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KR860007276A - 글리코시드 및 그 제조방법 - Google Patents

글리코시드 및 그 제조방법 Download PDF

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Publication number
KR860007276A
KR860007276A KR1019860001555A KR860001555A KR860007276A KR 860007276 A KR860007276 A KR 860007276A KR 1019860001555 A KR1019860001555 A KR 1019860001555A KR 860001555 A KR860001555 A KR 860001555A KR 860007276 A KR860007276 A KR 860007276A
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KR
South Korea
Prior art keywords
group
carboxyl group
salt
alkoxycarbonyl
carboxyl
Prior art date
Application number
KR1019860001555A
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English (en)
Other versions
KR880000704B1 (ko
Inventor
쇼헤이 시바야마
유지 마쯔자끼
쇼지 요시무라
마사요시 이토오
요시야수 시토리
도모야 오가와
Original Assignee
간도오이시세이야꾸 가부시끼가이샤
곤도오 야스노리
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Publication of KR860007276A publication Critical patent/KR860007276A/ko
Application granted granted Critical
Publication of KR880000704B1 publication Critical patent/KR880000704B1/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H3/00—Compounds containing only hydrogen atoms and saccharide radicals having only carbon, hydrogen, and oxygen atoms
    • C07H3/06—Oligosaccharides, i.e. having three to five saccharide radicals attached to each other by glycosidic linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H9/00—Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical
    • C07H9/06—Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical the hetero ring containing nitrogen as ring hetero atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

내용 없음

Description

글리코시드 및 그 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (8)

  1. 일반식
    을 갖는 글리코시드
    여기에서, R1은
    기, 알콕시카르보닐기, 가르목실기 및 카르복실기의 염에서 선택되며,
    R1이
    기일때, R2는 알콕시 카르보닐기, 카르복실기 또는 카르복실기의 염이고,
    R1이 알콕시카르보닐기, 카르복실기 또는 카르복실기의 염일대, R2는
    기이며,
    R3는 수소원자 또는 아세틸기이다.
  2. 제 1 항에 있어서, R1은
    기이고, R2는 알콕시카르보닐기, 카르복실기 및 카르복실기의 염인 글리코시드.
  3. 제 1 항에 있어서, R1은 알콕시카르보닐기, 카르보닐기 또는 카르복실기의 염이고, R2는
    기인 글리코시드
  4. 제 1 항에 있어서, 알콕시카르보닐기는 메톡시카르보닐기인 글리코시드.
  5. 일반식
    를
    갖는 글리코시드의 제조방법.
    여기에서, R4는 아세틸기, R5는 메톡시카르보닐기 그리고 R6는 트리플루오로메탄황산화은(silver trifluoromethane sulfonate)의 존재하에
    (Ⅱ)
    와의 반응으로 구성되는
    기이다.
  6. 제 5 항에 있어서, 반응은 용매내에서 수행되는 글리코시드의 제조방법.
  7. 제 6 항에 있어서, 용매는 테트라히드로푸란, 아세토니트릴 및 염화메틸렌에서 선택되는 글리코시드의 제조방법.
  8. 제 5 항에 있어서, 반응은 실온내지 -50℃에서 약 5 내지 60분간 수행되는 글리코시드의 제조방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019860001555A 1985-03-06 1986-03-05 글리 코시드의 제조방법 KR880000704B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP43970 1985-03-06
JP60043970A JPS61204190A (ja) 1985-03-06 1985-03-06 グリコシド及びその製造方法
JP?60-43970 1985-03-06

Publications (2)

Publication Number Publication Date
KR860007276A true KR860007276A (ko) 1986-10-10
KR880000704B1 KR880000704B1 (ko) 1988-04-25

Family

ID=12678563

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019860001555A KR880000704B1 (ko) 1985-03-06 1986-03-05 글리 코시드의 제조방법

Country Status (12)

Country Link
US (1) US4675391A (ko)
EP (1) EP0194563A3 (ko)
JP (1) JPS61204190A (ko)
KR (1) KR880000704B1 (ko)
CN (1) CN1018646B (ko)
AU (1) AU561320B2 (ko)
ES (1) ES8704180A1 (ko)
FI (1) FI79543C (ko)
HU (1) HU195228B (ko)
MC (1) MC1740A1 (ko)
NO (1) NO164660C (ko)
ZA (1) ZA861619B (ko)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1262130A (en) * 1985-10-11 1989-10-03 Shoji Yoshimura Process for preparing n-glycolylneuraminic acid derivatives
JPS6287598A (ja) * 1985-10-11 1987-04-22 Mect Corp Ｎ−グリコリルノイラミン酸誘導体
JP2517293B2 (ja) * 1987-06-25 1996-07-24 メクト株式会社 細胞、組織修復剤
AU7176091A (en) * 1989-12-29 1991-07-24 Symex Corp. Chromogenic 7- or 8-position modified n-acetylneuraminic acid substrates and methods for diagnosing human influenza therewith
CN1309685C (zh) * 2002-03-26 2007-04-11 佐治亚-太平洋树脂公司 缓释氮肥

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4248999A (en) * 1976-10-28 1981-02-03 Sankyo Company Limited 5-Fluorouracil derivatives and process for preparing thereof
JPS5738774A (en) * 1980-08-19 1982-03-03 Chugai Pharmaceut Co Ltd Uracil derivative and its preparation
DE3474632D1 (en) * 1983-03-01 1988-11-24 Crc Ricerca Chim Pharmaceutical compositions containing the cytidine monophosphate of 5-acetamido-3,5-dideoxy-d-glycero-d-galactononulosaminic acid
JPS60181295A (ja) * 1984-02-27 1985-09-14 Pentel Kk 酸化皮膜を有するアルミニウムまたはアルミニウム合金基体の製造方法

Also Published As

Publication number Publication date
FI860930A0 (fi) 1986-03-05
ES8704180A1 (es) 1987-03-16
HU195228B (en) 1988-04-28
EP0194563A3 (en) 1988-06-01
NO164660B (no) 1990-07-23
AU5411686A (en) 1986-09-11
ES552676A0 (es) 1987-03-16
FI79543C (fi) 1990-01-10
EP0194563A2 (en) 1986-09-17
NO860837L (ko) 1986-09-08
JPH0560474B2 (ko) 1993-09-02
NO164660C (no) 1990-10-31
MC1740A1 (fr) 1987-02-26
KR880000704B1 (ko) 1988-04-25
ZA861619B (en) 1986-11-26
CN1018646B (zh) 1992-10-14
JPS61204190A (ja) 1986-09-10
HUT42501A (en) 1987-07-28
FI860930A (fi) 1986-09-07
CN86102125A (zh) 1987-01-07
AU561320B2 (en) 1987-05-07
US4675391A (en) 1987-06-23
FI79543B (fi) 1989-09-29

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