[go: up one dir, main page]

IT1172381B - Esteri di derivati 3-(3-sostituito-ammino-2-idrossi-propossi)-4-sostituito-1,2,5-tiadiazolici utili come agenti bloccanti beta-adrenergici e per il trattamento del glaucoma - Google Patents

Esteri di derivati 3-(3-sostituito-ammino-2-idrossi-propossi)-4-sostituito-1,2,5-tiadiazolici utili come agenti bloccanti beta-adrenergici e per il trattamento del glaucoma

Info

Publication number
IT1172381B
IT1172381B IT49538/83A IT4953883A IT1172381B IT 1172381 B IT1172381 B IT 1172381B IT 49538/83 A IT49538/83 A IT 49538/83A IT 4953883 A IT4953883 A IT 4953883A IT 1172381 B IT1172381 B IT 1172381B
Authority
IT
Italy
Prior art keywords
substituted
thiadiazolics
glaucoma
beta
hydroxy
Prior art date
Application number
IT49538/83A
Other languages
English (en)
Other versions
IT8349538A0 (it
Inventor
William L Matier
Paul W Erhardt
Ghanshyam Patil
Original Assignee
American Hospital Supply Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Hospital Supply Corp filed Critical American Hospital Supply Corp
Publication of IT8349538A0 publication Critical patent/IT8349538A0/it
Application granted granted Critical
Publication of IT1172381B publication Critical patent/IT1172381B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IT49538/83A 1982-12-22 1983-12-19 Esteri di derivati 3-(3-sostituito-ammino-2-idrossi-propossi)-4-sostituito-1,2,5-tiadiazolici utili come agenti bloccanti beta-adrenergici e per il trattamento del glaucoma IT1172381B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/452,280 US4508725A (en) 1982-12-22 1982-12-22 Esters of 3-(3-substituted-amino-2-hydroxypropoxy)-4-substituted-1,2,5-thiadiazole derivatives

Publications (2)

Publication Number Publication Date
IT8349538A0 IT8349538A0 (it) 1983-12-19
IT1172381B true IT1172381B (it) 1987-06-18

Family

ID=23795857

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49538/83A IT1172381B (it) 1982-12-22 1983-12-19 Esteri di derivati 3-(3-sostituito-ammino-2-idrossi-propossi)-4-sostituito-1,2,5-tiadiazolici utili come agenti bloccanti beta-adrenergici e per il trattamento del glaucoma

Country Status (14)

Country Link
US (1) US4508725A (it)
EP (1) EP0131006B1 (it)
JP (1) JPS60500288A (it)
AU (1) AU567908B2 (it)
CA (1) CA1230879A (it)
DE (1) DE3382578T2 (it)
ES (1) ES8504159A1 (it)
IE (1) IE59617B1 (it)
IT (1) IT1172381B (it)
MX (1) MX156097A (it)
NO (1) NO164095C (it)
NZ (1) NZ206385A (it)
WO (1) WO1984002525A1 (it)
ZA (1) ZA838829B (it)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623652A (en) 1981-11-12 1986-11-18 American Hospital Supply Corporation Esters of thiadiazole oxypropanolaine derivatives and pharmaceutical uses
US5320839A (en) * 1991-10-11 1994-06-14 Alcon Laboratories, Inc. Topical ophthalmic compositions comprising 4-(3-substituted amino-2-hydroxypropoxy)-1,2,5-thiadiazoles and methods for their use
JPH06511242A (ja) * 1991-10-11 1994-12-15 アルコン　ラボラトリーズ　インコーポレイテッド ４−（３−置換アミノ−２−ヒドロキシプロポキシ）−１，２，５−チアジアゾール類を含む局所的目薬組成物およびそれ等の使用方法
US5821370A (en) * 1994-10-24 1998-10-13 Eli Lilly And Company Heterocyclic compounds and their preparation and use
US6750238B1 (en) * 2000-05-12 2004-06-15 The University Of Toledo Aralkyl ester soft drugs
US7049326B2 (en) * 2000-05-12 2006-05-23 The University Of Toledo Method and compositions for temporarily incapacitating subjects
US6756047B2 (en) * 2000-05-12 2004-06-29 The University Of Toledo Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs
US20110092507A1 (en) * 2009-10-20 2011-04-21 Chin-Tsai Fan Process for preparing R-(+)-3-morpholino-4-(3- tert-butylamino-2-hydroxypropoxy)-1,2,5-thiadiazole

