[go: up one dir, main page]

IL70540A0 - Microbicidal agents containing quinolonecarboxylic acids and method of using them - Google Patents

Microbicidal agents containing quinolonecarboxylic acids and method of using them

Info

Publication number
IL70540A0
IL70540A0 IL70540A IL7054083A IL70540A0 IL 70540 A0 IL70540 A0 IL 70540A0 IL 70540 A IL70540 A IL 70540A IL 7054083 A IL7054083 A IL 7054083A IL 70540 A0 IL70540 A0 IL 70540A0
Authority
IL
Israel
Prior art keywords
agents containing
microbicidal agents
quinolonecarboxylic acids
chlorine
fluorine
Prior art date
Application number
IL70540A
Other versions
IL70540A (en
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of IL70540A0 publication Critical patent/IL70540A0/en
Publication of IL70540A publication Critical patent/IL70540A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Processing Of Solid Wastes (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Quinoline Compounds (AREA)
  • Cosmetics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Combating microorganisms, particularly in agriculture, with a 1-cyclopropyl-1,4-dihydro-4-oxo-quinolinecarboxylic acid of the formula <IMAGE> in which R1 is hydrogen, fluorine, chlorine, bromine or nitro, R2 is hydrogen, chlorine, fluorine or the group <IMAGE> particularly a 4-piperazinyl radical, or an acid addition, alkali metal, alkaline earth metal or heavy metal salt thereof which is tolerated by plants, or a hydrate thereof. Some of the compounds are known.
IL70540A 1982-12-29 1983-12-26 Plant bactericidal and fungicidal compositions containing 1-cycloproply-quinolonecarboxylic acid and method for using them IL70540A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19823248507 DE3248507A1 (en) 1982-12-29 1982-12-29 MICROBICIDE AGENTS BASED ON CHINOLONIC CARBONIC ACID

Publications (2)

Publication Number Publication Date
IL70540A0 true IL70540A0 (en) 1984-03-30
IL70540A IL70540A (en) 1987-07-31

Family

ID=6182079

Family Applications (1)

Application Number Title Priority Date Filing Date
IL70540A IL70540A (en) 1982-12-29 1983-12-26 Plant bactericidal and fungicidal compositions containing 1-cycloproply-quinolonecarboxylic acid and method for using them

Country Status (13)

Country Link
US (1) US4563459A (en)
EP (1) EP0113091B1 (en)
JP (1) JPS59130802A (en)
AT (1) ATE21011T1 (en)
AU (1) AU563747B2 (en)
BR (1) BR8307166A (en)
CA (1) CA1232198A (en)
DE (2) DE3248507A1 (en)
DK (1) DK603883A (en)
GR (1) GR81542B (en)
HU (1) HU194482B (en)
IL (1) IL70540A (en)
ZA (1) ZA839647B (en)

