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JPS55100356A - Benzenediol derivative - Google Patents

Benzenediol derivative

Info

Publication number
JPS55100356A
JPS55100356A JP900779A JP900779A JPS55100356A JP S55100356 A JPS55100356 A JP S55100356A JP 900779 A JP900779 A JP 900779A JP 900779 A JP900779 A JP 900779A JP S55100356 A JPS55100356 A JP S55100356A
Authority
JP
Japan
Prior art keywords
phenyl
formula
phenylene
benzenediol
hydroxycynnamoyloxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP900779A
Other languages
Japanese (ja)
Inventor
Setsuo Fujii
Eizo Hattori
Munehiko Nara
Mitsuteru Hirata
Koichiro Watanabe
Masami Takimoto
Masahiko Nagakura
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kowa Co Ltd
Original Assignee
Kowa Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kowa Co Ltd filed Critical Kowa Co Ltd
Priority to JP900779A priority Critical patent/JPS55100356A/en
Publication of JPS55100356A publication Critical patent/JPS55100356A/en
Pending legal-status Critical Current

Links

Landscapes

  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Furan Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Indole Compounds (AREA)

Abstract

NEW MATERIAL:A benzenediol derviative or its acid addition salt of formula I [A is p-phenylene, or pentamethylene; B is -(CH2)n- (n is an integer of 0-2), or or -CH=CH-; R1 is (substituted) lower alkyl, phenyl, cyclohexyl, pyridyl, furyl, thienyl, naphthyl or indolyl, excluding the case that A is p-phenylene, B is -(CH2)2 - and R1 is phenyl].
EXAMPLE: p-(p-Hydroxycynnamoyloxy)phenyl p-guanidinobenzoate.
USE: Effective to inhibit the activity of proteinase, and useful as a remedy for pancreatic diseases of man and animal, an antiplasmic agent, and a preservative for fresh foods such as meat and fish.
PROCESS: Reaction of a hydroxybenzoate of formula II with a carboxylic acid of formula III or its reactive derivative affords the objective compound I.
COPYRIGHT: (C)1980,JPO&Japio
JP900779A 1979-01-29 1979-01-29 Benzenediol derivative Pending JPS55100356A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP900779A JPS55100356A (en) 1979-01-29 1979-01-29 Benzenediol derivative

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP900779A JPS55100356A (en) 1979-01-29 1979-01-29 Benzenediol derivative

Publications (1)

Publication Number Publication Date
JPS55100356A true JPS55100356A (en) 1980-07-31

Family

ID=11708588

Family Applications (1)

Application Number Title Priority Date Filing Date
JP900779A Pending JPS55100356A (en) 1979-01-29 1979-01-29 Benzenediol derivative

Country Status (1)

Country Link
JP (1) JPS55100356A (en)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0222608A2 (en) * 1985-11-12 1987-05-20 Ono Pharmaceutical Co., Ltd. Derivatives of p-guanidinobenzoic acid and pharmaceutical agents containing them as active ingredient
US4843094A (en) * 1985-11-12 1989-06-27 Ono Pharmaceutical Co., Ltd. Derivatives of p-guantidinobenzoic acid and pharmaceutical agents containing them as active ingredient
WO1991018869A1 (en) * 1990-06-08 1991-12-12 Asahi Kasei Kogyo Kabushiki Kaisha Phenyl 4-guanidinobenzoate derivative, process for producing the same, and protease inhibitor containing the same
US5376655A (en) * 1985-11-12 1994-12-27 Ono Pharmaceutical Co., Ltd. Derivatives of p-guanidinobenzoic acid and pharmaceutical agents containing them as an active ingredient
US6388122B1 (en) 1996-04-10 2002-05-14 Ono Pharmaceutical Co., Ltd. Tryptase inhibitor and novel guanidino derivatives

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS492107A (en) * 1972-04-19 1974-01-10
JPS53147044A (en) * 1977-05-25 1978-12-21 Ono Pharmaceut Co Ltd Guanidinobenzoic acid derivative and its preparation

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS492107A (en) * 1972-04-19 1974-01-10
JPS53147044A (en) * 1977-05-25 1978-12-21 Ono Pharmaceut Co Ltd Guanidinobenzoic acid derivative and its preparation

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0222608A2 (en) * 1985-11-12 1987-05-20 Ono Pharmaceutical Co., Ltd. Derivatives of p-guanidinobenzoic acid and pharmaceutical agents containing them as active ingredient
US4843094A (en) * 1985-11-12 1989-06-27 Ono Pharmaceutical Co., Ltd. Derivatives of p-guantidinobenzoic acid and pharmaceutical agents containing them as active ingredient
US5077428A (en) * 1985-11-12 1991-12-31 Ono Pharmaceutical Co., Ltd. Pharmacologically active derivatives of p-guanidinobenzoic acid
US5376655A (en) * 1985-11-12 1994-12-27 Ono Pharmaceutical Co., Ltd. Derivatives of p-guanidinobenzoic acid and pharmaceutical agents containing them as an active ingredient
WO1991018869A1 (en) * 1990-06-08 1991-12-12 Asahi Kasei Kogyo Kabushiki Kaisha Phenyl 4-guanidinobenzoate derivative, process for producing the same, and protease inhibitor containing the same
US6388122B1 (en) 1996-04-10 2002-05-14 Ono Pharmaceutical Co., Ltd. Tryptase inhibitor and novel guanidino derivatives

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