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ITFI20020239A1 - Processo per la preparazione di composti peptidici biciclici. - Google Patents

Processo per la preparazione di composti peptidici biciclici.

Info

Publication number
ITFI20020239A1
ITFI20020239A1 IT000239A ITFI20020239A ITFI20020239A1 IT FI20020239 A1 ITFI20020239 A1 IT FI20020239A1 IT 000239 A IT000239 A IT 000239A IT FI20020239 A ITFI20020239 A IT FI20020239A IT FI20020239 A1 ITFI20020239 A1 IT FI20020239A1
Authority
IT
Italy
Prior art keywords
preparation
compounds
bicyclic
peptid
intermediates
Prior art date
Application number
IT000239A
Other languages
English (en)
Inventor
Carlo Alberto Maggi
Stefano Manzini
Davide Poma
Aldo Salimbeni
Damiano Turozzi
Original Assignee
Menarini Ricerche Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Menarini Ricerche Spa filed Critical Menarini Ricerche Spa
Priority to IT000239A priority Critical patent/ITFI20020239A1/it
Priority to KR1020057009808A priority patent/KR101081256B1/ko
Priority to AT03782304T priority patent/ATE440105T1/de
Priority to JP2004557990A priority patent/JP4593284B2/ja
Priority to ES03782304T priority patent/ES2330102T3/es
Priority to PCT/EP2003/013696 priority patent/WO2004052923A2/en
Priority to CA2508696A priority patent/CA2508696C/en
Priority to AU2003289958A priority patent/AU2003289958A1/en
Priority to US10/537,731 priority patent/US7999068B2/en
Priority to PL377635A priority patent/PL207850B1/pl
Priority to CNB200380105180XA priority patent/CN1318445C/zh
Priority to EP03782304A priority patent/EP1576000B1/en
Priority to BR0317029-2A priority patent/BR0317029A/pt
Priority to MXPA05005969A priority patent/MXPA05005969A/es
Priority to DE60328915T priority patent/DE60328915D1/de
Priority to RU2005117345/04A priority patent/RU2330045C9/ru
Publication of ITFI20020239A1 publication Critical patent/ITFI20020239A1/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/22—Tachykinins, e.g. Eledoisins, Substance P; Related peptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IT000239A 2002-12-06 2002-12-06 Processo per la preparazione di composti peptidici biciclici. ITFI20020239A1 (it)

Priority Applications (16)

Application Number Priority Date Filing Date Title
IT000239A ITFI20020239A1 (it) 2002-12-06 2002-12-06 Processo per la preparazione di composti peptidici biciclici.
KR1020057009808A KR101081256B1 (ko) 2002-12-06 2003-12-04 바이사이클릭 펩타이드 화합물의 제조 방법
AT03782304T ATE440105T1 (de) 2002-12-06 2003-12-04 Verfahren zur herstellung von dem bicyclischen hexapeptide nepadutant
JP2004557990A JP4593284B2 (ja) 2002-12-06 2003-12-04 二環式ヘキサペプチド、ネパデュタントの製造方法
ES03782304T ES2330102T3 (es) 2002-12-06 2003-12-04 Proceso para la preparacion del hexapeptido biciclico nepadutant.
PCT/EP2003/013696 WO2004052923A2 (en) 2002-12-06 2003-12-04 Process for the preparation of bicyclic hexa-peptide nepadutant
CA2508696A CA2508696C (en) 2002-12-06 2003-12-04 Process for the preparation of bicyclic peptide compounds
AU2003289958A AU2003289958A1 (en) 2002-12-06 2003-12-04 Process for the preparation of bicyclic hexa-peptide nepadutant
US10/537,731 US7999068B2 (en) 2002-12-06 2003-12-04 Process for the preparation of bicyclic peptide compounds
PL377635A PL207850B1 (pl) 2002-12-06 2003-12-04 Sposób wytwarzania bicyklicznych związków peptydowych
CNB200380105180XA CN1318445C (zh) 2002-12-06 2003-12-04 双环肽化合物的制备方法
EP03782304A EP1576000B1 (en) 2002-12-06 2003-12-04 Process for the preparation of bicyclic hexa-peptide nepadutant
BR0317029-2A BR0317029A (pt) 2002-12-06 2003-12-04 Processo para a preparação de compostos peptìdicos bicìclicos
MXPA05005969A MXPA05005969A (es) 2002-12-06 2003-12-04 Proceso para la preparacion de compuestos peptidos biciclicos.
DE60328915T DE60328915D1 (de) 2002-12-06 2003-12-04 Verfahren zur herstellung von dem bicyclischen hexapeptide nepadutant
RU2005117345/04A RU2330045C9 (ru) 2002-12-06 2003-12-04 Способ получения бициклических пептидных соединений

