IL44237A - 2-benzofuranyl-piperidine(or-tetrahydropyridine)derivatives their preparation and pharmaceutical compositions containing them - Google Patents

2-benzofuranyl-piperidine(or-tetrahydropyridine)derivatives their preparation and pharmaceutical compositions containing them

Info

Publication number: IL44237A
Authority: IL; Israel
Prior art keywords: group; hydrogen; represent; general formula; compounds
Prior art date: 1973-03-02

Application number

IL44237A

Other languages

English (en)

Other versions

IL44237A0 (en

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1973-03-02

Filing date

1974-02-19

Publication date

1977-08-31

1974-02-19 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1974-05-16 Publication of IL44237A0 publication Critical patent/IL44237A0/xx

1976-11-24 Priority to IL50987A priority Critical patent/IL50987A/xx

1977-08-31 Publication of IL44237A publication Critical patent/IL44237A/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/30—Oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Psychiatry (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Hydrogenated Pyridines (AREA)

IL44237A 1973-03-02 1974-02-19 2-benzofuranyl-piperidine(or-tetrahydropyridine)derivatives their preparation and pharmaceutical compositions containing them IL44237A (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
IL50987A IL50987A (en)	1974-02-19	1976-11-24	4-(2-benzofuranyl)-piperidine and tetrahydropyridine derivatices their preparation and pharmaceutical compositions containin them

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
CH310373A CH592656A5 (de)	1973-03-02	1973-03-02

Publications (2)

Publication Number	Publication Date
IL44237A0 IL44237A0 (en)	1974-05-16
IL44237A true IL44237A (en)	1977-08-31

Family

ID=4248678

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL44237A IL44237A (en)	1973-03-02	1974-02-19	2-benzofuranyl-piperidine(or-tetrahydropyridine)derivatives their preparation and pharmaceutical compositions containing them

Country Status (24)

Country	Link
US (1)	US4210655A (de)
JP (2)	JPS599557B2 (de)
AR (4)	AR205619A1 (de)
AT (1)	AT336014B (de)
BE (1)	BE811767A (de)
CA (1)	CA1045139A (de)
CH (1)	CH592656A5 (de)
CS (5)	CS176296B2 (de)
DD (1)	DD113007A5 (de)
DE (1)	DE2408476A1 (de)
DK (1)	DK147318C (de)
ES (1)	ES423711A1 (de)
FR (1)	FR2219781B1 (de)
GB (1)	GB1465581A (de)
HU (1)	HU172464B (de)
IE (1)	IE38907B1 (de)
IL (1)	IL44237A (de)
LU (1)	LU69510A1 (de)
MX (1)	MX3765E (de)
NL (1)	NL179206C (de)
SE (1)	SE410856B (de)
SU (6)	SU560531A3 (de)
YU (2)	YU52374A (de)
ZA (1)	ZA741362B (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH609054A5 (en) *	1975-11-26	1979-02-15	Ciba Geigy Ag	Process for the preparation of a novel piperidine derivative
EP0006524A1 (de) *	1978-06-22	1980-01-09	Ciba-Geigy Ag	Neue Tetrahydropyridin- und Piperidinderivate und deren Säureadditionssalze, Verfahren zu deren Herstellung und solche enthaltende pharmazeutische Zusammensetzungen
US4284638A (en) *	1978-11-21	1981-08-18	Ciba-Geigy Corporation	Pharmaceutical compositions with central depressant and antipsychotic activity having a butyrophenone derivative which is substituted in the 4-position and a C-(2-benzofuranyl)-piperidine or C-(2-benzofuranyl)-tetrahydro-pyridine
US5045551A (en) *	1989-09-19	1991-09-03	Allergan, Inc.	Acetylenes disubstituted with a heteroaromatic group and a 2-substituted chromanyl, thiochromanyl or 1,2,3,4-tetrahydroquinolinyl group having retinoid-like activity
US5455254A (en) *	1991-02-15	1995-10-03	Mondadori; Cesare	Substituted benzofuranylpiperidine as a nootropic agent
RU2095339C1 (ru) *	1991-10-17	1997-11-10	Циба-Гейги АГ	Производные гидрохинона в свободном виде или в виде соли, способы их получения, производные пиперидина и способы их получения
WO1993016695A1 (en) *	1992-02-21	1993-09-02	Ciba-Geigy Ag	Brofaromine as an agent for treating post-traumatic stress
US5693807A (en) *	1992-10-14	1997-12-02	Ciba-Geigy Corporation	Substituted hydroquinone derivatives
ATE180780T1 (de) *	1993-08-05	1999-06-15	Hoechst Marion Roussel Inc	2-(piperidin-4-yl, pyridin-4-yl und tetrahydropyridin-4-yl)-benzofuran-7-carbamat derivate, ihre herstellung und verwendung als acetylcholinesterase inhibitoren
GB9605065D0 (en) *	1996-03-11	1996-05-08	Merck Sharp & Dohme	Therapeutic agents
WO2000073269A2 (en)	1999-06-02	2000-12-07	Regents Of The University Of Minnesota	Nicotine receptor ligands
WO2011162364A1 (ja) *	2010-06-23	2011-12-29	住友化学株式会社	有害節足動物防除組成物および複素環化合物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR1461633A (fr) *	1964-11-11	1966-02-25	Belge Produits Chimiques Sa	Nouveaux dérivés benzofuranniques, leurs sels et procédés de préparation de cesdérivés et de leurs sels
GB1041525A (en) *	1964-11-11	1966-09-07	Belge Produits Chimiques Sa	Benzofuran derivatives and processes for preparing the same
IE39264B1 (en) *	1973-05-25	1978-08-30	Ciba Geigy Ag	New pharmaceutical preparations

