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MX2011013790A - Derivados de flavina. - Google Patents

Derivados de flavina.

Info

Publication number
MX2011013790A
MX2011013790A MX2011013790A MX2011013790A MX2011013790A MX 2011013790 A MX2011013790 A MX 2011013790A MX 2011013790 A MX2011013790 A MX 2011013790A MX 2011013790 A MX2011013790 A MX 2011013790A MX 2011013790 A MX2011013790 A MX 2011013790A
Authority
MX
Mexico
Prior art keywords
flavin derivatives
derivatives
flavin
infectives
compositions
Prior art date
Application number
MX2011013790A
Other languages
English (en)
Inventor
Kenneth F Blount
Andrew Roughton
Philip Wickens
Brian R Dixon
Judd Berman
David Osterman
Bruce R Evans
Jeffrey A Leiby
Heinrich J Schostarez
Dennis Underwood
Angelica Bello
David Moon
Vinh Pham
Stephanie Avola
Nick Baboulas
Manuel Navia
Harpreet Kaur
Jeffrey Wilson
Philip D G Coish
Paul Adrian Aristoff
Jayhuk Myung
Thomas R Belliotti
Robert A Chrusciel
Frank Sciavolino
Original Assignee
Biorelix Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biorelix Inc filed Critical Biorelix Inc
Publication of MX2011013790A publication Critical patent/MX2011013790A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

La presente invención se refiere a derivados novedosos de flavina y otros derivados de flavina, su uso y composiciones para usarse como ligandos riboswitch y/o anti-infecciosos. La invención también proporciona un método para hacer derivados novedosos de flavina.
MX2011013790A 2009-06-30 2010-06-30 Derivados de flavina. MX2011013790A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22193709P 2009-06-30 2009-06-30
US30323710P 2010-02-10 2010-02-10
PCT/US2010/001876 WO2011008247A1 (en) 2009-06-30 2010-06-30 Flavin derivatives

Publications (1)

Publication Number Publication Date
MX2011013790A true MX2011013790A (es) 2012-03-14

Family

ID=43449644

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2011013790A MX2011013790A (es) 2009-06-30 2010-06-30 Derivados de flavina.

Country Status (10)

Country Link
US (1) US20120295903A1 (es)
EP (1) EP2448926A4 (es)
JP (1) JP2012532126A (es)
KR (1) KR20120089437A (es)
CN (1) CN102471283A (es)
AU (1) AU2010273207A1 (es)
CA (1) CA2765942A1 (es)
MX (1) MX2011013790A (es)
SG (1) SG177323A1 (es)
WO (1) WO2011008247A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102011105653A1 (de) 2011-06-22 2012-12-27 TriOpto Tec GmbH 10H-Benzo[g]pteridin-2,4-dion-Derivate, Verfahren zur Herstellung und Verwendung derselben
DE102011105660A1 (de) 2011-06-22 2012-12-27 TriOpto Tec GmbH Verwendung von 10H-Benzo[g]pteridin-2,4-dion-Derivaten
DE102011105657A1 (de) 2011-06-22 2012-12-27 TriOpto Tec GmbH 10H-Benzo[g]pteridin-2,4-dion-Derivate, Verfahren zur Herstellung und Verwendung derselben
WO2014184272A2 (en) * 2013-05-14 2014-11-20 Medizinische Hochschule Hannover Means and methods for treating cancer
CN104045641A (zh) * 2013-10-11 2014-09-17 镇江市高等专科学校 光黄素的合成方法
CN109554320A (zh) * 2018-11-16 2019-04-02 华南农业大学 Pa4608蛋白作为靶点在制备抗菌药物中的应用
CN113372281A (zh) * 2020-03-09 2021-09-10 河北中科金辉药业有限公司 一种特硝唑的合成方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3920650A (en) * 1973-09-19 1975-11-18 Morton Norwich Products Inc Isoalloxazines
JP2011530595A (ja) * 2008-08-11 2011-12-22 バイオレリックス・インコーポレイテッド フラビン誘導体
EP2531223A4 (en) * 2010-02-04 2013-06-26 Biorelix Inc NEW METHODS AND DEVICES

Also Published As

Publication number Publication date
CN102471283A (zh) 2012-05-23
EP2448926A1 (en) 2012-05-09
EP2448926A4 (en) 2013-04-10
WO2011008247A1 (en) 2011-01-20
CA2765942A1 (en) 2011-01-20
SG177323A1 (en) 2012-02-28
JP2012532126A (ja) 2012-12-13
US20120295903A1 (en) 2012-11-22
KR20120089437A (ko) 2012-08-10
AU2010273207A1 (en) 2012-02-23

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Legal Events

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