MA41253A - Composés, compositions et procédés pour augmenter l'activité du cftr - Google Patents
Composés, compositions et procédés pour augmenter l'activité du cftrInfo
- Publication number
- MA41253A MA41253A MA041253A MA41253A MA41253A MA 41253 A MA41253 A MA 41253A MA 041253 A MA041253 A MA 041253A MA 41253 A MA41253 A MA 41253A MA 41253 A MA41253 A MA 41253A
- Authority
- MA
- Morocco
- Prior art keywords
- cftr
- compositions
- activity
- compounds
- processes
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
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- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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- A61K31/4245—Oxadiazoles
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
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WO2016105485A2 (fr) | 2016-06-30 |
CN107207487B (zh) | 2021-12-28 |
ES2962673T3 (es) | 2024-03-20 |
AU2015371294A1 (en) | 2017-06-29 |
BR112017013710A2 (pt) | 2018-01-02 |
US20170369480A1 (en) | 2017-12-28 |
JP6700284B2 (ja) | 2020-05-27 |
AU2022228100A1 (en) | 2022-09-29 |
EP3237411B1 (fr) | 2023-06-07 |
NZ732701A (en) | 2022-12-23 |
SA517381828B1 (ar) | 2022-09-07 |
KR20170096034A (ko) | 2017-08-23 |
US10392372B2 (en) | 2019-08-27 |
RU2017126232A3 (fr) | 2019-06-17 |
US11098035B2 (en) | 2021-08-24 |
EP3237411A2 (fr) | 2017-11-01 |
CA2971858A1 (fr) | 2016-06-30 |
CN107207487A (zh) | 2017-09-26 |
IL276426A (en) | 2020-09-30 |
RU2767460C2 (ru) | 2022-03-17 |
AU2020256305A1 (en) | 2020-11-12 |
WO2016105485A3 (fr) | 2016-09-01 |
IL252987A0 (en) | 2017-08-31 |
MX2017008380A (es) | 2018-04-11 |
SG11201704859UA (en) | 2017-07-28 |
IL252987B (en) | 2020-08-31 |
JP2018500343A (ja) | 2018-01-11 |
AU2015371294B2 (en) | 2020-07-16 |
KR102677444B1 (ko) | 2024-06-20 |
US20200190072A1 (en) | 2020-06-18 |
RU2017126232A (ru) | 2019-01-29 |
BR112017013710B1 (pt) | 2023-11-07 |
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