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT000239A ITFI20020239A1 (it) 2002-12-06 2002-12-06 Processo per la preparazione di composti peptidici biciclici.

Publications (1)

Publication Number Publication Date
ITFI20020239A1 true ITFI20020239A1 (it) 2004-06-07

Family

ID=32500550

Family Applications (1)

Application Number Title Priority Date Filing Date
IT000239A ITFI20020239A1 (it) 2002-12-06 2002-12-06 Processo per la preparazione di composti peptidici biciclici.

Country Status (16)

Country Link
US (1) US7999068B2 (it)
EP (1) EP1576000B1 (it)
JP (1) JP4593284B2 (it)
KR (1) KR101081256B1 (it)
CN (1) CN1318445C (it)
AT (1) ATE440105T1 (it)
AU (1) AU2003289958A1 (it)
BR (1) BR0317029A (it)
CA (1) CA2508696C (it)
DE (1) DE60328915D1 (it)
ES (1) ES2330102T3 (it)
IT (1) ITFI20020239A1 (it)
MX (1) MXPA05005969A (it)
PL (1) PL207850B1 (it)
RU (1) RU2330045C9 (it)
WO (1) WO2004052923A2 (it)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007111952A2 (en) * 2006-03-22 2007-10-04 The Scripps Research Institute Method of preparing glycopeptides
CN103864901B (zh) * 2012-12-17 2017-02-08 深圳翰宇药业股份有限公司 一种制备奈帕坦特及其中间体的方法及所述中间体
CN109503698B (zh) * 2018-12-13 2021-01-01 无限极（中国）有限公司 一种多肽及其制备方法与应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1277835B1 (it) 1995-03-13 1997-11-12 Menarini Farma Ind Composti biciclici, loro preparazione ed uso in composizioni farmaceutiche

Also Published As

Publication number Publication date
JP4593284B2 (ja) 2010-12-08
WO2004052923A3 (en) 2005-02-24
EP1576000A2 (en) 2005-09-21
AU2003289958A8 (en) 2004-06-30
PL377635A1 (pl) 2006-02-06
EP1576000B1 (en) 2009-08-19
CA2508696C (en) 2014-05-06
MXPA05005969A (es) 2005-11-17
RU2005117345A (ru) 2006-02-27
CN1720260A (zh) 2006-01-11
RU2330045C9 (ru) 2008-11-20
US7999068B2 (en) 2011-08-16
ES2330102T3 (es) 2009-12-04
KR101081256B1 (ko) 2011-11-08
CN1318445C (zh) 2007-05-30
KR20050089966A (ko) 2005-09-09
PL207850B1 (pl) 2011-02-28
BR0317029A (pt) 2005-10-25
US20090163695A1 (en) 2009-06-25
CA2508696A1 (en) 2004-06-24
WO2004052923A2 (en) 2004-06-24
AU2003289958A1 (en) 2004-06-30
DE60328915D1 (de) 2009-10-01
JP2006520743A (ja) 2006-09-14
ATE440105T1 (de) 2009-09-15
RU2330045C2 (ru) 2008-07-27

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