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MA32834B1 - 3-aminocyclopentanecarboxamides servant de modulateurs de recepteurs de chimiokines - Google Patents

3-aminocyclopentanecarboxamides servant de modulateurs de recepteurs de chimiokines

Info

Publication number
MA32834B1
MA32834B1 MA33895A MA33895A MA32834B1 MA 32834 B1 MA32834 B1 MA 32834B1 MA 33895 A MA33895 A MA 33895A MA 33895 A MA33895 A MA 33895A MA 32834 B1 MA32834 B1 MA 32834B1
Authority
MA
Morocco
Prior art keywords
shimokin
aminocyclopentaneicarboxamide
acts
receptor modulator
formulas
Prior art date
Application number
MA33895A
Other languages
Arabic (ar)
English (en)
Inventor
Rajesh Venkateswaran Devraj
Wei Huang
Robert Owen Hughes
Jr Donald Joseph Rogier
John Isidro Trujillo
Steve Ronald Turner
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MA32834B1 publication Critical patent/MA32834B1/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P3/02—Nutrients, e.g. vitamins, minerals
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    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
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    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
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    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Transplantation (AREA)
  • Vascular Medicine (AREA)
  • Nutrition Science (AREA)
  • Hospice & Palliative Care (AREA)
  • Virology (AREA)
  • Ophthalmology & Optometry (AREA)

Abstract

L'invention porte sur un composé de formule I(a) ou I(b) ou sur un sel pharmaceutiquement acceptable de celui-ci. Dans les formules, les divers substituants sont tels que définis dans la description.
MA33895A 2008-11-26 2011-05-26 3-aminocyclopentanecarboxamides servant de modulateurs de recepteurs de chimiokines MA32834B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11805308P 2008-11-26 2008-11-26
PCT/IB2009/055232 WO2010061329A1 (fr) 2008-11-26 2009-11-20 3-aminocyclopentanecarboxamides en tant que modulateurs des récepteurs de chimiokines

Publications (1)

Publication Number Publication Date
MA32834B1 true MA32834B1 (fr) 2011-11-01

Family

ID=41693100

Family Applications (1)

Application Number Title Priority Date Filing Date
MA33895A MA32834B1 (fr) 2008-11-26 2011-05-26 3-aminocyclopentanecarboxamides servant de modulateurs de recepteurs de chimiokines

Country Status (39)

Country Link
US (2) US8293903B2 (fr)
EP (1) EP2370442B9 (fr)
JP (1) JP5108153B2 (fr)
KR (1) KR101374412B1 (fr)
CN (1) CN102227429B (fr)
AP (1) AP3113A (fr)
AU (1) AU2009321221B2 (fr)
BR (1) BRPI0920936A2 (fr)
CA (1) CA2743030C (fr)
CL (1) CL2011001223A1 (fr)
CO (1) CO6361921A2 (fr)
CR (1) CR20110275A (fr)
CU (1) CU24022B1 (fr)
CY (1) CY1114020T1 (fr)
DK (1) DK2370442T5 (fr)
DO (1) DOP2011000154A (fr)
EA (1) EA020470B1 (fr)
EC (1) ECSP11011081A (fr)
ES (1) ES2415430T3 (fr)
GE (1) GEP20146064B (fr)
HK (1) HK1161261A1 (fr)
HR (1) HRP20130409T2 (fr)
IL (1) IL212732A (fr)
MA (1) MA32834B1 (fr)
ME (1) ME01144B (fr)
MX (1) MX2011005526A (fr)
MY (1) MY152557A (fr)
NI (1) NI201100102A (fr)
NZ (1) NZ592919A (fr)
PE (1) PE20110831A1 (fr)
PL (1) PL2370442T3 (fr)
PT (1) PT2370442E (fr)
RS (2) RS52810B9 (fr)
SI (1) SI2370442T1 (fr)
SV (1) SV2011003923A (fr)
TN (1) TN2011000254A1 (fr)
UA (1) UA99978C2 (fr)
WO (1) WO2010061329A1 (fr)
ZA (1) ZA201104069B (fr)

