IL53904A0 - Azacycloalkanes, azacycloalkenes and derivatives thereof - Google Patents

Azacycloalkanes, azacycloalkenes and derivatives thereof

Info

Publication number: IL53904A0
Authority: IL; Israel
Prior art keywords: azacycloalkenes; azacycloalkanes; derivatives
Prior art date: 1977-01-27

Application number

IL53904A

Other versions

IL53904A (en

Original Assignee

Hoechst Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-01-27

Filing date

1978-01-26

Publication date

1978-04-30

1978-01-26 Application filed by Hoechst Ag filed Critical Hoechst Ag

1978-04-30 Publication of IL53904A0 publication Critical patent/IL53904A0/en

1981-07-31 Publication of IL53904A publication Critical patent/IL53904A/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/12—Oxygen or sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/12—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with only hydrogen atoms attached to the ring nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/16—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with acylated ring nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
- C07D211/94—Oxygen atom, e.g. piperidine N-oxide

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
Neurology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

IL53904A 1977-01-27 1978-01-26 -phenyltolyl azacycloalkane or azacycloalkene derivatives,their preparation and pharmaceutical compositions comprising them IL53904A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US76329477A	1977-01-27	1977-01-27

Publications (2)

Publication Number	Publication Date
IL53904A0 true IL53904A0 (en)	1978-04-30
IL53904A IL53904A (en)	1981-07-31

Family

ID=25067423

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL53904A IL53904A (en)	1977-01-27	1978-01-26	-phenyltolyl azacycloalkane or azacycloalkene derivatives,their preparation and pharmaceutical compositions comprising them

Country Status (18)

Country	Link
JP (1)	JPS5395963A (en)
AT (1)	ATA57578A (en)
BE (1)	BE863402A (en)
CA (1)	CA1103677A (en)
DE (1)	DE2802306A1 (en)
DK (1)	DK38778A (en)
ES (1)	ES466239A1 (en)
FI (1)	FI780237A7 (en)
FR (1)	FR2378770A1 (en)
GB (1)	GB1600654A (en)
GR (1)	GR74891B (en)
HU (1)	HU179982B (en)
IL (1)	IL53904A (en)
NL (1)	NL7800969A (en)
NO (1)	NO780290L (en)
PT (1)	PT67585B (en)
SE (1)	SE7801046L (en)
ZA (1)	ZA78493B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4387229A (en)	1977-09-13	1983-06-07	Pfizer Inc.	3-[2-Hydroxy-4-(substituted)phenyl]azacycloalkanols and derivatives thereof
HU226635B1 (en)	1995-01-23	2009-05-28	Asubio Pharma Co	Piperidine and piperazine derivatives, medicines containing them as active ingredient and their use
HUP9904335A3 (en)	1996-07-22	2001-07-30	Daiichi Asubio Pharma Co Ltd	Arylpiperidinol and arylpiperidine derivatives and drugs containing the same
WO1998003172A1 (en) *	1996-07-22	1998-01-29	Suntory Limited	Arylpiperidinol and arylpiperidine derivatives and drugs containing the same
DE602004016316D1 (en) *	2003-04-04	2008-10-16	Lundbeck & Co As H	4- (2-PHENYLSULFANYL-PHENYL) -PIPERIDINE DERIVATIVES AS SEROTONIN RECOVERY INHIBITORS
UA81300C2 (en) *	2003-04-04	2007-12-25	Lundbeck & Co As H	Derivates of 4-(2-fenilsulfanilfenil)-1,2,3,6-tetrahydropiridin as retarding agents of serotonin recapture
MXPA06013162A (en) *	2004-05-12	2007-02-13	Pfizer Prod Inc	Piperidine derivatives as nk1 and nk3 antagonists.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3674806A (en) *	1969-04-30	1972-07-04	Reynolds Tobacco Co R	1,3,3,4,4-pentasubstituted pyrrolidines

