MX9203740A - Derivados de anti-inflamatorios de 1,1-dioxido de 2-metil-2h-1,2-benzo-(o-tieno-)tiacine-3-carboxamida, y composiciones de los mismos. - Google Patents

Derivados de anti-inflamatorios de 1,1-dioxido de 2-metil-2h-1,2-benzo-(o-tieno-)tiacine-3-carboxamida, y composiciones de los mismos.

Info

Publication number: MX9203740A
Authority: MX; Mexico
Prior art keywords: tiacine; teno; carboxamide; benzo; dioxide
Prior art date: 1983-12-21

Application number

MX9203740A

Other languages

English (en)

Inventor

Anthony Marfat

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-12-21

Filing date

1992-06-29

Publication date

1992-09-01

1992-06-29 Application filed by Pfizer filed Critical Pfizer

1992-09-01 Publication of MX9203740A publication Critical patent/MX9203740A/es

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C68/00—Preparation of esters of carbonic or haloformic acids
- C07C68/02—Preparation of esters of carbonic or haloformic acids from phosgene or haloformates
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Steroid Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

MX9203740A 1983-12-21 1992-06-29 Derivados de anti-inflamatorios de 1,1-dioxido de 2-metil-2h-1,2-benzo-(o-tieno-)tiacine-3-carboxamida, y composiciones de los mismos. MX9203740A (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US56390283A	1983-12-21	1983-12-21
US06/606,113 US4551452A (en)	1983-12-21	1984-05-02	Anti-inflammatory 2-methyl-2H-1,2-benzo-(or -thieno-)thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor

Publications (1)

Publication Number	Publication Date
MX9203740A true MX9203740A (es)	1992-09-01

Family

ID=27073413

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
MX005836A MX174596B (es)	1983-12-21	1984-12-20	Procedimiento para la preparacion de derivados enol-eter de oxicams
MX9203740A MX9203740A (es)	1983-12-21	1992-06-29	Derivados de anti-inflamatorios de 1,1-dioxido de 2-metil-2h-1,2-benzo-(o-tieno-)tiacine-3-carboxamida, y composiciones de los mismos.

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
MX005836A MX174596B (es)	1983-12-21	1984-12-20	Procedimiento para la preparacion de derivados enol-eter de oxicams

Country Status (26)

Country	Link
US (1)	US4551452A (es)
EP (1)	EP0147177B1 (es)
KR (1)	KR860002035B1 (es)
AU (1)	AU552940B2 (es)
BG (1)	BG47946A3 (es)
CA (1)	CA1255302A (es)
DD (1)	DD229125A5 (es)
DE (1)	DE3466776D1 (es)
DK (1)	DK166678B1 (es)
EG (1)	EG17049A (es)
ES (1)	ES8604215A1 (es)
FI (1)	FI79850C (es)
GR (1)	GR82512B (es)
HK (1)	HK58589A (es)
HU (1)	HU201063B (es)
IE (1)	IE57680B1 (es)
IL (1)	IL73873A (es)
MX (2)	MX174596B (es)
NO (1)	NO161317C (es)
NZ (1)	NZ210632A (es)
PH (1)	PH21447A (es)
PL (1)	PL145989B1 (es)
PT (1)	PT79700B (es)
RO (1)	RO90048A (es)
SG (1)	SG27001G (es)
YU (1)	YU43677B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4616012A (en) *	1983-11-25	1986-10-07	Schering Corporation	Carboxyalkyl dipeptides as antiglaucoma agents
US4778795A (en) *	1983-11-25	1988-10-18	Schering Corporation	Carboxyalkyl dipeptides as antiglaucoma agents
US5017567A (en) *	1983-11-25	1991-05-21	Schering Corporation	Carboxyalkyl dipeptides as antiglaucoma agents
US4906635A (en) *	1983-11-25	1990-03-06	Schering Corporation	Carboxyalkyl dipeptides as antiglaucoma agents
US4623486A (en) *	1985-05-29	1986-11-18	Pfizer Inc.	[4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
KR890001236B1 (ko) *	1985-10-02	1989-04-28	화이자 인코포레이티드	소염제 조성물의 제조방법
US4771071A (en) *	1986-05-05	1988-09-13	Merck & Co., Inc.	Antihypercholesterolemic compounds
HU199833B (en) *	1986-05-16	1990-03-28	Pfizer	Process for producing benzothiazine dioxide derivatives
US5081118A (en) *	1987-10-26	1992-01-14	Pfizer Inc.	Benzothiazine dioxide derivatives
IL87951A (en) *	1987-10-29	1992-03-29	Chem Pharm Forsch Gmbh	Carbonic acid esters of 6-chloro-4-(1-hydroxyethoxy)-2-methyl-n-(2-pyridyl)-2h-thieno(2,3-e)-1,2-thiazine-3-carboxamide 1,1-dioxide,their preparation and pharmaceutical compositions containing them
ZA945190B (en) *	1993-07-30	1995-02-24	Kotobuki Seiyaku Co Ltd	Carboxymethylidenecycloheptimidazole derivatives method or manufacturing the same and therapeutic agents containing these compounds
IT1308633B1 (it)	1999-03-02	2002-01-09	Nicox Sa	Nitrossiderivati.
CN100389114C (zh) *	2006-01-17	2008-05-21	南京新港医药有限公司	一种安吡昔康的精制方法
US20090221703A1 (en)	2006-07-09	2009-09-03	Chongxi Yu	High penetration composition and uses thereof
US20090238763A1 (en) *	2006-07-09	2009-09-24	Chongxi Yu	High penetration compositions and uses thereof
EP2084165B1 (en) *	2006-10-11	2013-06-12	Techfields Biochem Co. Ltd	Positively charged water-soluble prodrugs of oxicams and related compounds with very high skin penetration rate
MX2009013136A (es) *	2007-06-04	2010-04-30	Techfields Inc	Profarmacos de nsaias con piel y membranas con indices de penetracion muy altos y nuevos usos medicinales.
CN107261149A (zh)	2008-12-04	2017-10-20	于崇曦	高穿透性组合物及其应用
WO2013093931A2 (en)	2011-09-19	2013-06-27	Sun Pharma Advanced Research Company Ltd.	Novel prodrugs of phenolic drugs

