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KR840009110A - 알파-아미노 벤질 페니실린의 에스테르 화합물의 제조방법 - Google Patents

알파-아미노 벤질 페니실린의 에스테르 화합물의 제조방법 Download PDF

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Publication number
KR840009110A
KR840009110A KR1019830002338A KR830002338A KR840009110A KR 840009110 A KR840009110 A KR 840009110A KR 1019830002338 A KR1019830002338 A KR 1019830002338A KR 830002338 A KR830002338 A KR 830002338A KR 840009110 A KR840009110 A KR 840009110A
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KR
South Korea
Prior art keywords
alpha
formula
ester compound
benzyl penicillin
amino benzyl
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Application number
KR1019830002338A
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English (en)
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KR850000612B1 (ko
Inventor
정재규, (외 1)
Original Assignee
김동회
주식회사 종근당
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by 김동회, 주식회사 종근당 filed Critical 김동회
Priority to KR1019830002338A priority Critical patent/KR850000612B1/ko
Publication of KR840009110A publication Critical patent/KR840009110A/ko
Application granted granted Critical
Publication of KR850000612B1 publication Critical patent/KR850000612B1/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Cephalosporin Compounds (AREA)

Abstract

내용 없음

Description

알파-아미노 벤질 페니실린의 에스테르 화합물의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (5)

  1. 공지의 화합물인 구조식(Ⅲ)의 메틸렌-(비스)-알파-아미노 페닐 아세트 아미노 페니실란산의 염을 비프로톤성 극성 용매중 상간 이동 촉매 존재하에 공지의 화합물 구조식(Ⅳ)의 알파-클로로 디에틸 카르보네이트와 반응시켜 구조식(Ⅴ)의 에스테르 화합물을 만든 다음 공지의 방법으로 가수 분해하여 구조식(Ⅰ)의 1′-에톡시 카르보닐 옥시에틸-6-[디(-)알파-아미니 페닐 아세트 아미도] 페니실라-네이트 염산염을 제조하는 방법.
  4. (상기 구조식에서 M은 알칼리 금속을 나타낸다)
  5. ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019830002338A 1983-05-27 1983-05-27 알파-아미노 벤질 페니실린의 에스테르 화합물의 제조 방법 KR850000612B1 (ko)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1019830002338A KR850000612B1 (ko) 1983-05-27 1983-05-27 알파-아미노 벤질 페니실린의 에스테르 화합물의 제조 방법

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
KR1019830002338A KR850000612B1 (ko) 1983-05-27 1983-05-27 알파-아미노 벤질 페니실린의 에스테르 화합물의 제조 방법

Publications (2)

Publication Number Publication Date
KR840009110A true KR840009110A (ko) 1984-12-24
KR850000612B1 KR850000612B1 (ko) 1985-05-01

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019830002338A KR850000612B1 (ko) 1983-05-27 1983-05-27 알파-아미노 벤질 페니실린의 에스테르 화합물의 제조 방법

Country Status (1)

Country Link
KR (1) KR850000612B1 (ko)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1375492B1 (en) * 2001-03-30 2011-08-17 Nippon Soda Co., Ltd. Process for producing (dioxolenon-4-yl)methyl ester derivative

Also Published As

Publication number Publication date
KR850000612B1 (ko) 1985-05-01

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