Application Number Title Priority Date Filing Date
NLAANVRAGE7200400,A NL177116C (en) 1971-01-22 1972-01-11 PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-HISTAMINE ACTIVITY AND SUITABLE ACTIVE BENZYL-PHTHALAZONE ANALOG.

Country Status (21)

Country Link
AR (1) AR197293A1 (en)
AT (1) AT313288B (en)
AU (1) AU3767472A (en)
BE (1) BE778269A (en)
CA (1) CA1010041A (en)
CH (1) CH572914A5 (en)
DE (1) DE2164058C3 (en)
DK (1) DK136981B (en)
ES (1) ES398949A1 (en)
FI (1) FI53704C (en)
FR (1) FR2122517B1 (en)
GB (1) GB1377231A (en)
HK (1) HK62577A (en)
HU (1) HU163979B (en)
IL (1) IL38496A (en)
NL (1) NL177116C (en)
OA (1) OA04087A (en)
PL (1) PL88930B1 (en)
SE (1) SE404604B (en)
YU (1) YU35361B (en)
ZA (1) ZA718712B (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE49205T1 (en) * 1984-09-14 1990-01-15 Asta Pharma Ag SUBSTITUTE BENZYLPHTHALAZINONE DERIVATIVES.
ES2053678T3 (en) * 1987-11-13 1994-08-01 Asta Medica Ag PROCEDURE FOR PREPARING AN AZELASTIN CONTENT MEDICATION FOR NASAL AND / OR EYE APPLICATION.
ATE106883T1 (en) * 1987-11-13 1994-06-15 Asta Medica Ag AZELASTINE EMBONATE, PROCESS FOR ITS PRODUCTION AND PHARMACEUTICAL PREPARATIONS CONTAINING AZELASTINE EMBONATE AS THE ACTIVE SUBSTANCE.
PT88984B (en) * 1987-11-13 1993-01-29 Asta Medica Ag METHOD FOR THE PREPARATION OF AZELASTINE EMBONATE AND EARMACEUTICAL COMPOSITIONS CONTAINING AS ACTIVE INGREDIENT
DE3836579A1 (en) * 1987-11-13 1989-05-24 Asta Pharma Ag Azelastine-containing pharmaceutical compositions for use in the nose and/or on the eye
DE3912292A1 (en) * 1988-04-20 1989-11-09 Asta Pharma Ag Azelastine-containing pharmaceuticals with controlled release of active substance
US5110814A (en) * 1989-01-11 1992-05-05 Asta Pharma Ag Azelastine and its salts used to combat psoriasis
DK0396069T3 (en) * 1989-05-05 1994-07-25 Asta Medica Ag Salts of azelastine with improved solubility
DE4207234A1 (en) * 1992-03-07 1993-09-09 Asta Medica Ag NEW AMINOCARBONIC ACID DERIVATIVES WITH ANTIALLERGIC / ANTIASTHMIC EFFECT AND METHOD FOR THE PRODUCTION THEREOF
DE4345224C2 (en) * 1993-12-18 1999-07-01 Asta Medica Ag Process for the preparation of acid addition salts of azelastine and flezelastin
DE4343409C2 (en) * 1993-12-18 1997-03-20 Asta Medica Ag Improved process for the production of hexahydroazepinones and hexahydroazepinols
GB2389530B (en) 2002-06-14 2007-01-10 Cipla Ltd Pharmaceutical compositions
PL2377557T3 (en) 2004-11-24 2017-05-31 Meda Pharmaceuticals Inc. Compositions comprising azelastine and methods of use thereof
US20070020330A1 (en) 2004-11-24 2007-01-25 Medpointe Healthcare Inc. Compositions comprising azelastine and methods of use thereof
US8758816B2 (en) 2004-11-24 2014-06-24 Meda Pharmaceuticals Inc. Compositions comprising azelastine and methods of use thereof
WO2007122156A1 (en) * 2006-04-20 2007-11-01 Glaxo Group Limited 2-substituted 4-benzylphthalazinone derivatives as histamine h1 and h3 antagonists

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1046625B (en) * 1957-08-15 1958-12-18 Hydrierwerk Rodleben Veb Process for the production of basic substituted phthalazones
GB1100911A (en) * 1963-08-20 1968-01-24 Benger Lab Ltd Phthalazine derivatives
DK119061B (en) * 1966-10-28 1970-11-09 Hydrierwerk Rodleben Veb Process for the preparation of basic substituted phthalazones or salts or quaternary ammonium compounds thereof.

