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LU91306I2 - Mitratapide, optionnellement sous forme d'un sel d'addition acide pharmaceutiquement acceptable (YARVITAN) - Google Patents

Mitratapide, optionnellement sous forme d'un sel d'addition acide pharmaceutiquement acceptable (YARVITAN)

Info

Publication number
LU91306I2
LU91306I2 LU91306C LU91306C LU91306I2 LU 91306 I2 LU91306 I2 LU 91306I2 LU 91306 C LU91306 C LU 91306C LU 91306 C LU91306 C LU 91306C LU 91306 I2 LU91306 I2 LU 91306I2
Authority
LU
Luxembourg
Prior art keywords
yarvitan
mitratapide
optionally
pharmaceutically acceptable
acid addition
Prior art date
Application number
LU91306C
Other languages
English (en)
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/455,304 external-priority patent/US5521186A/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of LU91306I2 publication Critical patent/LU91306I2/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
LU91306C 1994-10-27 2007-01-17 Mitratapide, optionnellement sous forme d'un sel d'addition acide pharmaceutiquement acceptable (YARVITAN) LU91306I2 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP94203120 1994-10-27
US08/455,304 US5521186A (en) 1994-10-27 1995-05-31 Apolipoprotein-β synthesis inhibitors
PCT/EP1995/004111 WO1996013499A1 (fr) 1994-10-27 1995-10-19 Inhibiteurs de synthese d'apolipoproteines-b

Publications (1)

Publication Number Publication Date
LU91306I2 true LU91306I2 (fr) 2007-03-19

Family

ID=26136684

Family Applications (1)

Application Number Title Priority Date Filing Date
LU91306C LU91306I2 (fr) 1994-10-27 2007-01-17 Mitratapide, optionnellement sous forme d'un sel d'addition acide pharmaceutiquement acceptable (YARVITAN)

Country Status (30)

Country Link
US (1) US5929075A (fr)
EP (1) EP0788496B1 (fr)
JP (1) JP3025907B2 (fr)
KR (1) KR100227231B1 (fr)
CN (1) CN1068000C (fr)
AP (1) AP779A (fr)
AT (1) ATE198889T1 (fr)
AU (1) AU697744C (fr)
BG (1) BG63694B1 (fr)
BR (1) BR9509436A (fr)
CA (1) CA2203274C (fr)
CY (1) CY2256B1 (fr)
CZ (1) CZ286476B6 (fr)
DE (3) DE122007000005I2 (fr)
DK (1) DK0788496T3 (fr)
ES (1) ES2155535T3 (fr)
FI (1) FI119548B (fr)
GR (1) GR3035519T3 (fr)
HR (1) HRP950532B1 (fr)
HU (1) HU219862B (fr)
IL (1) IL115771A (fr)
LU (1) LU91306I2 (fr)
NO (1) NO311937B1 (fr)
NZ (1) NZ295353A (fr)
OA (1) OA10479A (fr)
PT (1) PT788496E (fr)
RO (1) RO118715B1 (fr)
SK (1) SK281908B6 (fr)
TR (1) TR199501295A2 (fr)
WO (1) WO1996013499A1 (fr)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU746890B2 (en) * 1997-11-03 2002-05-02 Janssen Pharmaceutica N.V. Compositions of lipid lowering agents
EE200000796A (et) * 1998-04-27 2002-06-17 Janssen Pharmaceutica N.V. Ravimkuulike, selle valmistamismeetod ja farmatseutiline doseerimisvorm, ravimkuulikeste kasutaminefarmatseutilise doseerimisvormi valmistamiseks ning farmatseutiline pakend
CA2355822A1 (fr) * 1998-12-22 2000-06-29 Janssen Pharmaceutica N.V. Composes s-oxide permettant d'abaisser le taux de lipides
DE19945982A1 (de) 1999-09-24 2001-03-29 Knoll Ag Geschwindigkeitsbestimmte Partikel
US20050132022A1 (en) * 2003-12-12 2005-06-16 International Business Machines Corporation Computer system with LAN-based I/O
AU2005205933B2 (en) * 2004-01-21 2010-02-18 Elanco Animal Health Ireland Limited Mitratapide oral solution
US7649002B2 (en) 2004-02-04 2010-01-19 Pfizer Inc (3,5-dimethylpiperidin-1yl)(4-phenylpyrrolidin-3-yl)methanone derivatives as MCR4 agonists
US7262318B2 (en) * 2004-03-10 2007-08-28 Pfizer, Inc. Substituted heteroaryl- and phenylsulfamoyl compounds
CA2562015A1 (fr) * 2004-04-09 2005-10-20 Janssen Pharmaceutica Nv Schema posologique intermittent destine a des sujets obeses ou en surpoids
US20050288340A1 (en) * 2004-06-29 2005-12-29 Pfizer Inc Substituted heteroaryl- and phenylsulfamoyl compounds
PA8660701A1 (es) 2005-02-04 2006-09-22 Pfizer Prod Inc Agonistas de pyy y sus usos
WO2006129193A2 (fr) * 2005-05-27 2006-12-07 Pfizer Products Inc. Polytherapie pour le traitement de l'obesite ou le maintien du poids apres une perte ponderale
JP2009503050A (ja) * 2005-08-04 2009-01-29 ファイザー・リミテッド ピペリジノイル−ピロリジンおよびピペリジノイル−ピペリジン化合物
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
DK1989196T3 (da) * 2006-02-23 2013-04-15 Pfizer Ltd Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister
US8383660B2 (en) 2006-03-10 2013-02-26 Pfizer Inc. Dibenzyl amine compounds and derivatives
WO2008059335A1 (fr) 2006-11-13 2008-05-22 Pfizer Products Inc. Dérivés diaryle, dipyridinyle et aryl-pyridinyle et leurs utilisations
WO2008070496A2 (fr) 2006-12-01 2008-06-12 Bristol-Myers Squibb Company Inhibiteurs d'amino cetp étendus
US8765979B2 (en) 2007-05-25 2014-07-01 Janssen Pharmaceutica Synthesis of (2S-cis)-2-(bromomethyl)-2-(4-chlorophenyl)-1,3 dioxolane-4-methanol methanesulfonate(ester)
JP5530438B2 (ja) * 2008-08-06 2014-06-25 ファイザー・リミテッド Ｍｃ４作動薬としてのジアゼピンおよびジアゾカン化合物
WO2011144653A1 (fr) * 2010-05-19 2011-11-24 Sandoz Ag Procédé pour la préparation de triazolones chirales
CN112074505B (zh) 2018-03-08 2024-04-05 因赛特公司 作为PI3K-γ抑制剂的氨基吡嗪二醇化合物
US11046658B2 (en) 2018-07-02 2021-06-29 Incyte Corporation Aminopyrazine derivatives as PI3K-γ inhibitors