Families Citing this family (48)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3420743A1 (en) * 1984-06-04 1985-12-05 Bayer Ag, 5090 Leverkusen 7-AMINO-1-CYCLOPROPYL-6,8-DIHALOGEN-1,4-DIHYDRO-4-OXO-3-CHINOLINE CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THEIR CONTAINING ANTIBACTERIAL AGENTS
US5468861A (en) * 1984-06-04 1995-11-21 Bayer Aktiengesellschaft 8-chloro-1-cyclopropyl-6,7-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid and alkyl esters thereof
DE3420798A1 (en) * 1984-06-04 1985-12-05 Bayer Ag, 5090 Leverkusen 7- (3-ARYL-L-PIPERAZINYL) - AND 7- (3-CYCLOHEXYL-L-PIPERAZINYL) -3-CHINOLONIC CARBONIC ACIDS
DE3426483A1 (en) * 1984-07-18 1986-01-30 Bayer Ag, 5090 Leverkusen METHOD FOR PRODUCING HALOGENATED CHINOLON CARBONIC ACIDS
DE3441788A1 (en) * 1984-11-15 1986-05-15 Bayer Ag, 5090 Leverkusen ALKYL-1-CYCLOPROPYL-1,4-DIHYDRO-4-OXO-3-CHINOLINE CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THE ANTIBACTERIAL AGENTS CONTAINING THEM
FR2574404B1 (en) * 1984-12-12 1987-04-24 Provesan Sa 1-SUBSTITUTED DERIVATIVES OF 6-FLUORO-7- (PYRROL-1-YL) -1,4-DIHYDRO-4-OXOQUINOLEIN-3-CARBOXYLIC ACID, THEIR PREPARATION AND THEIR APPLICATION AS MEDICAMENTS
DE3508816A1 (en) * 1985-01-10 1986-07-10 Bayer Ag, 5090 Leverkusen 6,7-DISUBSTITUTED 1-CYCLOPROPYL-1,4-DIHYDRO-4-OXO-1,8-NAPHTYRIDINE-3-CARBONIC ACIDS
DE3504643A1 (en) * 1985-02-12 1986-08-14 Bayer Ag, 5090 Leverkusen 1-CYCLOPROPYL-1,4-DIHYDRO-4-OXO-7- (4- (2-OXO-1,3-DIOXOL-4-YL-METHYL) -1-PIPERAZINYL) -3-QUINOLINE CARBONIC ACIDS, METHOD FOR YOURSELF PRODUCTION AND THIS ANTIBACTERIAL AGENT
DE3509546A1 (en) * 1985-03-16 1986-09-25 Bayer Ag, 5090 Leverkusen 7-AMINO-1- (SUBST.CYCLOPROPYL) -1,4-DIHYDRO-4-OXO-3-CHINOLINE CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THE ANTIBACTERIAL AGENTS CONTAINING THEM
DE3608745A1 (en) * 1985-07-24 1987-01-29 Bayer Ag BACTERICIDAL PREPARATIONS FOR APPLICATION IN THE VETERINE MEDICINE AREA
AU594983B2 (en) * 1985-10-29 1990-03-22 Dainippon Pharmaceutical Co. Ltd. Novel quinoline derivatives and processes for preparation thereof
DE3542002A1 (en) * 1985-11-28 1987-06-04 Bayer Ag 1-CYCLOPROPYL-6-FLUOR-1,4-DIHYDRO-4-OXO-7- (1-PIPERAZINYL) -3-QUINOLINE CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THEIR ANTIBACTERIAL AGENTS CONTAINING THEM
US4940710A (en) * 1986-01-17 1990-07-10 American Cyanamid Company 7-(substituted)piperazinyl-1-ethyl-6-fluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids
US5210193A (en) * 1986-01-17 1993-05-11 American Cyanamid Company Piperazine derivatives
AU592845B2 (en) * 1986-01-20 1990-01-25 Kyorin Pharmaceutical Co. Ltd. Process for the preparation of quinolonecarboxylic acid derivatives
DE3705621C2 (en) * 1986-02-25 1997-01-09 Otsuka Pharma Co Ltd Heterocyclic substituted quinolonecarboxylic acid derivatives
US5153204A (en) * 1986-03-01 1992-10-06 Bayer Aktiengesellschaft 7-(1-Pyrrolidinyl)-quinolonecarboxylic acid derivatives
DE3606698A1 (en) * 1986-03-01 1987-09-03 Bayer Ag 7- (1-PYRROLIDINYL) -CHINOLONCARBONIC ACID DERIVATIVES
US4762845A (en) * 1986-05-21 1988-08-09 Abbott Laboratories 7-(3-Substituted imino-1-pyrrolidinyl)-quinolone-3-carboxylic acids
GR1000201B (en) * 1988-06-23 1992-03-20 Tsetis Kleon Method for the synthesis of 1-cyclopropyl-6-fluoro-1,4 dihydro-4-oxo-7-chloro-quinoline-3-carboxylic acid as basis for the preparation of 1-cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-7-piperazine-quinoline-3-carboxylic acids
US5064958A (en) * 1988-11-23 1991-11-12 Pfizer Inc. 1,3-genzoxazine, 2,4-dione derivatives
US4939290A (en) * 1988-11-23 1990-07-03 Pfizer Inc. Benzoic acid derivatives
