[go: up one dir, main page]

MA49887A - Administration sous-cutanée d'un antagoniste du récepteur p2y12 - Google Patents

Administration sous-cutanée d'un antagoniste du récepteur p2y12

Info

Publication number
MA49887A
MA49887A MA049887A MA49887A MA49887A MA 49887 A MA49887 A MA 49887A MA 049887 A MA049887 A MA 049887A MA 49887 A MA49887 A MA 49887A MA 49887 A MA49887 A MA 49887A
Authority
MA
Morocco
Prior art keywords
receptor antagonist
subcutaneous administration
subcutaneous
administration
antagonist
Prior art date
Application number
MA049887A
Other languages
English (en)
French (fr)
Inventor
Martine Baumann
Markus Kramberg
Markus Rey
Markus Riederer
Sebastien Roux
Original Assignee
Idorsia Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idorsia Pharmaceuticals Ltd filed Critical Idorsia Pharmaceuticals Ltd
Publication of MA49887A publication Critical patent/MA49887A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0021Intradermal administration, e.g. through microneedle arrays, needleless injectors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MA049887A 2017-03-15 2018-03-14 Administration sous-cutanée d'un antagoniste du récepteur p2y12 MA49887A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP2017056175 2017-03-15

Publications (1)

Publication Number Publication Date
MA49887A true MA49887A (fr) 2020-06-24

Family

ID=61899166

Family Applications (1)

Application Number Title Priority Date Filing Date
MA049887A MA49887A (fr) 2017-03-15 2018-03-14 Administration sous-cutanée d'un antagoniste du récepteur p2y12

Country Status (19)

Country Link
US (1) US11179390B2 (uk)
EP (1) EP3595666A1 (uk)
JP (2) JP7580918B2 (uk)
KR (1) KR102510832B1 (uk)
CN (1) CN110381947A (uk)
AU (1) AU2018234056B2 (uk)
BR (1) BR112019014567A2 (uk)
CA (1) CA3050831A1 (uk)
CL (1) CL2019002318A1 (uk)
EA (1) EA201992123A1 (uk)
IL (1) IL269286B2 (uk)
MA (1) MA49887A (uk)
MX (1) MX2019009559A (uk)
MY (1) MY205605A (uk)
PH (1) PH12019502111A1 (uk)
SG (1) SG11201908128YA (uk)
TW (1) TWI765002B (uk)
UA (1) UA125531C2 (uk)
WO (1) WO2018167139A1 (uk)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102552795B1 (ko) 2016-09-22 2023-07-06 이도르시아 파마슈티컬스 리미티드 결정질 형태
AU2021309018A1 (en) * 2020-07-15 2023-03-16 Idorsia Pharmaceuticals Ltd Aqueous pharmaceutical composition comprising a P2Y12 receptor antagonist
KR20240033005A (ko) 2021-07-13 2024-03-12 이도르시아 파마슈티컬스 리미티드 4-((r)-2-{[6-((s)-3-메톡시-피롤리딘-1-일)-2-페닐-피리미딘-4-카르보닐]-아미노}-3-포스포노-프로피오닐)-피페라진-1-카르복실산부틸 에스테르의 합성 방법
MX2024011264A (es) 2022-03-14 2024-09-23 Viatris Asia Pacific Pte Ltd Un proceso para la sintesis de acido (r)-2-((terc-butoxicarbonil)a mino)-3- (dietoxifosforil)propanoico o de derivados fosfonato del mismo.