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4051144A (en) * 1968-05-22 1977-09-27 Charles E. Frosst & Co. Sinister-3,5-disubstituted oxozolidines their preparation and use
US3655663A (en) * 1969-04-21 1972-04-11 Burton K Wasson 4-(3-secondary amino-2-hydroxy-proxy) 1 2 5-thiadiazoles
FR2132570B1 (it) * 1971-04-09 1974-08-02 Lipha
US3729477A (en) * 1971-09-09 1973-04-24 Frosst & Co Charles E Certain 4-(3-amino-2-hydroxypropoxy)-1,2,5-thiadiazole-3-carboxamides
US4083992A (en) * 1972-12-15 1978-04-11 Imperial Chemical Industries Limited Alkanolamine derivatives
US3891639A (en) * 1973-04-19 1975-06-24 Merck Sharp & Dohme 4-{8 3-Amino-2-acyloxypropoxy{9 -1,2,5-thiadiazole compounds
US4011217A (en) * 1973-04-19 1977-03-08 Merck Sharp & Dohme (I.A.) Corporation 4-(3-amino-2-acyloxypropoxy)-1,2,5-thiadiazole compounds
DE2609486A1 (de) * 1975-08-07 1977-05-12 Hoffmann La Roche Imidazo eckige klammer auf 1,5-a eckige klammer zu eckige klammer auf 1,4 eckige klammer zu diazepin-verbindungen und verfahren zu ihrer herstellung
US4127674A (en) * 1977-03-21 1978-11-28 Allergan Pharmaceuticals, Inc. Method of treatment for glaucoma
US4387103A (en) * 1980-11-28 1983-06-07 American Hospital Supply Corporation Method for treatment or prophylaxis of cardiac disorders
ZA827646B (en) * 1981-11-12 1983-08-31 American Hospital Supply Corp Esters of aryloxypropanolamine derivatives

Also Published As

Publication number Publication date
WO1984002525A1 (en) 1984-07-05
ES528225A0 (es) 1985-04-16
US4508725A (en) 1985-04-02
AU2334184A (en) 1984-07-17
ZA838829B (en) 1985-03-27
NO843352L (no) 1984-08-22
IE832730L (en) 1984-06-22
EP0131006B1 (en) 1992-06-10
ES8504159A1 (es) 1985-04-16
NO164095C (no) 1990-09-05
IT8349538A0 (it) 1983-12-19
IE59617B1 (en) 1994-03-09
DE3382578T2 (de) 1993-03-25
JPS60500288A (ja) 1985-03-07
NZ206385A (en) 1986-08-08
AU567908B2 (en) 1987-12-10
NO164095B (no) 1990-05-21
EP0131006A4 (en) 1985-06-06
EP0131006A1 (en) 1985-01-16
MX156097A (es) 1988-07-07
DE3382578D1 (de) 1992-07-16
CA1230879A (en) 1987-12-29

Similar Documents

Publication Publication Date Title
IT8249249A0 (it) Procedimento per la fabbricazione di pannolini elasticizzati
ES525743A0 (es) Procedimiento para la fabricacion de 4'-demetil-epipodofilotoxin-b-d-etiliden-glucosido y derivado acilico del mismo
IT8419543A0 (it) Derivati di 3-cefem-4-carbossilati e loro sali, esteri e solvati aventi proprieta' antibatteriche.
IT1166551B (it) Procedimento per la fabbricazione di impiantati nonche' impiantati realizzati con detto procedimento
IT8267795A0 (it) Composizione per trattamento del glaucoma
KR900701323A (ko) 신규한 녹내장 치료용 안과 제제
IT1172381B (it) Esteri di derivati 3-(3-sostituito-ammino-2-idrossi-propossi)-4-sostituito-1,2,5-tiadiazolici utili come agenti bloccanti beta-adrenergici e per il trattamento del glaucoma
IT1149483B (it) Macchina perfezionata per la formatura di croissants e simili
IT8005106A0 (it) Composti per il trattamento del glaucoma.
ITMI941494A0 (it) Derivati del fenilcarbammato atti all'impiego come anticolinesterasici
IT8267796A0 (it) Composizione per trattamento del glaucoma
IT8267794A0 (it) Composizione per trattamento del glaucoma
IT8220803A0 (it) Procedimento per la preparazione del 2,3-diidro-2,2-dimetilbenzofuran-7olo.
IT7826768A0 (it) Procedimento per l'eliminazione di nitrosammine delle dinitro-aniline.
IT8319024A0 (it) Composizione medicinale per il trattamento di certe neurovirosi.
IT1153293B (it) Derivati del 4-idrossi-2-metil-2h-1, 2-benzotiazina-3-carbossamide 1, 1-biossido e procedimento per la loro preparazione
DE69301522D1 (de) Apparat für die Herstellung von Halbleiter-Einrichtungen
IT1179508B (it) Procedimento per la preparazione di derivati del 2,3-diidrobenzopiranone
IT1158004B (it) Apparecchio e procedimento per l'impilamento di articoli di forma appiattita particolarmente pannolini ed assorbenti
IT8922875A0 (it) Procedimento per la preparazione del clotrimazolo
IT1163943B (it) Derivati 15-cicloalifatici di 13,14-dideidro carboprostacicline e procedimento per la loro preparazione
IT8049235A0 (it) Procedimento per la produzione di 3-(4)-formiltriciclo(5,2,1,0,2,6)-de cene-8
IT1089343B (it) Procedimento per la preparazione di esteri 0,0-dialchil-s-(n-metil-carbossiami dometil)-tiol-fosforici
IT8047950A0 (it) Composizioni farmaceutiche impiegabili per il trattamento dell'ipertensione
IT1156990B (it) Procedimento per la preparazione del cloridrato di p clorofenossiacetil piperonilpierazina

Legal Events

Date Code Title Description
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19941027