IT8919049A0 - Procedimento per la preparazione di fluoxetina cloridrato. - Google Patents
Procedimento per la preparazione di fluoxetina cloridrato.Info
- Publication number
- IT8919049A0 IT8919049A0 IT8919049A IT1904989A IT8919049A0 IT 8919049 A0 IT8919049 A0 IT 8919049A0 IT 8919049 A IT8919049 A IT 8919049A IT 1904989 A IT1904989 A IT 1904989A IT 8919049 A0 IT8919049 A0 IT 8919049A0
- Authority
- IT
- Italy
- Prior art keywords
- procedure
- preparation
- fluoxetine hydrochloride
- fluoxetine
- hydrochloride
- Prior art date
Links
- GIYXAJPCNFJEHY-UHFFFAOYSA-N N-methyl-3-phenyl-3-[4-(trifluoromethyl)phenoxy]-1-propanamine hydrochloride (1:1) Chemical compound Cl.C=1C=CC=CC=1C(CCNC)OC1=CC=C(C(F)(F)F)C=C1 GIYXAJPCNFJEHY-UHFFFAOYSA-N 0.000 title 1
- 229960000389 fluoxetine hydrochloride Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/08—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions not involving the formation of amino groups, hydroxy groups or etherified or esterified hydroxy groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT8919049A IT1228209B (it) | 1989-01-10 | 1989-01-10 | Procedimento per la preparazione di fluoxetina cloridrato. |
AT90100314T ATE107623T1 (de) | 1989-01-10 | 1990-01-08 | Verfahren zur herstellung von fluoxetinhydrochlorid. |
DE69010017T DE69010017T2 (de) | 1989-01-10 | 1990-01-08 | Verfahren zur Herstellung von Fluoxetinhydrochlorid. |
ES90100314T ES2057187T3 (es) | 1989-01-10 | 1990-01-08 | Procedimiento para la preparacion de clorhidrato de fluoxetina. |
EP90100314A EP0380924B1 (en) | 1989-01-10 | 1990-01-08 | Process for the preparation of fluoxetine hydrochloride |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT8919049A IT1228209B (it) | 1989-01-10 | 1989-01-10 | Procedimento per la preparazione di fluoxetina cloridrato. |
Publications (2)
Publication Number | Publication Date |
---|---|
IT8919049A0 true IT8919049A0 (it) | 1989-01-10 |
IT1228209B IT1228209B (it) | 1991-06-05 |
Family
ID=11154121
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT8919049A IT1228209B (it) | 1989-01-10 | 1989-01-10 | Procedimento per la preparazione di fluoxetina cloridrato. |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP0380924B1 (it) |
AT (1) | ATE107623T1 (it) |
DE (1) | DE69010017T2 (it) |
ES (1) | ES2057187T3 (it) |
IT (1) | IT1228209B (it) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL99316A (en) | 1991-08-27 | 1995-03-15 | Teva Pharma | Production of fluoxetine and new intermediates |
US5618968A (en) * | 1993-02-05 | 1997-04-08 | Pliva Farmaceutska Kemijska, Prehrambena I Kozmeticka Industrija, Dionicko Drustvo | N-substituted derivatives of N-methyl-3-(p-trifluoromethylphenoxy)-3-phenylpropylamine and the procedure for their preparation |
ES2101650B1 (es) * | 1995-06-29 | 1998-01-16 | Lilly Sa | Procedimiento de preparacion de n-metil-3-fenil-3-(p-trifluorometilfenoxi) propilamina. |
ES2101654B1 (es) * | 1995-07-24 | 1998-01-16 | Lilly Sa | Procedimiento de preparacion de n-metil-3-fenil-3-(p-trifluorometilfe noxi) propilamina. |
ES2101655B1 (es) * | 1995-07-28 | 1998-01-16 | Lilly Sa | Procedimiento de preparacion de n-metil-3-fenil-3-(p-trifluorometilfe noxi) propilamina. |
ES2103680B1 (es) * | 1995-08-03 | 1998-04-01 | Lilly Sa | Procedimiento de preparacion de n-metil-3-fenil-3- (p-trifluorometilfenoxi)propilamina. |
ES2103681B1 (es) * | 1995-09-19 | 1998-04-01 | Lilly Sa | Procedimiento de preparacion de n-metil-3-fenil - (p-trifluorometilfenoxi) propilamina. |
US5936124A (en) * | 1998-06-22 | 1999-08-10 | Sepacor Inc. | Fluoxetine process from benzoylpropionic acid |
US6025517A (en) * | 1998-08-03 | 2000-02-15 | Sepracor Inc. | Fluoxetine process from benzoylacetonitrile |
US6846957B2 (en) | 2002-11-22 | 2005-01-25 | Board Of Regents, The University Of Texas System | Synthesis of 3-aminomethyl-1-propanol, a fluoxetine precursor |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4314081A (en) * | 1974-01-10 | 1982-02-02 | Eli Lilly And Company | Arloxyphenylpropylamines |
GB2060618A (en) * | 1979-09-14 | 1981-05-07 | Wyeth John & Brother Ltd | 3-Aryl-3-Aryloxypropylamines |
-
1989
- 1989-01-10 IT IT8919049A patent/IT1228209B/it active
-
1990
- 1990-01-08 AT AT90100314T patent/ATE107623T1/de not_active IP Right Cessation
- 1990-01-08 EP EP90100314A patent/EP0380924B1/en not_active Expired - Lifetime
- 1990-01-08 DE DE69010017T patent/DE69010017T2/de not_active Expired - Fee Related
- 1990-01-08 ES ES90100314T patent/ES2057187T3/es not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
IT1228209B (it) | 1991-06-05 |
EP0380924A1 (en) | 1990-08-08 |
ES2057187T3 (es) | 1994-10-16 |
DE69010017T2 (de) | 1994-10-06 |
ATE107623T1 (de) | 1994-07-15 |
DE69010017D1 (de) | 1994-07-28 |
EP0380924B1 (en) | 1994-06-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19940203 |