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IN2003KO00001A - - Google Patents

Info

Publication number
IN2003KO00001A
IN2003KO00001A IN1KO2003A IN2003KO00001A IN 2003KO00001 A IN2003KO00001 A IN 2003KO00001A IN 1KO2003 A IN1KO2003 A IN 1KO2003A IN 2003KO00001 A IN2003KO00001 A IN 2003KO00001A
Authority
IN
India
Application number
Inventor
Mark R Schmitt
Donald R Kirsch
Jane E Harris
Carl F Beyer
Klaus-Juergen Pees
Paul Carter
Waldemar Pfrengle
Guido Albert
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Publication of IN2003KO00001A publication Critical patent/IN2003KO00001A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IN1KO2003 2000-06-30 2003-01-01 IN2003KO00001A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US21558500P 2000-06-30 2000-06-30

Publications (1)

Publication Number Publication Date
IN2003KO00001A true IN2003KO00001A (en) 2005-12-02

Family

ID=22803554

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1KO2003 IN2003KO00001A (en) 2000-06-30 2003-01-01

Country Status (24)

Country Link
US (1) US7329663B2 (en)
EP (1) EP1307200A2 (en)
JP (1) JP2004502691A (en)
KR (1) KR20030013475A (en)
CN (1) CN1592624A (en)
AR (1) AR034553A1 (en)
AU (2) AU7306201A (en)
BG (1) BG107277A (en)
BR (1) BR0112038A (en)
CA (1) CA2413802A1 (en)
CZ (1) CZ20024150A3 (en)
EA (1) EA006483B1 (en)
GE (1) GEP20053688B (en)
HK (1) HK1052646A1 (en)
HU (1) HUP0300798A3 (en)
IL (1) IL152869A0 (en)
IN (1) IN2003KO00001A (en)
MX (1) MXPA02011913A (en)
NO (1) NO20026195L (en)
NZ (1) NZ523807A (en)
PL (1) PL360027A1 (en)
SK (1) SK18412002A3 (en)
WO (1) WO2002002563A2 (en)
ZA (1) ZA200300793B (en)