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4218458A (en) * 1978-06-23 1980-08-19 Janssen Pharmaceutica, N.V. Heterocyclic derivatives of (4-aryloxy-methyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles
US4313953A (en) * 1978-06-23 1982-02-02 Janssen Pharmaceutica, N.V. Heterocyclic derivatives of (4-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles
US4766125A (en) * 1981-06-23 1988-08-23 Janssen Pharmaceutica N.V. N-aryl-piperazinealkanamides useful for protecting hearts from myocardial injury caused by ischaemia, anoxia or hypoxia
US4619931A (en) * 1983-02-28 1986-10-28 Janssen Pharmaceutica, N.V. [[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles
CA1292472C (fr) * 1985-12-03 1991-11-26 Alfonsus Guilielmus Knaeps Derives des ({4-¬4-(4-phenyl-1-piperazinyl)-phenoxymethyl|- 1,3-dioxolan-2-yl}methyl)-1h-imidazoles et 1h-1,2,4-triazoles
NZ223799A (en) * 1987-03-25 1989-12-21 Janssen Pharmaceutica Nv Azolylmethyl-dioxolanylmethoxyphenyl-piperazinyl-phenyl-triazolones and antimicrobial compositions
CA1331757C (fr) * 1988-02-29 1994-08-30 Janssen Pharmaceutica Naamloze Vennootschap 5-lipoxygenase inhibant les 4-(4-phenyl-1-piperazinyl)phenols
AU6359594A (en) * 1993-03-04 1994-09-26 Cytoven International N.V. Pharmaceutical tryptophan containing dipeptide compositions and methods of use thereof
US5521186A (en) * 1994-10-27 1996-05-28 Janssen Pharmaceutica N.V. Apolipoprotein-β synthesis inhibitors

Also Published As

Publication number Publication date
EP0788496A1 (fr) 1997-08-13
EP0788496B1 (fr) 2001-01-24
NO971895D0 (no) 1997-04-24
DE69519995T2 (de) 2001-08-23
CY2256B1 (en) 2003-07-04
CA2203274C (fr) 2002-02-19
SK281908B6 (sk) 2001-09-11
CN1068000C (zh) 2001-07-04
NO971895L (no) 1997-04-24
FI119548B (fi) 2008-12-31
CA2203274A1 (fr) 1996-05-09
ATE198889T1 (de) 2001-02-15
DE122007000005I1 (de) 2007-04-26
NO311937B1 (no) 2002-02-18
US5929075A (en) 1999-07-27
WO1996013499A1 (fr) 1996-05-09
HU219862B (hu) 2001-08-28
AU697744C (en) 2002-08-22
IL115771A0 (en) 1996-01-19
IL115771A (en) 2000-02-29
BG101402A (en) 1997-10-31
HRP950532B1 (en) 2001-06-30
CZ286476B6 (en) 2000-04-12
JP3025907B2 (ja) 2000-03-27
AP9700968A0 (en) 1997-04-30
DK0788496T3 (da) 2001-06-18
HUT77360A (hu) 1998-03-30
CN1161695A (zh) 1997-10-08
RO118715B1 (ro) 2003-09-30
NZ295353A (en) 1998-08-26
TR199501295A2 (tr) 1996-06-21
AU697744B2 (en) 1998-10-15
AP779A (en) 1999-11-03
BG63694B1 (bg) 2002-09-30
DE122007000005I2 (de) 2008-04-24
SK50797A3 (en) 1998-04-08
JPH09511759A (ja) 1997-11-25
KR100227231B1 (ko) 1999-11-01
FI971784A (fi) 1997-04-25
ES2155535T3 (es) 2001-05-16
GR3035519T3 (en) 2001-06-29
BR9509436A (pt) 1998-01-06
DE69519995D1 (en) 2001-03-01
MX9703074A (es) 1997-07-31
CZ119897A3 (cs) 1998-03-18
AU3868095A (en) 1996-05-23
PT788496E (pt) 2001-07-31
OA10479A (en) 2002-04-09
FI971784A0 (fi) 1997-04-25
HRP950532A2 (en) 1997-08-31

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