MX9708055A - Oxygenated-heterocycle containing sulfonamide inhibitors of aspartyl protease. - Google Patents
Oxygenated-heterocycle containing sulfonamide inhibitors of aspartyl protease.Info
- Publication number
- MX9708055A MX9708055A MX9708055A MX9708055A MX9708055A MX 9708055 A MX9708055 A MX 9708055A MX 9708055 A MX9708055 A MX 9708055A MX 9708055 A MX9708055 A MX 9708055A MX 9708055 A MX9708055 A MX 9708055A
- Authority
- MX
- Mexico
- Prior art keywords
- hiv
- aspartyl protease
- oxygenated
- heterocycle containing
- compounds
- Prior art date
Links
- 108010017640 Aspartic Acid Proteases Proteins 0.000 title abstract 2
- 102000004580 Aspartic Acid Proteases Human genes 0.000 title abstract 2
- 229940124530 sulfonamide Drugs 0.000 title abstract 2
- 150000003456 sulfonamides Chemical class 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 241000713772 Human immunodeficiency virus 1 Species 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 2
- 230000002401 inhibitory effect Effects 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 241000725303 Human immunodeficiency virus Species 0.000 abstract 1
- 108010016183 Human immunodeficiency virus 1 p16 protease Proteins 0.000 abstract 1
- 241000713340 Human immunodeficiency virus 2 Species 0.000 abstract 1
- 108010016191 Human immunodeficiency virus 2 p16 protease Proteins 0.000 abstract 1
- 239000003443 antiviral agent Substances 0.000 abstract 1
- 239000003696 aspartic proteinase inhibitor Substances 0.000 abstract 1
Landscapes
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
The present invention relates to a novel class of sulfonamides which are aspartyl protease inhibitors. This invention also relates to pharmaceutical compositions comprising these compounds. The compounds and pharmaceutical compositions of this invention are particularly well suited for inhibiting HIV-1 and HIV-2 protease activity and consequently, may be advantageously used as anti-viral agents against the HIV-1 and HIV-2 viruses. This invention also relates to methods for inhibiting the activity of HIV aspartyl protease using the compounds of this invention.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08424810 | 1995-04-19 | ||
| PCT/US1996/005473 WO1996033187A1 (en) | 1995-04-19 | 1996-04-18 | Oxygenated-heterocycle containing sulfonamide inhibitors of aspartyl protease |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MXPA97008055A MXPA97008055A (en) | 1998-01-01 |
| MX9708055A true MX9708055A (en) | 1998-01-31 |
Family
ID=39165677
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9708055A MX9708055A (en) | 1996-04-18 | 1996-04-18 | Oxygenated-heterocycle containing sulfonamide inhibitors of aspartyl protease. |
Country Status (1)
| Country | Link |
|---|---|
| MX (1) | MX9708055A (en) |
-
1996
- 1996-04-18 MX MX9708055A patent/MX9708055A/en unknown
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