Families Citing this family (49)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6255309B1 (en) 1999-03-19 2001-07-03 American Cyanomid Co. Fungicidal trifluoromethylalkylamino-triazolopyrimidines
JP2004513170A (en) * 2000-11-13 2004-04-30 ビーエーエスエフ　アクチェンゲゼルシャフト 7- (R) -aminotriazolopyrimidines, their production and their use for controlling phytopathogenic fungi
EP1381610B1 (en) * 2001-04-11 2004-08-25 Basf Aktiengesellschaft 6-(2-chloro-6-fluoro-phenyl)-triazolopyrimidines
NZ528745A (en) * 2001-04-11 2005-03-24 Basf Ag 5-halogen-6-phenyl-7-fluoralkylamino-triazolopyrimidines as fungicides and their preparation process
DE10121101A1 (en) * 2001-04-27 2002-10-31 Bayer Ag triazolopyrimidines
DE10121162A1 (en) * 2001-04-30 2002-10-31 Bayer Ag triazolopyrimidines
DE10124208A1 (en) 2001-05-18 2002-11-21 Bayer Ag Use of triazolopyrimidine derivatives for protecting technical materials, particularly wood, paints and plastics, against microbes, particularly fungi
CN1271071C (en) * 2001-07-18 2006-08-23 巴斯福股份公司 Substituted (6-2-tolyl)-triazolopyrimidines as fungicides
ATE384064T1 (en) * 2002-03-21 2008-02-15 Basf Ag FUNGICIDAL TRIAZOLOPYRIMIDINES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE FOR CONTROLLING HARMFUL FUNGI AND AGENTS CONTAINING SAME
JPWO2004011467A1 (en) * 2002-07-29 2005-12-15 北興化学工業株式会社 Triazolopyrimidine derivatives and agricultural and horticultural fungicides
UA80304C2 (en) * 2002-11-07 2007-09-10 Basf Ag Substituted 6-(2-halogenphenyl)triazolopyrimidines
EA200501388A1 (en) * 2003-03-31 2006-02-24 Басф Акциенгезельшафт 7-ALKYNYLAMINOTRIAZOLOPYRIMIDINES, METHOD FOR THEIR RECEPTION AND THEIR APPLICATION FOR THE FIGHT AGAINST PHYTOPATHOGENIC MUSHRIA, AND ALSO CONTAINING THEIR MEANS
DE10325133A1 (en) * 2003-06-04 2004-12-23 Bayer Cropscience Ag triazolopyrimidines
WO2004108136A1 (en) * 2003-06-04 2004-12-16 Vernalis (Cambridge) Limited Triazolo `1 , 5-a!pyrimidines and their use in medicine
DE10328173A1 (en) * 2003-06-24 2005-01-13 Bayer Cropscience Ag triazolopyrimidines
DE10328171A1 (en) * 2003-06-24 2005-01-13 Bayer Cropscience Ag triazolopyrimidines
DE10328481A1 (en) * 2003-06-25 2005-01-13 Bayer Ag triazolopyrimidines
AU2004276240A1 (en) * 2003-09-24 2005-04-07 Wyeth Holdings Corporation 6-[(substituted)phenyl]triazolopyrimidines as anticancer agents
US7419982B2 (en) 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
DE602004014525D1 (en) 2003-09-24 2008-07-31 Wyeth Corp 6-ARYL-7-HALO-IMIDAZOÄ1,2-AÜPYRIMIDINE AS A MEDIUM AGAINST CANCER
JPWO2005037837A1 (en) * 2003-10-17 2006-12-28 日本化薬株式会社 Substituted 2-amino- [1,2,4] triazolo [1,5-a] pyrimidine derivatives and uses thereof
JP4606015B2 (en) * 2003-11-25 2011-01-05 日本化薬株式会社 Novel pharmaceutical uses of [1,2,4] triazolo [1,5-a] pyrimidine derivatives
MY179926A (en) 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
US20070135453A1 (en) * 2003-12-17 2007-06-14 Basf Aktiengesellschaft 6-(2,4,6-Trihalophenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
JP2007514678A (en) * 2003-12-17 2007-06-07 ビーエーエスエフ　アクチェンゲゼルシャフト 6- (2,3,6-trifluorophenyl) triazolopyrimidine, its preparation and its use for controlling harmful fungi, and a composition comprising said compound
CN1938313A (en) * 2004-03-30 2007-03-28 巴斯福股份公司 6-(2-fluorophenyl)-triazolopyrimidines, method for producing them, their use for controlling parasitic fungi and agents containing the same
WO2005113555A1 (en) * 2004-05-17 2005-12-01 Basf Aktiengesellschaft Triazolopyrimidine compounds and their use for controlling pathogenic fungi
CN1964629A (en) * 2004-06-09 2007-05-16 巴斯福股份公司 Triazolopyrimidine compounds and use thereof for controlling harmful fungi
MXPA06013943A (en) * 2004-06-25 2007-03-15 Basf Ag Triazolopyrimidine compounds and their use for controlling pathogenic fungi.
US20070155738A1 (en) * 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
CA2608890C (en) * 2005-05-20 2011-08-02 Alantos-Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
WO2007011759A2 (en) * 2005-07-15 2007-01-25 Kalypsys, Inc. Inhibitors of mitotic kinesin
JP2009519954A (en) * 2005-12-16 2009-05-21 ワイス Dimers and adducts of 6-[(substituted) phenyl] triazolopyrimidines useful as anticancer agents
AR059649A1 (en) * 2006-02-28 2008-04-16 Basf Ag 6- 7-AMINO PHENYL - AMINO (1,2,4) -TRIAZOLO (1,5-A) PYRIMIDINS AND ITS USE FOR THE FIGHT OF DANGINE FUNGES
WO2007116011A2 (en) * 2006-04-10 2007-10-18 Basf Se Substituted triazolopyrimidines, method for the production thereof, use thereof for controlling harmful fungi, and substances containing the same
JP5231829B2 (en) * 2007-02-15 2013-07-10 石原産業株式会社 Pyridyl-triazolopyrimidine derivatives or salts thereof, pest control agents containing them, and methods for producing them
NZ583267A (en) 2007-08-14 2012-03-30 Bayer Schering Pharma Ag Fused bicyclic pyrimidines
CN103889428A (en) 2010-10-04 2014-06-25 肝炎与病毒研究所 Novel inhibitors of secretion of hepatitis b virus antigens
CN104395298A (en) * 2012-06-22 2015-03-04 住友化学株式会社 Fused heterocyclic compound
CN103360398B (en) * 2013-07-22 2015-03-25 山东大学 Triazolopyrimidine HIV-1 retrovirus inhibitor and its preparation method and application thereof
GB201504565D0 (en) 2015-03-18 2015-05-06 Takeda Pharmaceutical Novel compounds
KR101995533B1 (en) * 2017-03-21 2019-07-02 한국화학연구원 Novel [1,2,4]triazolo[4,3-a]quinoxaline amino phenyl derivatives or pharmaceutically acceptable salts thereof, preparation method therof and pharmaceutical composition for use in preventing or treating bromodomain extra-terminal(BET) protein activity related diseases containing the same as an active ingredient
US11390626B2 (en) 2019-01-29 2022-07-19 Tosk, Inc. Pyrazolopyrimidine modulators of RAS GTPase
CN115397826A (en) * 2020-04-14 2022-11-25 宾夕法尼亚大学理事会 Substituted {1,2,4,}triazolo{1,5-A}pyrimidines and their application to stabilize microtubules
EP4143194A1 (en) 2020-05-01 2023-03-08 Gilead Sciences, Inc. Cd73 inhibiting 2,4-dioxopyrimidine compounds
US20230279006A1 (en) * 2020-07-08 2023-09-07 Klotho Therapeutics, Inc. Novel compounds and methods for increasing klotho gene expression
US12180220B2 (en) 2020-10-14 2024-12-31 Tosk, Inc. Heteroaryl modulators of RAS GTPase
WO2023077030A1 (en) 2021-10-29 2023-05-04 Gilead Sciences, Inc. Cd73 compounds
WO2023143194A1 (en) * 2022-01-25 2023-08-03 瑞石生物医药有限公司 Ccr4 small molecule antagonist and use thereof

