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MX2007003922A - Nuevas propenonas ciclicas y aciclicas para tratar trastornos del sistema nervioso central. - Google Patents

Nuevas propenonas ciclicas y aciclicas para tratar trastornos del sistema nervioso central.

Info

Publication number
MX2007003922A
MX2007003922A MX2007003922A MX2007003922A MX2007003922A MX 2007003922 A MX2007003922 A MX 2007003922A MX 2007003922 A MX2007003922 A MX 2007003922A MX 2007003922 A MX2007003922 A MX 2007003922A MX 2007003922 A MX2007003922 A MX 2007003922A
Authority
MX
Mexico
Prior art keywords
propenones
acyclic
cns disorders
novel cyclic
treating cns
Prior art date
Application number
MX2007003922A
Other languages
English (en)
Inventor
Christopher Graham Rap Parsons
Ivars Kalvinsh
Markus Henrich
Tanja Weil
Valerjans Kauss
Wojciech Danysz
Dina Trifanova
Ronalds Zemribo
Original Assignee
Merz Pharma Gmbh & Co Kgaa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merz Pharma Gmbh & Co Kgaa filed Critical Merz Pharma Gmbh & Co Kgaa
Publication of MX2007003922A publication Critical patent/MX2007003922A/es

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/80Radicals substituted by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/12Ketones
    • A61K31/121Ketones acyclic
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    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/72Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction of compounds containing >C = O groups with the same or other compounds containing >C = O groups
    • C07C45/74Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction of compounds containing >C = O groups with the same or other compounds containing >C = O groups combined with dehydration
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Abstract

La invencion se refiere a nuevos derivados de propenona ciclicos y no ciclicos asi como a sus sales farmaceuticamente aceptables. La invencion se refiere ademas a un procedimiento para la preparacion de estos compuestos. Los compuestos de la invencion son utiles como medicamentos.
MX2007003922A 2004-10-05 2005-10-05 Nuevas propenonas ciclicas y aciclicas para tratar trastornos del sistema nervioso central. MX2007003922A (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US61619304P 2004-10-05 2004-10-05
US65642605P 2005-02-24 2005-02-24
US70723905P 2005-08-11 2005-08-11
PCT/GB2005/003817 WO2006037996A1 (en) 2004-10-05 2005-10-05 Novel cyclic and acyclic propenones for treating cns disorders

Publications (1)

Publication Number Publication Date
MX2007003922A true MX2007003922A (es) 2007-06-07

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KR20130097813A (ko) 2008-04-21 2013-09-03 오토노미, 인코포레이티드 귀 질환 및 병태를 치료하기 위한 귀 조제물
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IL182356A0 (en) 2007-07-24
EP1804781A1 (en) 2007-07-11
JP2008515867A (ja) 2008-05-15
BRPI0517549A (pt) 2008-10-14
KR20070056138A (ko) 2007-05-31
CA2580221A1 (en) 2006-04-13
AU2005291075A1 (en) 2006-04-13
WO2006037996A1 (en) 2006-04-13
EA200700807A1 (ru) 2007-08-31
US20060074083A1 (en) 2006-04-06

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