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3591584A (en) *	1968-08-27	1971-07-06	Pfizer	Benzothiazine dioxides
US3787324A (en) *	1971-03-01	1974-01-22	Warner Lambert Co	4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3892740A (en) *	1974-10-15	1975-07-01	Pfizer	Process for the production of carboxamides of oxo-1,2-benzothiazine-1,1-dioxides
AU518216B2 (en) *	1977-09-06	1981-09-17	Hafslund Nycomed Pharma Aktiengesellschaft	Thienothiazine derivatives
US4309427A (en) *	1981-01-15	1982-01-05	Pfizer Inc.	Benzothiazine dioxide derivatives
IT1168064B (it) *	1981-11-12	1987-05-20	Prodotti Antibiotici Spa	Composto ad azione antinfiammatoria
IT8219486A0 (it) *	1982-02-05	1982-02-05	Chiesi Farma Spa	Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche.

1984
- 1984-05-02 US US06/606,113 patent/US4551452A/en not_active Expired - Lifetime
- 1984-11-28 PH PH31504A patent/PH21447A/en unknown
- 1984-12-18 PT PT79700A patent/PT79700B/pt unknown
- 1984-12-19 NZ NZ210632A patent/NZ210632A/en unknown
- 1984-12-19 GR GR82512A patent/GR82512B/el unknown
- 1984-12-19 EP EP84308926A patent/EP0147177B1/en not_active Expired
- 1984-12-19 RO RO84116745A patent/RO90048A/ro unknown
- 1984-12-19 PL PL1984251040A patent/PL145989B1/pl unknown
- 1984-12-19 EG EG786/84A patent/EG17049A/xx active
- 1984-12-19 IE IE3260/84A patent/IE57680B1/en not_active IP Right Cessation
- 1984-12-19 CA CA000470471A patent/CA1255302A/en not_active Expired
- 1984-12-19 SG SG305/89A patent/SG27001G/en unknown
- 1984-12-19 DE DE8484308926T patent/DE3466776D1/de not_active Expired
- 1984-12-20 KR KR1019840008144A patent/KR860002035B1/ko not_active IP Right Cessation
- 1984-12-20 DK DK614984A patent/DK166678B1/da active
- 1984-12-20 DD DD84271297A patent/DD229125A5/de not_active IP Right Cessation
- 1984-12-20 AU AU36997/84A patent/AU552940B2/en not_active Expired
- 1984-12-20 IL IL73873A patent/IL73873A/xx not_active IP Right Cessation
- 1984-12-20 ES ES538907A patent/ES8604215A1/es not_active Expired
- 1984-12-20 NO NO845145A patent/NO161317C/no not_active IP Right Cessation
- 1984-12-20 YU YU2160/84A patent/YU43677B/xx unknown
- 1984-12-20 HU HU844756A patent/HU201063B/hu unknown
- 1984-12-20 BG BG067990A patent/BG47946A3/xx unknown
- 1984-12-20 MX MX005836A patent/MX174596B/es unknown
- 1984-12-20 FI FI845074A patent/FI79850C/fi active IP Right Grant
1989
- 1989-07-20 HK HK585/89A patent/HK58589A/xx not_active IP Right Cessation
1992
- 1992-06-29 MX MX9203740A patent/MX9203740A/es unknown