Family Cites Families (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3870035A (en) 1970-07-17 1975-03-11 Survival Technology Method and apparatus for self-administering pre-hospital phase treatment of coronary prone individuals in the early minutes or hours after the onset of heart attack symptoms
US4004577A (en) 1972-12-04 1977-01-25 Survival Technology, Inc. Method of treating heart attack patients prior to the establishment of qualified direct contact personal care
JPS5373586A (en) 1976-12-09 1978-06-30 Mitsubishi Chem Ind Ltd New penicillin derivatives
US4795433A (en) 1985-05-20 1989-01-03 Survival Technology, Inc. Automatic injector for emergency treatment
US4658830A (en) 1984-08-08 1987-04-21 Survival Technology, Inc. Method and apparatus for initiating reperfusion treatment by an unattended individual undergoing heart attack symptoms
US5078680A (en) 1984-08-08 1992-01-07 Survival Technology, Inc. Automatic injector for emergency treatment
GR861289B (en) 1985-05-20 1986-09-16 Survival Technology Injection method and apparatus with electrical blood absorbing stimulation
CA2020437A1 (en) 1989-07-05 1991-01-06 Yoshihide Fuse Cinnamamide derivative
US6855715B1 (en) 1999-06-14 2005-02-15 Eli Lilly And Company Serine protease inhibitors
US6861424B2 (en) 2001-06-06 2005-03-01 Schering Aktiengesellschaft Platelet adenosine diphosphate receptor antagonists
CA2507657C (en) 2002-12-11 2011-05-31 Schering Aktiengesellschaft 2-aminocarbonyl-quinoline compounds as platelet adenosine diphosphate receptor antagonists
DK1611144T3 (da) 2003-04-09 2010-11-22 Wyeth Llc Derivater af 2-(8,9-dioxo-2,6-diazabicyclo(5.2.0)non-1(7)-en-2-yl)alkyl-phosphonsyre og deres avendelse som n-methyl-D-aspartat (NMDA)-receptor-antagonister
AU2003249865A1 (en) * 2003-06-24 2005-01-21 Actelion Pharmaceuticals Ltd Pyrazolidinedione derivatives and their use as platelet aggregation inhibitors
TW200640877A (en) 2005-04-28 2006-12-01 Actelion Pharmaceuticals Ltd Pyrimidine derivatives
RU2423358C2 (ru) 2005-10-21 2011-07-10 Актелион Фармасьютиклз Лтд Новые пиперазины в качестве антималярийных агентов
AR063258A1 (es) 2006-10-13 2009-01-14 Actelion Pharmaceuticals Ltd Derivados de 2-aminocarbonil-piridina, una composicion farmaceutica que los contiene y su uso en la preparacion de un medicamento para el tratamiento de trastornos vasculares oclusivos.
CL2007003038A1 (es) 2006-10-25 2008-06-06 Actelion Pharmaceuticals Ltd Compuestos derivados de 2-fenil-6-aminocarbonil-pirimidina; composicion farmaceutica; y uso en el tratamiento de trastornos vasculares oclusivos.
JP4785881B2 (ja) 2007-02-27 2011-10-05 大塚製薬株式会社 医薬
MY153427A (en) 2007-04-23 2015-02-13 Sanofi Aventis Quinoline-carboxamide derivatives as p2y12 antagonists
US20090048216A1 (en) 2007-05-02 2009-02-19 Portola Pharmaceuticals, Inc. Intravenous and oral dosing of a direct-acting and reversible p2y12 inhibitor
SI2225253T1 (sl) 2007-11-29 2012-09-28 Actelion Pharmaceuticals Ltd Derivati fosfonske kisline in njihova uporaba kot antagonisti receptorja P2Y12
WO2009080227A2 (en) 2007-12-26 2009-07-02 Sanofi-Aventis Pyrazole-carboxamide derivatives as p2y12 antagonists
JP5504171B2 (ja) 2007-12-26 2014-05-28 サノフイ P2y12アンタゴニストとしてのヘテロサイクリックピラゾール−カルボキサミド
AR071652A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2- fenil-piridina substituidos
AR071653A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2-fenil-4-ciclopropil-pirimidina
CA2756542C (en) 2009-04-08 2017-08-22 Actelion Pharmaceuticals Ltd 6-(3-aza-bicyclo[3.1.0]hex-3-yl)-2-phenyl-pyrimidines
CN102405220B (zh) 2009-04-22 2015-05-27 埃科特莱茵药品有限公司 噻唑衍生物及其作为p2y12受体拮抗剂的用途
WO2011137459A1 (en) 2010-04-30 2011-11-03 Portola Pharmaceuticals, Inc. Dosage forms of elinogrel and methods of injectable administration thereof
EP2585161A1 (en) 2010-06-23 2013-05-01 Stefan Kralev Medical device for self-administration of patients with acute coronary events
KR102552795B1 (ko) 2016-09-22 2023-07-06 이도르시아 파마슈티컬스 리미티드 결정질 형태