Family Cites Families (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD55956A (en) *
DE55956C (en) CH. GROOMBRIDGE und W. A. SOUTH in London, 40 New Bond Street Brake crank for horse-drawn tram and other wagons
DE61269C (en) 1891-04-01 1892-03-23 J. NEWBURG in Berlin O., Am Schlesischen Bahnhof Nr. 5 Washing machine
JPS5827773B2 (en) * 1980-02-08 1983-06-11 持田製薬株式会社 Cancer metastasis inhibitor
US4444774A (en) * 1982-07-29 1984-04-24 American Cyanamid Company 7-Heteroaryl[1,2,4]triazolo[1,5-a]pyrimidines
GB8719368D0 (en) * 1987-08-15 1987-09-23 Wellcome Found Heterocyclic compounds
JPH02212488A (en) * 1989-02-13 1990-08-23 Shinichiro Shimizu Triazolepyridmine derivative
US5593996A (en) * 1991-12-30 1997-01-14 American Cyanamid Company Triazolopyrimidine derivatives
US5387747A (en) * 1992-02-24 1995-02-07 Laboratoires Upsa Triazolopyrimidine derivatives which are angiotensin II receptor antagonists, their methods of preparation and pharmaceutical compositions in which they are present
IL108747A (en) * 1993-03-04 1999-03-12 Shell Int Research Fungicidal compositions containing 6-substituted-5,7-dihalo-1,2,4-triazolo Ú1,5-a¾pyrimidine derivatives certain new such derivatives and their preparation
GB9321162D0 (en) * 1993-10-13 1993-12-01 Boots Co Plc Therapeutic agents
US5869486A (en) * 1995-02-24 1999-02-09 Ono Pharmaceutical Co., Ltd. Fused pyrimidines and pyriazines as pharmaceutical compounds
US6255309B1 (en) * 1999-03-19 2001-07-03 American Cyanomid Co. Fungicidal trifluoromethylalkylamino-triazolopyrimidines
US5948783A (en) * 1997-04-14 1999-09-07 American Cyanamid Company Fungicidal trifluoromethylalkylamino-triazolopyrimidines
US6117876A (en) * 1997-04-14 2000-09-12 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
US5994360A (en) * 1997-07-14 1999-11-30 American Cyanamid Company Fungicidal 5-alkyl-triazolopyrimidines
US6020338A (en) * 1998-02-11 2000-02-01 American Cyanamid Company Fungicidal 7-alkyl-triazolopyrimidines
US6380202B1 (en) * 1998-09-25 2002-04-30 Basf Aktiengesellschaft Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines
FR2784380B1 (en) * 1998-09-25 2002-09-06 American Cyanamid Co TRIAZOLOPYRIMIDINES 7-OXY- AND 7-THIO-SUBSTITUTED FUNGICIDES
US6165940A (en) * 1998-09-25 2000-12-26 American Cyanamid Co. Non-aqueous suspension concentrate
MY125533A (en) * 1999-12-06 2006-08-30 Bristol Myers Squibb Co Heterocyclic dihydropyrimidine compounds
JP2001322933A (en) * 2000-05-15 2001-11-20 Ucb Sa CD40 signal blocker
DE10121102A1 (en) * 2001-04-27 2002-11-07 Bayer Ag triazolopyrimidines
DE10121101A1 (en) * 2001-04-27 2002-10-31 Bayer Ag triazolopyrimidines
DE10121162A1 (en) * 2001-04-30 2002-10-31 Bayer Ag triazolopyrimidines
US7037902B2 (en) * 2002-07-03 2006-05-02 Receptron, Inc. Affinity small molecules for the EPO receptor
US7419982B2 (en) * 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
AU2004276240A1 (en) * 2003-09-24 2005-04-07 Wyeth Holdings Corporation 6-[(substituted)phenyl]triazolopyrimidines as anticancer agents