Also Published As

Publication number Publication date
AT313288B (en) 1974-02-11
YU35361B (en) 1980-12-31
BE778269A (en) 1972-07-19
DE2164058B2 (en) 1980-10-23
FI53704B (en) 1978-03-31
IL38496A0 (en) 1972-03-28
CA1010041A (en) 1977-05-10
AR197293A1 (en) 1974-03-29
NL7200400A (en) 1972-07-25
HK62577A (en) 1977-12-30
FR2122517B1 (en) 1975-08-01
DE2164058A1 (en) 1972-07-27
HU163979B (en) 1973-12-28
SE404604B (en) 1978-10-16
DK136981B (en) 1977-12-27
ZA718712B (en) 1972-09-27
ES398949A1 (en) 1975-06-01
CH572914A5 (en) 1976-02-27
PL88930B1 (en) 1976-10-30
IL38496A (en) 1975-05-22
FI53704C (en) 1978-07-10
AU3767472A (en) 1973-07-12
SU440838A3 (en) 1974-08-25
DE2164058C3 (en) 1981-08-13
DK136981C (en) 1978-06-05
YU11272A (en) 1980-06-30
FR2122517A1 (en) 1972-09-01
GB1377231A (en) 1974-12-11
OA04087A (en) 1979-10-30
NL177116B (en) 1985-03-01