Also Published As

Publication number Publication date
WO2018167139A1 (en) 2018-09-20
NZ757938A (en) 2024-07-05
US11179390B2 (en) 2021-11-23
PH12019502111A1 (en) 2020-03-16
AU2018234056A1 (en) 2019-10-31
MX2019009559A (es) 2019-10-15
JP2023052576A (ja) 2023-04-11
EP3595666A1 (en) 2020-01-22
AU2018234056B2 (en) 2023-05-25
UA125531C2 (uk) 2022-04-13
JP7580918B2 (ja) 2024-11-12
KR102510832B1 (ko) 2023-03-15
TW201840323A (zh) 2018-11-16
IL269286B2 (en) 2023-08-01
TWI765002B (zh) 2022-05-21
BR112019014567A2 (pt) 2020-02-18
MY205605A (en) 2024-10-29
CN110381947A (zh) 2019-10-25
JP2020510043A (ja) 2020-04-02
KR20190124297A (ko) 2019-11-04
SG11201908128YA (en) 2019-10-30
CA3050831A1 (en) 2018-09-20
IL269286A (en) 2019-11-28
EA201992123A1 (ru) 2020-02-25
IL269286B1 (en) 2023-04-01
US20200129510A1 (en) 2020-04-30
CL2019002318A1 (es) 2020-01-10

Similar Documents

Publication Publication Date Title
FIC20240021I1 (fi) Adagrasibi tai sen farmaseuttisesti hyväksyttävä suola
MA41117A (fr) Imagerie d'un corps
HUE059827T2 (hu) VEGF-antagonista alkalmazása angiogén szembetegségek kezelésére
EP3888593C0 (en) Biceps tenodesis delivery tools
EP3344295A4 (en) CHIMERIC ANTI-SIALYL TN ANTIGEN RECEPTORS
MA49887A (fr) Administration sous-cutanée d'un antagoniste du récepteur p2y12
IL271777A (en) Preparations for intravenous administration of medical substances
LT3713928T (lt) Nauji bradikinino b2 receptoriaus antagonistai
EA201890156A1 (ru) Антагонисты рецептора cgrp
EP3334413A4 (en) DISPENSER
MA54761A (fr) Administration d'un inhibiteur de signalisation de trans-signalisation par il-6 sélectif
DK3914321T3 (da) Lægemiddeladministrationsanordning
IL283673A (en) Deuterated analogs of acetyl-leucine
MA42689A (fr) Micropropagation d'un dattier t-r
MA42698A (fr) Micropropagation d'un dattier hdt
FR3027173B1 (fr) Architecture d'un reseau de telecommunication
IL271694A (en) Novel uses of a pure 6HT–5 receptor antagonist
EP3854781A4 (en) DP ANTAGONIST
EP3368401A4 (en) ANCHOR ADAPTER
EP3668703A4 (en) Selective deposit of a functional agent
DK3512518T3 (da) Buprenophinformuleringer med langvarig frigivelse
EP3406614A4 (en) OPIOID RECEPTOR ANTAGONIST CONJUGATE AND USE THEREOF
HUE055083T2 (hu) Tiszta 5-HT6 receptor antagonisztika kombinációja az NMDA receptor antagonistájával
FR3030165B1 (fr) Synchronisation d'un reseau cpl
DK3681564T3 (da) Lægemiddeladministrationsanordning