IT1211681B - PEPTIDES AND PEPTIDAL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS - Google Patents
PEPTIDES AND PEPTIDAL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONSInfo
- Publication number
- IT1211681B IT1211681B IT8748235A IT4823587A IT1211681B IT 1211681 B IT1211681 B IT 1211681B IT 8748235 A IT8748235 A IT 8748235A IT 4823587 A IT4823587 A IT 4823587A IT 1211681 B IT1211681 B IT 1211681B
- Authority
- IT
- Italy
- Prior art keywords
- peptidal
- medications
- peptides
- derivatives
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/0227—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the (partial) peptide sequence -Phe-His-NH-(X)2-C(=0)-, e.g. Renin-inhibitors with n = 2 - 6; for n > 6 see C07K5/06 - C07K5/10
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB868619182A GB8619182D0 (en) | 1986-08-06 | 1986-08-06 | Peptides & derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
IT8748235A0 IT8748235A0 (en) | 1987-07-28 |
IT1211681B true IT1211681B (en) | 1989-11-03 |
Family
ID=10602311
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT8748235A IT1211681B (en) | 1986-08-06 | 1987-07-28 | PEPTIDES AND PEPTIDAL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS |
Country Status (7)
Country | Link |
---|---|
JP (1) | JPS6348295A (en) |
BE (1) | BE1001618A4 (en) |
CH (1) | CH673655A5 (en) |
DE (1) | DE3725137A1 (en) |
FR (1) | FR2602511A1 (en) |
GB (2) | GB8619182D0 (en) |
IT (1) | IT1211681B (en) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5071837A (en) * | 1990-11-28 | 1991-12-10 | Warner-Lambert Company | Novel renin inhibiting peptides |
NZ241099A (en) * | 1991-01-02 | 1994-08-26 | Merrell Dow Pharma | Difluorostatone analogues and derivatives and pharmaceutical compositions |
WO1995001958A1 (en) * | 1993-07-08 | 1995-01-19 | Merrell Pharmaceuticals Inc. | Difluoro statone analogs |
KR100308839B1 (en) * | 1993-09-09 | 2002-10-04 | 메렐 파마슈티칼스 인크. | Difluoro startone antiviral analogs |
US6114380A (en) * | 1995-12-18 | 2000-09-05 | Merrell Pharmaceuticals Inc. | Difluoro statone analogs |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FI88400C (en) * | 1984-08-06 | 1993-05-10 | Upjohn Co | FRAMEWORK FOR THE FRAME STATION INHIBITION OF PEPTIDER |
IL77748A (en) * | 1985-02-04 | 1991-11-21 | Merrell Dow Pharma | Amino acid and peptide derivatives as peptidase inhibitors |
CH672792A5 (en) * | 1985-02-19 | 1989-12-29 | Sandoz Ag | |
EP0218688B1 (en) * | 1985-04-19 | 1990-09-12 | The Upjohn Company | Dihalo-statine substituted renin inhibitors |
HU200473B (en) * | 1985-11-01 | 1990-06-28 | Pfizer | Process for producing polypeptides containing difluorocyclostatine and pharmaceutical compositions comprising same |
ES2056930T3 (en) * | 1987-07-01 | 1994-10-16 | Pfizer | FLUORINE CONTAINING RENINE INHIBITORS. |
JPH10183253A (en) * | 1996-12-24 | 1998-07-14 | Nisshin Steel Co Ltd | Production of cold rolled steel sheet or hot dip plated steel sheet excellent in surface property and workability |
-
1986
- 1986-08-06 GB GB868619182A patent/GB8619182D0/en active Pending
-
1987
- 1987-07-27 BE BE8700830A patent/BE1001618A4/en not_active IP Right Cessation
- 1987-07-27 FR FR8710662A patent/FR2602511A1/en not_active Withdrawn
- 1987-07-28 IT IT8748235A patent/IT1211681B/en active
- 1987-07-29 DE DE19873725137 patent/DE3725137A1/en not_active Withdrawn
- 1987-07-31 CH CH2936/87A patent/CH673655A5/de not_active IP Right Cessation
- 1987-08-03 GB GB8718325A patent/GB2196958B/en not_active Expired - Lifetime
- 1987-08-05 JP JP62196151A patent/JPS6348295A/en active Pending
Also Published As
Publication number | Publication date |
---|---|
GB2196958A (en) | 1988-05-11 |
GB8619182D0 (en) | 1986-09-17 |
FR2602511A1 (en) | 1988-02-12 |
IT8748235A0 (en) | 1987-07-28 |
GB8718325D0 (en) | 1987-09-09 |
BE1001618A4 (en) | 1989-12-19 |
JPS6348295A (en) | 1988-02-29 |
DE3725137A1 (en) | 1988-02-11 |
CH673655A5 (en) | 1990-03-30 |
GB2196958B (en) | 1990-07-04 |
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