Also Published As

Publication number Publication date
BG107277A (en) 2004-01-30
ZA200300793B (en) 2004-07-20
IL152869A0 (en) 2003-06-24
PL360027A1 (en) 2004-09-06
AU7306201A (en) 2002-01-14
US7329663B2 (en) 2008-02-12
WO2002002563A2 (en) 2002-01-10
HK1052646A1 (en) 2003-09-26
AU2001273062B2 (en) 2005-11-24
US20020068744A1 (en) 2002-06-06
NO20026195D0 (en) 2002-12-23
EP1307200A2 (en) 2003-05-07
SK18412002A3 (en) 2003-06-03
NO20026195L (en) 2003-02-27
MXPA02011913A (en) 2003-04-22
CZ20024150A3 (en) 2003-09-17
EA200300091A1 (en) 2003-08-28
BR0112038A (en) 2003-04-01
KR20030013475A (en) 2003-02-14
HUP0300798A3 (en) 2006-02-28
NZ523807A (en) 2004-09-24
GEP20053688B (en) 2005-12-12
WO2002002563A3 (en) 2003-01-03
CA2413802A1 (en) 2002-01-10
CN1592624A (en) 2005-03-09
AR034553A1 (en) 2004-03-03
JP2004502691A (en) 2004-01-29
HUP0300798A2 (en) 2003-07-28
EA006483B1 (en) 2005-12-29

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