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Publication number Priority date Publication date Assignee Title
PE20110831A1 (es) * 2008-11-26 2011-11-20 Pfizer 3-aminociclopentanocarboxamidas como moduladores del receptor de quimiocina
KR101303963B1 (ko) * 2011-04-08 2013-09-05 재단법인 경기과학기술진흥원 (1ｒ,2ｒ,3ｒ)-3-아미노사이클로펜탄-1,2-디올을 포함하는 항알러지용 조성물
CN106659765B (zh) 2014-04-04 2021-08-13 德玛医药 二脱水半乳糖醇及其类似物或衍生物用于治疗非小细胞肺癌和卵巢癌的用途
JP2016029038A (ja) * 2014-07-17 2016-03-03 参天製薬株式会社 加齢黄斑変性の予防または治療剤
JOP20190040A1 (ar) * 2016-09-14 2019-03-10 Novartis Ag توليفة من ناهضات fxr
TWI830733B (zh) * 2018-05-11 2024-02-01 中國大陸商迪哲（江蘇）醫藥有限公司 環戊烷化合物
JP7412034B1 (ja) 2022-11-02 2024-01-12 鈴木製機株式会社 搬送システム

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Also Published As

Publication number Publication date
ES2415430T3 (es) 2013-07-25
HK1161261A1 (en) 2012-08-24
CR20110275A (es) 2011-07-01
AU2009321221B2 (en) 2013-04-04
RS52810B9 (sr) 2019-06-28
ES2415430T9 (es) 2013-11-25
AU2009321221A1 (en) 2010-06-03
EP2370442B1 (fr) 2013-04-24
GEP20146064B (en) 2014-03-25
SV2011003923A (es) 2011-07-28
RS52810B (en) 2013-10-31
US8946413B2 (en) 2015-02-03
CN102227429B (zh) 2014-05-28
CL2011001223A1 (es) 2011-09-02
JP2012509931A (ja) 2012-04-26
CA2743030C (fr) 2013-10-22
WO2010061329A1 (fr) 2010-06-03
ECSP11011081A (es) 2011-12-30
CA2743030A1 (fr) 2010-06-03
TN2011000254A1 (fr) 2012-12-17
PL2370442T3 (pl) 2013-08-30
MY152557A (en) 2014-10-31
CO6361921A2 (es) 2012-01-20
EA020470B1 (ru) 2014-11-28
PT2370442E (pt) 2013-06-27
KR20110075036A (ko) 2011-07-05
DK2370442T3 (da) 2013-06-17
IL212732A (en) 2016-06-30
AP3113A (en) 2015-01-31
EP2370442A1 (fr) 2011-10-05
AP2011005732A0 (en) 2011-06-30
BRPI0920936A2 (pt) 2020-08-11
ME01144B (me) 2013-03-20
HRP20130409T2 (hr) 2013-11-22
MX2011005526A (es) 2011-06-06
ZA201104069B (en) 2012-02-29
JP5108153B2 (ja) 2012-12-26
DOP2011000154A (es) 2011-07-31
KR101374412B1 (ko) 2014-03-17
DK2370442T5 (da) 2013-09-23
US20130197008A1 (en) 2013-08-01
CU20110121A7 (es) 2013-05-31
CU24022B1 (es) 2014-07-30
IL212732A0 (en) 2011-07-31
RS52810B8 (sr) 2019-08-30
EP2370442B9 (fr) 2013-09-04
HRP20130409T1 (en) 2013-06-30
EA201170721A1 (ru) 2011-12-30
UA99978C2 (en) 2012-10-25
NZ592919A (en) 2013-05-31
SI2370442T1 (sl) 2013-06-28
NI201100102A (es) 2011-09-27
US20110144129A1 (en) 2011-06-16
US8293903B2 (en) 2012-10-23
PE20110831A1 (es) 2011-11-20
CN102227429A (zh) 2011-10-26
CY1114020T1 (el) 2016-07-27

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