JPS5726686A - Preparation of indole derivative - Google Patents
Preparation of indole derivativeInfo
- Publication number
- JPS5726686A JPS5726686A JP9940280A JP9940280A JPS5726686A JP S5726686 A JPS5726686 A JP S5726686A JP 9940280 A JP9940280 A JP 9940280A JP 9940280 A JP9940280 A JP 9940280A JP S5726686 A JPS5726686 A JP S5726686A
- Authority
- JP
- Japan
- Prior art keywords
- indole
- preparation
- indole derivative
- derivative
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Plural Heterocyclic Compounds (AREA)
Abstract
PURPOSE: To obtain an indole derivative useful as an intermediate for synthesizing tryptophane in high yield, by reacting indole with an oxazolone derivative in the presence of a Lewis acid.
CONSTITUTION: Indole is reacted with an oxazolone derivative shown by the formula I (R is aryl; X is alkoxy or dialkylamino) in the presence of a Lewis acid (e.g., stannic chloride, etc.) in a solvent, e.g., dichloroethane, etc. at -10°C to room temperature for 1W24hr, to give a compound shown by the formula II.
COPYRIGHT: (C)1982,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP9940280A JPS5726686A (en) | 1980-07-22 | 1980-07-22 | Preparation of indole derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP9940280A JPS5726686A (en) | 1980-07-22 | 1980-07-22 | Preparation of indole derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS5726686A true JPS5726686A (en) | 1982-02-12 |
Family
ID=14246493
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP9940280A Pending JPS5726686A (en) | 1980-07-22 | 1980-07-22 | Preparation of indole derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5726686A (en) |
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS6136312A (en) * | 1984-07-27 | 1986-02-21 | Nippon Kasei Kk | Production of urea formaldehyde resin |
JPS6136311A (en) * | 1984-07-27 | 1986-02-21 | Nippon Kasei Kk | Production of urea formaldehyde resin |
WO1991007107A1 (en) * | 1989-11-13 | 1991-05-30 | Pfizer Inc. | Oxazolidinedione hypoglycemic agents |
US5498621A (en) * | 1992-05-01 | 1996-03-12 | Pfizer Inc. | Oxazolidinedione hypoglycemic agents |
-
1980
- 1980-07-22 JP JP9940280A patent/JPS5726686A/en active Pending
Cited By (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS6136312A (en) * | 1984-07-27 | 1986-02-21 | Nippon Kasei Kk | Production of urea formaldehyde resin |
JPS6136311A (en) * | 1984-07-27 | 1986-02-21 | Nippon Kasei Kk | Production of urea formaldehyde resin |
JPH0542454B2 (en) * | 1984-07-27 | 1993-06-28 | Nippon Kasei Chem | |
JPH0542455B2 (en) * | 1984-07-27 | 1993-06-28 | Nippon Kasei Chem | |
WO1991007107A1 (en) * | 1989-11-13 | 1991-05-30 | Pfizer Inc. | Oxazolidinedione hypoglycemic agents |
US5498621A (en) * | 1992-05-01 | 1996-03-12 | Pfizer Inc. | Oxazolidinedione hypoglycemic agents |
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