FR2656611B1 (en) * 1990-01-04 1992-05-07 Hoechst France NEW QUINOLONES, THEIR SALTS, USEFUL AS ANTIMICROBIAL AGENTS, PREPARATION METHOD AND THEIR APPLICATION AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM.
AU4272793A (en) * 1993-04-24 1994-11-21 Korea Research Institute Of Chemical Technology Novel quinolone carboxylic acid derivatives and process for preparing the same
KR950018003A (en) * 1993-12-09 1995-07-22 스미스클라인 비참 피엘씨 Novel quinolone derivatives and methods for their preparation
WO1996002512A1 (en) * 1994-07-18 1996-02-01 Ube Industries, Ltd. Trifluoromethylquinolinecarboxylic acid derivative
WO1996005192A1 (en) * 1994-08-12 1996-02-22 Toyama Chemical Co., Ltd. Novel quinolone- or naphthyridonecarboxylic acid derivative or salt thereof
US5602254A (en) * 1995-05-26 1997-02-11 Warner-Lambert Company Method for making quinoline carboxylic acids or naphthyridine carboxylic acids in free base form
US7098219B2 (en) * 2000-08-01 2006-08-29 Wockhart Limited Inhibitors of cellular efflux pumps of microbes
JP2004518677A (en) 2000-12-21 2004-06-24 ファルマシア・アンド・アップジョン・カンパニー Antibacterial quinolone derivatives and their use to treat bacterial infections
US6878713B2 (en) 2001-04-25 2005-04-12 Wockhardt Limited Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments
US6964966B2 (en) * 2001-04-25 2005-11-15 Wockhardt Limited Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments
US6777420B2 (en) * 2001-06-15 2004-08-17 Microbiotix, Inc. Heterocyclic antibacterial compounds
DE10149557A1 (en) * 2001-10-08 2003-04-10 Jobeck Gmbh Preparation and use of this preparation for combating and / or preventing the causative agent of the fire blight Erwinia amylovora
BR0318460A (en) * 2003-09-04 2006-09-12 Wockhardt Ltd benzoquinolizine-2-carboxylic acid arginine salt tetrahydrate
WO2005026145A2 (en) * 2003-09-12 2005-03-24 Warner-Lambert Company Llc Quinolone antibacterial agents
CA2642754A1 (en) * 2006-02-13 2007-08-23 Trustees Of Boston University Compositions and methods for antibiotic potentiation and drug discovery
WO2008019292A2 (en) * 2006-08-04 2008-02-14 Trustees Of Boston University Compositions and methods for potentiating antibiotic activity
US7884099B2 (en) * 2007-11-16 2011-02-08 Cumbre Ip Ventures, L.P. Quinolone carboxylic acid-substituted rifamycin derivatives
EP2957561A1 (en) * 2014-06-18 2015-12-23 Université Paris 6 Pierre et Marie Curie UPMC Novel fluoroquinolones and use thereof to treat bacterial infections
BR112017023448A2 (en) * 2015-04-29 2018-07-31 The State Of Israel, Ministry Of Agriculture & Rural Development, Agricultural Research Organization (Aro) (Volcani Center) anti-phytopathogenic compositions
CN108617661A (en) * 2017-03-24 2018-10-09 中国海洋大学 A kind of application of alkaloid compound in agricultural drugs
CN109912504B (en) * 2019-04-04 2020-11-10 山东省联合农药工业有限公司 Quinoline carboxylic acid compound and preparation method and application thereof
CN109942488A (en) * 2019-04-04 2019-06-28 山东省联合农药工业有限公司 A kind of quinoline carboxylic acid ester's compound and preparation method thereof and purposes
CN110551124B (en) * 2019-06-14 2021-01-08 山东省联合农药工业有限公司 Quinolone compound or agriculturally and pharmaceutically acceptable salt thereof, and preparation method and application thereof
CN110122493B (en) * 2019-06-14 2022-04-12 山东省联合农药工业有限公司 Use of quinolone compounds for controlling bacterial harmful organisms in useful plants
CN114467947B (en) * 2020-10-26 2023-08-25 山东省联合农药工业有限公司 Synergistic bactericidal composition containing quinolone compounds and application thereof
KR102668356B1 (en) * 2022-01-07 2024-05-21 한국화학연구원 Fire blight control agent of nalidixic acid derivatives