Similar Documents

Publication Publication Date Title
NL158488B (en) PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH A CALMING ACTIVITY, THE PREPARED MEDICINAL PRODUCTS THEREFORE OBTAINED AND PROCESS FOR PREPARING SUITABLE ACTIVE SUBSTANCES.
NL162901C (en) METHOD FOR PREPARING MEDICINAL PRODUCTS WITH ACTIVE SUBSTANCES STABILIZED IN THE FORM OF CLATRATES, SO PRODUCED PRODUCTS PRODUCED, AND METHOD FOR PREPARING THE SUITABLE CLINATE.
NL179111C (en) PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH AN EXTENSIVE EFFECT ON THE CENTRAL NERVOUS SYSTEM AND MEDICINAL PHENYLBENODIAZEPINES THEREFOR.
NL153187B (en) PROCEDURE FOR PREPARING A PREPARATION WITH A WORM ANTI-WORK ACTIVITY, PREPARATION FORMED AND PROCEDURE FOR PREPARING SUITABLE COMPOUNDS.
NL162072B (en) PROCESS FOR PREPARING ANTI-NARCOTIC MEDICINAL PRODUCTS, PREPARED MEDICINAL PRODUCTS SO OBTAINED, AND PROCESS FOR PREPARING SUITABLE ACTIVE SUBSTANCES.
NL177021C (en) METHOD FOR PREPARING MEDICINES WITH ANTIBIOTIC ACTIVITY AND MEDICINE COMPOUNDS SUITABLE FOR THAT.
NL167168C (en) METHOD FOR PREPARING AN ORAL MEDICINAL PRODUCT WITH ANTI-ARTHRITIS ACTIVITY, FORMED MEDICINAL PRODUCTS, OBTAINED USING THIS METHOD AND METHOD FOR PREPARING SUITABLE ACTIVE SUBSTANCES
NL152864B (en) PROCEDURE FOR PREPARING A PHARMACEUTICAL PREPARATION WITH TRANSMETHYLING ACTIVITY, PREPARATIONS FORMED THEREFORE OBTAINED AND PROCEDURE FOR PREPARING THE ACTIVE SUBSTANCES THEREFORE.
NL177116C (en) PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-HISTAMINE ACTIVITY AND SUITABLE ACTIVE BENZYL-PHTHALAZONE ANALOG.
NL158797B (en) PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-SPASMODIC AND ANTI-ULCER ACTIVITY, PREPARED MEDICINAL PRODUCTS THEREFORE OBTAINED AND PROCEDURE FOR PREPARING SUITABLE ACTIVE SUBSTANCES THEREOF.
NL166939C (en) METHOD FOR PREPARING MEDICINAL PRODUCTS WITH FAVORABLE BLOOD INFLUENCE AND METHOD FOR PREPARING SUITABLE COMPOUNDS
NL160726C (en) DEVICE FOR DELIVERING AN ACTIVE AGENT, SUCH AS A MEDICINAL PRODUCT.
NL178318C (en) METHOD FOR PREPARING ANTI-EMETICALLY ACTIVE MEDICINAL PRODUCTS AND SUITABLE ACTIVE COMPOUNDS THEREFOR
NL170283C (en) METHOD FOR PREPARING COMPOUNDS WITH ANALGETIC AND ANTI-INFLAMMATIVE ACTIVITY, AND PREPARED MEDICINES PRODUCED THEREFOR
NL167414C (en) METHOD FOR PREPARING A MEDICINAL PRODUCT WITH DIURETIC, SALURETIC AND / OR SECRETOLYTIC ACTIVITY, AND METHOD FOR PREPARING THE ACTIVE BEZYLAMINE DERIVATIVES USED THEREOF
NL152246B (en) PROCEDURE FOR PREPARING A PREPARATION WITH ANTI-ARHYTHMIC ACTIVITY, PREPARATION FORMED, AND PROCEDURE FOR PREPARING A SUITABLE COMPOUND.
NL159384B (en) PROCEDURE FOR PREPARING A MEDICINAL PRODUCT WITH AN ADRENOLYTIC ACTIVITY, AS WELL AS A PROCEDURE FOR PREPARING AN ESTER OF 1-METHYL-10-METHOXYLUMILYSERGOL.
NL170134C (en) METHOD FOR PREPARING A MEDICINAL PRODUCT WITH ANTI-ADRENERGIC ACTIVITY AND MEDICINAL PRODUCT OBTAINED THEREOF, AND METHOD FOR PREPARING AN ANTI-ADRENERGICALLY ACTIVE 5- (1-HYDROXYHYDYYL-2-AMYOXYHYDYYLUSHYDYLYTHYL)
NL176569C (en) METHOD FOR PREPARING MEDICINES WITH DIURETIC ACTIVITY, AND METHOD FOR PREPARING SUITABLE COMPOUNDS.
NL176142C (en) METHOD FOR PREPARING ANTI-ANTI-ANTI-INFLAMMATORY MEDICINAL PRODUCTS AND A COETECLIPATE CONTAINING SUITABLE ACETYLSALICYLIC ACID
NL179056C (en) PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-ALLERGIC AND ANTI-INFLAMMATIVE ACTIVITY, AND MEDICINE COMPOUNDS SUITABLE THEREFOR.
NL161439C (en) METHOD FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS WITH NERVOUS ACTIVITY CONTAINING A 5-(3-DIMETHYLAMINO-PROPYLIDENE)-5H-DIBENZO A,D CYCLOHEPTENE-N-OXIDE, AND METHOD FOR THE PREPARATION OF SUITABLE COMPOUNDS THEREOF.
NL152256B (en) PROCEDURE FOR PREPARING MEDICINAL PRODUCTS CONTAINING BLOOD SUGAR MIRROR LOWERING ACTIVITY, THE MEDICINAL PRODUCTS PREPARED, AND PROCESS FOR PREPARING THE ACTIVE AMIDOALKYLBENZESULPHONYLUREE COMPOUNDS.
NL186287B (en) PROCESS FOR PREPARING AN ENZYME PREPARATION AND ITS USE IN THE PREPARATION OF BAKERY PRODUCTS.
NL174542C (en) METHOD FOR PREPARING A MEDICINAL OR DISINFECTANT WITH BACTERIOSTATIC ACTIVITY AND METHOD FOR PREPARING THE SUITABLE ACTIVE SUBSTANCES

Legal Events

Date Code Title Description
BB A search report has been drawn up
BC A request for examination has been filed
A85 Still pending on 85-01-01
V4 Discontinued because of reaching the maximum lifetime of a patent