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IT1211681B - PEPTIDES AND PEPTIDAL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS - Google Patents

PEPTIDES AND PEPTIDAL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS

Info

Publication number
IT1211681B
IT1211681B IT8748235A IT4823587A IT1211681B IT 1211681 B IT1211681 B IT 1211681B IT 8748235 A IT8748235 A IT 8748235A IT 4823587 A IT4823587 A IT 4823587A IT 1211681 B IT1211681 B IT 1211681B
Authority
IT
Italy
Prior art keywords
peptidal
medications
peptides
derivatives
preparation
Prior art date
Application number
IT8748235A
Other languages
Italian (it)
Other versions
IT8748235A0 (en
Inventor
Pfenninger Emil
Weidmann Beat
Stoll Andre
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of IT8748235A0 publication Critical patent/IT8748235A0/en
Application granted granted Critical
Publication of IT1211681B publication Critical patent/IT1211681B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0227Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the (partial) peptide sequence -Phe-His-NH-(X)2-C(=0)-, e.g. Renin-inhibitors with n = 2 - 6; for n > 6 see C07K5/06 - C07K5/10
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
IT8748235A 1986-08-06 1987-07-28 PEPTIDES AND PEPTIDAL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS IT1211681B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868619182A GB8619182D0 (en) 1986-08-06 1986-08-06 Peptides & derivatives

Publications (2)

Publication Number Publication Date
IT8748235A0 IT8748235A0 (en) 1987-07-28
IT1211681B true IT1211681B (en) 1989-11-03

Family

ID=10602311

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8748235A IT1211681B (en) 1986-08-06 1987-07-28 PEPTIDES AND PEPTIDAL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS

Country Status (7)

Country Link
JP (1) JPS6348295A (en)
BE (1) BE1001618A4 (en)
CH (1) CH673655A5 (en)
DE (1) DE3725137A1 (en)
FR (1) FR2602511A1 (en)
GB (2) GB8619182D0 (en)
IT (1) IT1211681B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5071837A (en) * 1990-11-28 1991-12-10 Warner-Lambert Company Novel renin inhibiting peptides
NZ241099A (en) * 1991-01-02 1994-08-26 Merrell Dow Pharma Difluorostatone analogues and derivatives and pharmaceutical compositions
WO1995001958A1 (en) * 1993-07-08 1995-01-19 Merrell Pharmaceuticals Inc. Difluoro statone analogs
KR100308839B1 (en) * 1993-09-09 2002-10-04 메렐 파마슈티칼스 인크. Difluoro startone antiviral analogs
US6114380A (en) * 1995-12-18 2000-09-05 Merrell Pharmaceuticals Inc. Difluoro statone analogs

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI88400C (en) * 1984-08-06 1993-05-10 Upjohn Co FRAMEWORK FOR THE FRAME STATION INHIBITION OF PEPTIDER
IL77748A (en) * 1985-02-04 1991-11-21 Merrell Dow Pharma Amino acid and peptide derivatives as peptidase inhibitors
CH672792A5 (en) * 1985-02-19 1989-12-29 Sandoz Ag
EP0218688B1 (en) * 1985-04-19 1990-09-12 The Upjohn Company Dihalo-statine substituted renin inhibitors
HU200473B (en) * 1985-11-01 1990-06-28 Pfizer Process for producing polypeptides containing difluorocyclostatine and pharmaceutical compositions comprising same
ES2056930T3 (en) * 1987-07-01 1994-10-16 Pfizer FLUORINE CONTAINING RENINE INHIBITORS.
JPH10183253A (en) * 1996-12-24 1998-07-14 Nisshin Steel Co Ltd Production of cold rolled steel sheet or hot dip plated steel sheet excellent in surface property and workability

Also Published As

Publication number Publication date
GB2196958A (en) 1988-05-11
GB8619182D0 (en) 1986-09-17
FR2602511A1 (en) 1988-02-12
IT8748235A0 (en) 1987-07-28
GB8718325D0 (en) 1987-09-09
BE1001618A4 (en) 1989-12-19
JPS6348295A (en) 1988-02-29
DE3725137A1 (en) 1988-02-11
CH673655A5 (en) 1990-03-30
GB2196958B (en) 1990-07-04

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