Also Published As

Publication number	Publication date
HU201063B (en)	1990-09-28
NO845145L (no)	1985-06-24
KR850004492A (ko)	1985-07-15
NO161317B (no)	1989-04-24
RO90048A (ro)	1986-09-30
PH21447A (en)	1987-10-28
AU3699784A (en)	1985-07-04
PT79700A (en)	1985-01-01
YU43677B (en)	1989-10-31
DD229125A5 (de)	1985-10-30
EP0147177A3 (en)	1985-08-14
HK58589A (en)	1989-07-28
SG27001G (en)	1989-08-11
NO161317C (no)	1989-08-02
KR860002035B1 (ko)	1986-11-17
CA1255302A (en)	1989-06-06
GR82512B (en)	1985-04-22
IE57680B1 (en)	1993-02-24
EG17049A (en)	1991-03-30
DK614984D0 (da)	1984-12-20
EP0147177B1 (en)	1987-10-14
FI845074L (fi)	1985-06-22
US4551452A (en)	1985-11-05
IL73873A (en)	1988-02-29
DK614984A (da)	1985-07-17
YU216084A (en)	1986-10-31
FI79850C (fi)	1990-03-12
FI79850B (fi)	1989-11-30
NZ210632A (en)	1987-02-20
PL251040A1 (en)	1985-10-22
PL145989B1 (en)	1988-12-31
FI845074A0 (fi)	1984-12-20
AU552940B2 (en)	1986-06-26
IL73873A0 (en)	1985-03-31
EP0147177A2 (en)	1985-07-03
MX174596B (es)	1994-05-30
DK166678B1 (da)	1993-06-28
ES8604215A1 (es)	1986-01-16
PT79700B (en)	1986-12-30
HUT37426A (en)	1985-12-28
ES538907A0 (es)	1986-01-16
BG47946A3 (en)	1990-10-15
IE843260L (en)	1985-06-21
DE3466776D1 (en)	1987-11-19

Publication	Publication Date	Title
NO844845L (no)	1985-06-06	Derivater av 2,2`-iminobisetanol
MX9203740A (es)	1992-09-01	Derivados de anti-inflamatorios de 1,1-dioxido de 2-metil-2h-1,2-benzo-(o-tieno-)tiacine-3-carboxamida, y composiciones de los mismos.
MX9203380A (es)	1992-09-01	Derivados de carbazolil-(4)-oxi-propanolamina y composiciones farmaceuticas que los contienen.
NO874764L (no)	1987-11-16	Fremgangsmaate for fremstilling av 2-aminopurinderivater.
DE3752371D1 (de)	2003-08-07	Fotoresistzusammensetzungen und ihre Bestandteile
FI802506A (fi)	1981-02-10	Anti-inflammatoriska 5-substituerade 2,3-diaryltiofener
FI872367A (fi)	1987-12-01	Foerfarande foer framstaellning av vattenhaltiga n-metylmorfolin-n-oxidloesningar.
ES2015047B3 (es)	1990-08-01	Nuevos derivados de 18-fenilestrano.
MX9202935A (es)	1992-06-30	Derivados de 2,3-dihidro-1h-indeno y composicion farmaceutica que los contiene.
FI793261A (fi)	1980-04-21	Farmaceutisk komposition som innehaoller 3,4-dihydro-3-oxo-2-kinoxaliner
NO890483D0 (no)	1989-02-07	Framgangsmaate for tilvirkning av formlegemer.
DK107482A (da)	1982-09-13	Fremstilling af 2,3-dichlor-5-trichlormethylpyridin
IT8320631A0 (it)	1983-04-15	Derivati n-carbammoilici dell'isotiazolo-(5,4b)piridin-one-3 e loro procedimentodi preparazione.
ATE125794T1 (de)	1995-08-15	Prodrogen von antiinflammatorischen 3-acyl-2- oxindol-1-carboxamiden.
BE850472A (fr)	1977-07-18	Derives d'imidazothiazole et theiazolopyrimidine antiinflammatoires
IT1174602B (it)	1987-07-01	Preparazione del 3.3.3-trifluoro-2-trifluorometilpropene
IT1085538B (it)	1985-05-28	Derivati di i 125 immidazol-steroidi
DE3762800D1 (de)	1990-06-28	Benzhydrylthiomethan-derivate enthaltende therapeutische zusammensetzungen.
IT1170097B (it)	1987-06-03	Composizioni n-cianoammidiche e loro addotti
IT8419778A0 (it)	1984-02-23	Derivati di benzammidi.
MC1285A1 (fr)	1980-07-22	Derives d'isoquinoleine
IT8223186A0 (it)	1982-09-09	Composizioni vulcanizzabili e loro impiego.
IT1206513B (it)	1989-04-27	Composizioni farmaceutiche adattivita'antibiotica-immunostimolante.
IT1212552B (it)	1989-11-30	Alcanolaminossi derivati di 3,4-diidro-2h-1.4-benzotiazin-3-one, loro procedimento di produzione e loro utilizzazione farmaceutica
IT7919012A0 (it)	1979-01-02	Derivati di 11-alcanoil-4"-deossi-4"-isonitriloleandomicina.