MA52337A - Nouveaux analogues d'oxaborole et utilisations de ces derniers - Google Patents
Nouveaux analogues d'oxaborole et utilisations de ces derniersInfo
- Publication number
- MA52337A MA52337A MA052337A MA52337A MA52337A MA 52337 A MA52337 A MA 52337A MA 052337 A MA052337 A MA 052337A MA 52337 A MA52337 A MA 52337A MA 52337 A MA52337 A MA 52337A
- Authority
- MA
- Morocco
- Prior art keywords
- oxaborole
- analogues
- latest
- new
- oxaborole analogues
- Prior art date
Links
- OHENQANLQNOMAO-UHFFFAOYSA-N oxaborole Chemical class O1B=CC=C1 OHENQANLQNOMAO-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201762465294P | 2017-03-01 | 2017-03-01 |
Publications (1)
Publication Number | Publication Date |
---|---|
MA52337A true MA52337A (fr) | 2021-03-03 |
Family
ID=63370509
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA052337A MA52337A (fr) | 2017-03-01 | 2018-03-01 | Nouveaux analogues d'oxaborole et utilisations de ces derniers |
Country Status (4)
Country | Link |
---|---|
US (2) | US10961261B2 (fr) |
EP (1) | EP3609504A4 (fr) |
MA (1) | MA52337A (fr) |
WO (1) | WO2018160845A1 (fr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
NZ745681A (en) | 2016-03-07 | 2022-05-27 | Agrofresh Inc | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
WO2018160845A1 (fr) | 2017-03-01 | 2018-09-07 | Anacor Pharmaceuticals, Inc. | Nouveaux analogues d'oxaborole et utilisations de ces derniers |
EP4204012A1 (fr) | 2020-08-31 | 2023-07-05 | Pfizer Inc. | Procédés de protection de l'arn |
TWI870837B (zh) | 2022-04-28 | 2025-01-21 | 日商日本農藥股份有限公司 | 具肟基之含氮雜環化合物及含有該化合物之農園藝用除草劑、以及彼等之使用方法 |
WO2024177602A1 (fr) * | 2023-02-20 | 2024-08-29 | Yeditepe Universitesi | Utilisation du bore pour le traitement de la leishmaniose d'origine neuronale |
Family Cites Families (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2509645A1 (fr) | 2002-12-18 | 2004-07-08 | Anacor Pharmaceuticals, Inc. | Antibiotiques contenant des complexes d'acide borinique et leurs procedes d'utilisation |
MXPA05013848A (es) | 2003-06-16 | 2006-09-04 | Anacor Pharmaceuticals Inc | Agentes terapeuticos que contienen boro hidroliticamente resistentes y metodos de uso. |
AR049915A1 (es) | 2004-06-14 | 2006-09-13 | Anacor Pharmaceuticals Inc | Compuestos con contenido de boro y metodos de uso de los mismos |
US7393856B2 (en) | 2004-06-14 | 2008-07-01 | Anacor Pharmaceuticals, Inc. | Anti-viral uses of borinic acid complexes |
DK2719388T3 (da) | 2006-02-16 | 2019-05-13 | Anacor Pharmaceuticals Inc | Borholdige små molekyler som antiinflammatoriske midler |
EP2015757A4 (fr) | 2006-05-02 | 2011-01-26 | Anacor Pharmaceuticals Inc | Substances thérapeutiques contenant du bore résistant à l'hydrolyse et méthodes d'utilisation |
EP2044091A4 (fr) | 2006-06-12 | 2010-08-04 | Anacor Pharmaceuticals Inc | Composés destinés au traitement d'une maladie périodontale |
JO3396B1 (ar) | 2007-06-20 | 2019-10-20 | Anacor Pharmaceuticals Inc | جزيئات صغيرة تحتوي على البورون |
WO2009111676A2 (fr) | 2008-03-06 | 2009-09-11 | Anacor Pharmaceuticals, Inc | Petites molécules contenant du bore utilisées en tant qu'agents anti-inflammatoires |
JP2011515359A (ja) * | 2008-03-18 | 2011-05-19 | グラクソ グループ リミテッド | 治療用トリアゾールアミド誘導体 |
