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MX9206042A - Nuevos derivados de tiadiazinonas, proceso para su fabricacion y preparado farmaceutico que los contiene - Google Patents

Nuevos derivados de tiadiazinonas, proceso para su fabricacion y preparado farmaceutico que los contiene

Info

Publication number
MX9206042A
MX9206042A MX9206042A MX9206042A MX9206042A MX 9206042 A MX9206042 A MX 9206042A MX 9206042 A MX9206042 A MX 9206042A MX 9206042 A MX9206042 A MX 9206042A MX 9206042 A MX9206042 A MX 9206042A
Authority
MX
Mexico
Prior art keywords
tiadiazinones
manufacture
pharmaceutical preparation
preparation containing
new derivatives
Prior art date
Application number
MX9206042A
Other languages
English (en)
Inventor
Rochus Jonas
Michael Klockow
Joachim Leibrock
Hans-Jochen Schliep
Christoph Seyfried
Michael Wolf
Original Assignee
Merck Patent Gmbh
Mit Beschrankter Haftung
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh, Mit Beschrankter Haftung filed Critical Merck Patent Gmbh
Publication of MX9206042A publication Critical patent/MX9206042A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/15Six-membered rings
    • C07D285/16Thiadiazines; Hydrogenated thiadiazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Rheumatology (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
MX9206042A 1991-10-23 1992-10-21 Nuevos derivados de tiadiazinonas, proceso para su fabricacion y preparado farmaceutico que los contiene MX9206042A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4134893A DE4134893A1 (de) 1991-10-23 1991-10-23 Thiadiazinone

Publications (1)

Publication Number Publication Date
MX9206042A true MX9206042A (es) 1993-04-01

Family

ID=6443196

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9206042A MX9206042A (es) 1991-10-23 1992-10-21 Nuevos derivados de tiadiazinonas, proceso para su fabricacion y preparado farmaceutico que los contiene

Country Status (16)

Country Link
US (1) US5276027A (es)
EP (1) EP0539806B1 (es)
JP (1) JP3193789B2 (es)
AT (1) ATE116644T1 (es)
AU (1) AU653444B2 (es)
CA (1) CA2081049A1 (es)
CZ (1) CZ281377B6 (es)
DE (2) DE4134893A1 (es)
DK (1) DK0539806T3 (es)
ES (1) ES2066540T3 (es)
HU (1) HU214337B (es)
MX (1) MX9206042A (es)
NO (1) NO303013B1 (es)
PL (1) PL171273B1 (es)
TW (1) TW309518B (es)
ZA (1) ZA928236B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW309520B (es) * 1994-04-26 1997-07-01 Mitsubishi Chem Corp
DE19500558A1 (de) * 1995-01-11 1996-07-18 Merck Patent Gmbh 3-Alkoxycarbonyl-thiadiazinone
DE19502699A1 (de) * 1995-01-28 1996-08-01 Merck Patent Gmbh Arylalkyl-thiadiazinone
DE19533975A1 (de) * 1995-09-14 1997-03-20 Merck Patent Gmbh Arylalkyl-diazinone
DE10150517A1 (de) * 2001-10-12 2003-04-17 Merck Patent Gmbh Verwendung von Phosphodiesterase IV-Inhibitoren
CZ2004516A3 (cs) * 2001-10-31 2004-08-18 Merckápatentágmbh Inhibitor fosfodiesterázy typu @Ź jeho kombinace s jinými drogami a jeho použití
DE602005005638T2 (de) 2004-02-04 2009-05-14 Nycomed Gmbh 2-(piperidin-4-yl)-4,5-dihydro-2h-pyridazin-3-on-derivate als pde4-inhibitoren
CN101602687A (zh) * 2008-06-13 2009-12-16 上海特化医药科技有限公司 6-硝基苯乙酮类化合物、其制备方法及用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4495185A (en) * 1981-11-12 1985-01-22 Imperial Chemical Industries, Plc 1,2,4-Triazin-3(2H) ones
AU614965B2 (en) * 1987-06-06 1991-09-19 Merck Patent Gesellschaft Mit Beschrankter Haftung Thiadiazinones
DE69131268T2 (de) * 1990-09-21 1999-12-30 Rohm And Haas Co., Philadelphia Dihydropyridazinone und Pyridazinone als Fungizide

Also Published As

Publication number Publication date
JPH05222017A (ja) 1993-08-31
CA2081049A1 (en) 1993-04-24
PL296314A2 (en) 1993-05-04
NO924098L (no) 1993-04-26
TW309518B (es) 1997-07-01
CZ263692A3 (en) 1993-05-12
NO924098D0 (no) 1992-10-22
DK0539806T3 (da) 1995-03-13
ES2066540T3 (es) 1995-03-01
DE59201148D1 (de) 1995-02-16
AU653444B2 (en) 1994-09-29
CZ281377B6 (cs) 1996-09-11
NO303013B1 (no) 1998-05-18
HUT67938A (en) 1995-05-29
EP0539806A1 (de) 1993-05-05
EP0539806B1 (de) 1995-01-04
ATE116644T1 (de) 1995-01-15
HU9203332D0 (en) 1992-12-28
ZA928236B (en) 1993-05-06
US5276027A (en) 1994-01-04
PL171273B1 (pl) 1997-03-28
DE4134893A1 (de) 1993-04-29
JP3193789B2 (ja) 2001-07-30
AU2723192A (en) 1993-04-29
HU214337B (hu) 1998-03-02

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Legal Events

Date Code Title Description
FG Grant or registration
MM Annulment or lapse due to non-payment of fees