1973
- 1973-03-02 CH CH310373A patent/CH592656A5/xx not_active IP Right Cessation
1974
- 1974-01-01 AR AR252581A patent/AR205619A1/es active
- 1974-02-19 IL IL44237A patent/IL44237A/en unknown
- 1974-02-20 IE IE00340/74A patent/IE38907B1/xx unknown
- 1974-02-21 SE SE7402294A patent/SE410856B/xx not_active IP Right Cessation
- 1974-02-22 DE DE19742408476 patent/DE2408476A1/de active Granted
- 1974-02-25 CA CA193,450A patent/CA1045139A/en not_active Expired
- 1974-02-28 NL NLAANVRAGE7402755,A patent/NL179206C/xx not_active IP Right Cessation
- 1974-02-28 CS CS8937A patent/CS176296B2/cs unknown
- 1974-02-28 SU SU2000455A patent/SU560531A3/ru active
- 1974-02-28 ES ES423711A patent/ES423711A1/es not_active Expired
- 1974-02-28 CS CS1495A patent/CS176266B2/cs unknown
- 1974-02-28 CS CS8938A patent/CS176297B2/cs unknown
- 1974-02-28 LU LU69510*A patent/LU69510A1/xx unknown
- 1974-02-28 DD DD176867A patent/DD113007A5/xx unknown
- 1974-02-28 FR FR7406834A patent/FR2219781B1/fr not_active Expired
- 1974-02-28 CS CS8939A patent/CS176298B2/cs unknown
- 1974-02-28 CS CS8940A patent/CS176299B2/cs unknown
- 1974-02-28 YU YU00523/74A patent/YU52374A/xx unknown
- 1974-02-28 HU HU74CI00001456A patent/HU172464B/hu unknown
- 1974-03-01 AT AT170674A patent/AT336014B/de not_active IP Right Cessation
- 1974-03-01 GB GB927974A patent/GB1465581A/en not_active Expired
- 1974-03-01 BE BE141551A patent/BE811767A/xx not_active IP Right Cessation
- 1974-03-01 ZA ZA00741362A patent/ZA741362B/xx unknown
- 1974-03-01 MX MX745143U patent/MX3765E/es unknown
- 1974-03-01 DK DK110174A patent/DK147318C/da not_active IP Right Cessation
- 1974-03-02 JP JP49024715A patent/JPS599557B2/ja not_active Expired
1975
- 1975-06-30 AR AR259412A patent/AR210858A1/es active
- 1975-06-30 AR AR259413A patent/AR208554A1/es active
1976
- 1976-05-05 AR AR263204A patent/AR211860A1/es active
- 1976-09-24 SU SU762404754A patent/SU612630A3/ru active
- 1976-09-24 SU SU762402851A patent/SU651702A3/ru active
- 1976-09-28 SU SU762404895A patent/SU646911A4/ru active
- 1976-11-02 SU SU762415644A patent/SU649321A3/ru active
1977
- 1977-08-24 SU SU772514703A patent/SU651703A3/ru active
1978
- 1978-04-05 US US05/893,104 patent/US4210655A/en not_active Expired - Lifetime
1980
- 1980-08-25 YU YU02123/80A patent/YU212380A/xx unknown
1982
- 1982-06-16 JP JP57102323A patent/JPS6046115B2/ja not_active Expired