EP2285384A4 (fr) | 2008-05-12 | 2012-04-25 | Anacor Pharmaceuticals Inc | Petites molécules contenant du bore |
EP2348863A4 (fr) | 2008-09-04 | 2012-03-07 | Anacor Pharmaceuticals Inc | Petites molécules contenant du bore |
US9493489B2 (en) | 2008-10-15 | 2016-11-15 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-protozoal agents |
WO2010045505A1 (fr) | 2008-10-15 | 2010-04-22 | Anacor Pharmaceuticals, Inc | Petites molécules contenant du bore en tant qu’agents antiprotozoaires |
PE20120052A1 (es) | 2008-12-17 | 2012-02-13 | Anacor Pharmaceuticals Inc | Polimorfos de (s)-3-amino-metil-7-(3-hidroxi-propoxi)-3h-benzo-[c][1,2]-oxaborol-1-ol |
JP2013500974A (ja) | 2009-07-28 | 2013-01-10 | アナコール ファーマシューティカルズ,インコーポレイテッド | 三置換ホウ素含有分子 |
US9440994B2 (en) * | 2009-08-14 | 2016-09-13 | Anacor Pharmaceuticals, Inc. | Boron containing small molecules as antiprotozoal agents |
US20110207701A1 (en) | 2009-08-19 | 2011-08-25 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
US20110124597A1 (en) | 2009-09-25 | 2011-05-26 | Anacor Pharmaceuticals, Inc. | Boron containing small molecules |
US9346834B2 (en) | 2009-10-20 | 2016-05-24 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
US8461134B2 (en) | 2009-11-11 | 2013-06-11 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
WO2011094450A1 (fr) | 2010-01-27 | 2011-08-04 | Anacor Pharmaceuticals, Inc | Petites molecules contenant du bore |
WO2011116348A1 (fr) | 2010-03-19 | 2011-09-22 | Anacor Pharmaceuticals, Inc. | Petites molécules borées en tant qu'agent anti-protozoaire |
HUE059033T2 (hu) | 2010-09-07 | 2022-10-28 | Anacor Pharmaceuticals Inc | Benzoxaborol-származékok bakteriális fertõzések kezelésére |
WO2012145734A1 (fr) * | 2011-04-22 | 2012-10-26 | The Ohio State University | Compositions antileshmaniennes et ses méthodes d'utilisation |
AR088669A1 (es) | 2011-11-21 | 2014-06-25 | Lilly Co Eli | Derivados de dihidrodibenzo[c][1,2]oxaborol y dihidroisoxazol utiles para el control de ectoparasitos |
AR088668A1 (es) | 2011-11-21 | 2014-06-25 | Lilly Co Eli | Moleculas pequeñas que contienen boro |
JP6298472B2 (ja) * | 2012-11-19 | 2018-03-20 | ノバルティス アーゲー | 寄生虫病の処置のための化合物および組成物 |
US9598443B2 (en) * | 2013-02-01 | 2017-03-21 | Anacor Pharmaceuticals, Inc. | Boron containing small molecules as antiprotozoal agents |
WO2015013318A1 (fr) | 2013-07-22 | 2015-01-29 | Anacor Pharmaceuticals, Inc. | Petites molécules contenant du bore |
WO2018160845A1 (fr) | 2017-03-01 | 2018-09-07 | Anacor Pharmaceuticals, Inc. | Nouveaux analogues d'oxaborole et utilisations de ces derniers |
-
2018
- 2018-03-01 WO PCT/US2018/020464 patent/WO2018160845A1/fr unknown
- 2018-03-01 EP EP18761407.8A patent/EP3609504A4/fr active Pending
- 2018-03-01 US US16/489,824 patent/US10961261B2/en active Active
- 2018-03-01 MA MA052337A patent/MA52337A/fr unknown
-
2021
- 2021-02-11 US US17/173,884 patent/US11691992B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
WO2018160845A1 (fr) | 2018-09-07 |
US20200024289A1 (en) | 2020-01-23 |
EP3609504A4 (fr) | 2021-03-03 |
US10961261B2 (en) | 2021-03-30 |
US20210253605A1 (en) | 2021-08-19 |
EP3609504A1 (fr) | 2020-02-19 |
US11691992B2 (en) | 2023-07-04 |
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