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4146625A (en) * 1976-07-16 1979-03-27 E. I. Du Pont De Nemours And Company Quinolonecarboxylic acids for control of bacterial diseases in plants
JPS53141286A (en) * 1977-05-16 1978-12-08 Kyorin Seiyaku Kk Novel substituted quinolinecarboxylic acid
US4264604A (en) * 1977-07-01 1981-04-28 Ciba-Geigy Corporation Quinolonecarboxylic acid derivatives as bactericides
JPS604820B2 (en) * 1979-02-26 1985-02-06 大塚製薬株式会社 Quinoline carboxylic acid derivative
DE3033157A1 (en) * 1980-09-03 1982-04-01 Bayer Ag, 5090 Leverkusen 7-AMINO-1-CYCLOPROPYL-4-OXO-1,4-DIHYDRO-NAPHTHYRIDINE-3-CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THE ANTIBACTERIAL AGENTS CONTAINING THEM

Also Published As

Publication number Publication date
ATE21011T1 (en) 1986-08-15
EP0113091B1 (en) 1986-07-30
JPS59130802A (en) 1984-07-27
HU194482B (en) 1988-02-29
DE3365027D1 (en) 1986-09-04
DE3248507A1 (en) 1984-07-05
US4563459A (en) 1986-01-07
GR81542B (en) 1984-12-11
AU2286383A (en) 1984-07-05
BR8307166A (en) 1984-08-07
IL70540A (en) 1987-07-31
DK603883D0 (en) 1983-12-28
CA1232198A (en) 1988-02-02
EP0113091A1 (en) 1984-07-11
ZA839647B (en) 1984-08-29
AU563747B2 (en) 1987-07-23
DK603883A (en) 1984-06-30

Similar Documents

Publication Publication Date Title
IL70540A0 (en) Microbicidal agents containing quinolonecarboxylic acids and method of using them
AU570021B2 (en) Analogs of mevalolactone
ES2055341T3 (en) BROMOSULFAMATE AS A BIOCIDE IN THE INHIBITION OF CORROSION, WHICH CONTAINS NITRITE.
PL123130B2 (en) Fungicide and method of manufacture of anilides of isoxazolylcarboxylic acid
AU8570482A (en) Pyridinecarbinols
EP0256128A4 (en) Indoleacetic acid derivatives and use thereof as plant growth regulators.
DE3267766D1 (en) N-cyclohexyl-chloroacetamides, their preparation and their use in combating undesired plant growth
ES8504829A1 (en) Alpha-hydroxy-beta-haloethylphosphinic acids and their salts, and their production and use.
AU554279B2 (en) Cycloalkyl (alpha-triazolyl-beta-hydroxy)-ketones
ES8700650A1 (en) 7-(Aryloxy)-2-naphthoxyalkanecarboxylic acid derivatives, processes for the preparation of these compounds, as well as agents having herbicidal activity containing these compounds.
ES8403113A1 (en) Pyridine derivatives, their preparation and use.
MX9705836A (en) Zinc salts of citraconamic acid and rubber compounds containing such salts.
EP0551632A3 (en) Process for the preparation of halogenoanthranilic acid
JPS5518259A (en) Available chlorine activity maintainer in water
ES475346A1 (en) Halogenated butyric acid chlorides, method for their preparation, and their use as intermediates in the preparation of pesticides.
CS127484A2 (en) Zpusob vyroby n ( trifluormethylfenyl) n propargylpipera zinu
ES8500266A1 (en) Benzoylparabanoic acids.
AU538931B2 (en) (n-thenyl-2-methyl) amino-2-imidazoline
GB1212474A (en) Polyhalo-(sulphonic acid anilides)
IL57555A (en) 1-trimethylsilylphenyl-3-benzoyl-urea derivatives,their production and their use as insecticides
IE812988L (en) 5 - aryl - cyclohexane -1,3-dione herbicides
JPS57159729A (en) Manufacture of trichloromethyl-substituted aromatic compounds and aromatic compounds obtained thereby
DE2964742D1 (en) Derivatives of 1h-inden-1-one, process for their preparation and their use in microbicidal agents and in combating microorganisms

Legal Events

Date Code Title Description
MM9K Patent not in force due to non-payment of renewal fees