Also Published As

Publication number	Publication date
JPS599557B2 (ja)	1984-03-03
ZA741362B (en)	1975-01-29
CS176266B2 (de)	1977-06-30
FR2219781A1 (de)	1974-09-27
US4210655A (en)	1980-07-01
AT336014B (de)	1977-04-12
SU651703A3 (ru)	1979-03-05
SU646911A4 (ru)	1979-02-05
FR2219781B1 (de)	1977-07-01
DK147318B (da)	1984-06-18
DE2408476A1 (de)	1974-09-12
SU649321A3 (ru)	1979-02-25
GB1465581A (en)	1977-02-23
YU212380A (en)	1983-04-27
AR205619A1 (es)	1976-05-21
YU37163B (de)	1984-08-31
NL7402755A (de)	1974-09-04
JPS584781A (ja)	1983-01-11
DE2408476C2 (de)	1990-12-06
SU612630A3 (ru)	1978-06-25
JPS6046115B2 (ja)	1985-10-14
CA1045139A (en)	1978-12-26
AR210858A1 (es)	1977-09-30
IE38907B1 (en)	1978-06-21
AU6619274A (en)	1975-09-04
AR211860A1 (es)	1978-03-31
NL179206C (nl)	1986-08-01
IE38907L (en)	1974-09-02
CH592656A5 (de)	1977-10-31
JPS49117474A (de)	1974-11-09
CS176296B2 (de)	1977-06-30
DK147318C (da)	1984-12-24
ES423711A1 (es)	1977-01-16
AR208554A1 (es)	1977-02-15
IL44237A0 (en)	1974-05-16
SU651702A3 (ru)	1979-03-05
MX3765E (es)	1981-06-25
SU560531A3 (ru)	1977-05-30
CS176297B2 (de)	1977-06-30
LU69510A1 (de)	1975-12-09
HU172464B (hu)	1978-09-28
BE811767A (fr)	1974-09-02
SE410856B (sv)	1979-11-12
CS176299B2 (de)	1977-06-30
YU52374A (en)	1982-06-18
ATA170674A (de)	1976-08-15
DD113007A5 (de)	1975-05-12
CS176298B2 (de)	1977-06-30

Publication	Publication Date	Title
CA1119601A (en)	1982-03-09	Tetrahydropyridine and piperidine derivatives and their acid addition salts, processes for their preparation and pharmaceutical preparations containing such compounds
US5478828A (en)	1995-12-26	Piperazinyl-and piperidinyl-cyclohexanols
US5292761A (en)	1994-03-08	Piperidine, tetrahydropyridine and pyrrolidine compounds
US3980658A (en)	1976-09-14	(Indolyl-piperidino or -1,2,5,6-tetrahydro-pyridyl)-p-fluoro-butyrophenones and salts thereof
CA2122911C (en)	2003-10-14	1,3-substituted cycloalkenes and cycloalkanes as central nervous system agents
US3946022A (en)	1976-03-23	Piperidine derivatives
IL44237A (en)	1977-08-31	2-benzofuranyl-piperidine(or-tetrahydropyridine)derivatives their preparation and pharmaceutical compositions containing them
US3821234A (en)	1974-06-28	1-pyrazoly-alkyl-4-phenyl-3,4-dehydropiperidines
US3458521A (en)	1969-07-29	4-phenylpiperidine derivatives
CA1120036A (en)	1982-03-16	4-(naphthylmethyl)piperidine derivatives
US4542132A (en)	1985-09-17	Cardiac stimulating cyclic sulfonamido substituted 4-piperidino-quinazoline derivatives, compositions, and method of use therefor
US4016281A (en)	1977-04-05	Tetralone and indanone compounds
US4600719A (en)	1986-07-15	Tetrahydropyridine and piperidine derivatives
US5486527A (en)	1996-01-23	Anticholinergic agents
US4166174A (en)	1979-08-28	Benzazocine derivatives and process for preparing the same
NO121212B (de)	1971-02-01
US3974280A (en)	1976-08-10	Benzothiophenes
US4076821A (en)	1978-02-28	4,4-Diphenylcycloalkylpiperidines and psychotropic compositions thereof
GB1565055A (en)	1980-04-16	Tetrahydropyridine and piperidine derivatives and processes for the preparation thereof
US5240942A (en)	1993-08-31	Piperidine, tetrahydropyridine and pyrrolidine compounds
IE64206B1 (en)	1995-07-12	Disubstituted piperidines and pyrrolidines as anticholinergic agents
US3391143A (en)	1968-07-02	9-piperidyl and 9-piperidylidene derivatives of acridan
US4345081A (en)	1982-08-17	Spiro[indoline-3,4'-piperidine]s
US4248876A (en)	1981-02-03	Piperidine derivatives
US4524207A (en)	1985-06-18	Process for preparing substituted 1,3-dihydrospiro[benzo(c)thiophene]s