1978
- 1978-01-20 DE DE19782802306 patent/DE2802306A1/en not_active Withdrawn
- 1978-01-21 ES ES466239A patent/ES466239A1/en not_active Expired
- 1978-01-25 FI FI780237A patent/FI780237A7/en not_active Application Discontinuation
- 1978-01-26 AT AT78575A patent/ATA57578A/en not_active Application Discontinuation
- 1978-01-26 PT PT67585A patent/PT67585B/en unknown
- 1978-01-26 DK DK38778A patent/DK38778A/en not_active Application Discontinuation
- 1978-01-26 NL NL7800969A patent/NL7800969A/en not_active Application Discontinuation
- 1978-01-26 HU HU78HO2044A patent/HU179982B/en unknown
- 1978-01-26 IL IL53904A patent/IL53904A/en unknown
- 1978-01-26 NO NO780290A patent/NO780290L/en unknown
- 1978-01-26 ZA ZA00780493A patent/ZA78493B/en unknown
- 1978-01-26 CA CA295,695A patent/CA1103677A/en not_active Expired
- 1978-01-27 SE SE7801046A patent/SE7801046L/en unknown
- 1978-01-27 JP JP747178A patent/JPS5395963A/en active Pending
- 1978-01-27 GB GB3384/78A patent/GB1600654A/en not_active Expired
- 1978-01-27 FR FR7802276A patent/FR2378770A1/en active Granted
- 1978-01-27 BE BE184696A patent/BE863402A/en unknown
1979
- 1979-12-21 GR GR55274A patent/GR74891B/el unknown

Also Published As

Publication number	Publication date
CA1103677A (en)	1981-06-23
FI780237A7 (en)	1978-07-28
ATA57578A (en)	1982-07-15
ES466239A1 (en)	1979-06-01
FR2378770B1 (en)	1981-06-19
DE2802306A1 (en)	1978-08-10
ZA78493B (en)	1978-12-27
FR2378770A1 (en)	1978-08-25
NL7800969A (en)	1978-07-31
GB1600654A (en)	1981-10-21
IL53904A (en)	1981-07-31
BE863402A (en)	1978-07-27
GR74891B (en)	1984-07-12
PT67585A (en)	1978-02-01
NO780290L (en)	1978-07-28
SE7801046L (en)	1978-07-28
HU179982B (en)	1983-01-28
PT67585B (en)	1979-11-12
DK38778A (en)	1978-07-28
JPS5395963A (en)	1978-08-22

Publication	Publication Date	Title
NZ192231A (en)	1981-11-19	2-chloro-5-trichloromethyl-pyridine and 2,3-dichloro-5-trichloromethylpyridine
AU3921478A (en)	1980-02-28	3,4,5 trihydroxypiperidine derivatives
AU4113878A (en)	1980-05-01	1-alkanoyl-proline derivatives
GB2003876A (en)	1979-03-21	Beta-haloethylamine derivatives
ZA785699B (en)	1980-05-28	Isochromans,isothiochromans,2-benzoxepins and 2-benzothiopins
GB1557019A (en)	1979-12-05	Metalsulphonamido-benzamide derivatives
GB2008579B (en)	1982-11-03	2-imino-imidazolidine derivatives
AU3888578A (en)	1980-02-21	4-hydroxy-2-benzimidazolinone derivatives
PH16029A (en)	1983-06-02	2-deoxyfortimicin a,4-n-alkyl and 4-n-acyl-2-deoxyfortimicin b derivatives
GB2009180B (en)	1982-05-26	25-alkylcholestrerol derivatives
IL53904A0 (en)	1978-04-30	Azacycloalkanes, azacycloalkenes and derivatives thereof
PH18632A (en)	1985-08-23	4-alkylthio-2-trifluoromethylalkanesulfonanilides and derivatives thereof
GB2009150B (en)	1982-08-18	Tetrahydrophtalamide derivatives
GB2005261B (en)	1982-03-17	2-oxazolydone derivatives
PT68947A (en)	1979-01-01	2,3-dicyanopyrazine derivatives
AU3313978A (en)	1979-08-16	Everninomicin derivatives
GB2003479A (en)	1979-03-14	3-amino-17alpha-aza-d-homoandrostane derivatives
GB2014131A (en)	1979-08-22	1-hydrocarbylpyrrole derivatives
GB2017104B (en)	1982-01-20	4-thia-2,6-diaza-bicyclo-(3,2,0-)-heptane derivatives
GB2000128B (en)	1982-02-03	15-substituted-omega-pentanorprostaglandin derivatives
JPS5448753A (en)	1979-04-17	Digoxigenine derivatives and manufacture
IL55865A0 (en)	1979-01-31	4-desacetoxy-4-oxovinblastine, 4-descetoxy-4-alpha-hydroxyvinblastine and related compounds
GB2008119B (en)	1982-05-19	Arylsteroid derivatives
AU4129978A (en)	1979-05-17	Eburnamenine derivatives
AU3347778A (en)	1979-08-30	1,2,4,-benzotriazine-di-n-oxide derivatives