IL121461A0 - Use of 1-[4-[4-aryl (or heteroaryl)-1-piperazinyl]butyl]-1H-azole derivatives - Google Patents
Use of 1-[4-[4-aryl (or heteroaryl)-1-piperazinyl]butyl]-1H-azole derivativesInfo
- Publication number
- IL121461A0 IL121461A0 IL12146196A IL12146196A IL121461A0 IL 121461 A0 IL121461 A0 IL 121461A0 IL 12146196 A IL12146196 A IL 12146196A IL 12146196 A IL12146196 A IL 12146196A IL 121461 A0 IL121461 A0 IL 121461A0
- Authority
- IL
- Israel
- Prior art keywords
- piperazinyl
- heteroaryl
- aryl
- butyl
- azole derivatives
- Prior art date
Links
- 125000001072 heteroaryl group Chemical group 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Otolaryngology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9514690A FR2742052B1 (en) | 1995-12-12 | 1995-12-12 | USE OF DERIVATIVES 1- (4- (4-ARYL (OR HETEROARYL) -1-PIPER AZINYL) -BUTY) -1H-AZOLE FOR THE TREATMENT OF DEPRESSION, OBSESSIVE COMPULSIVE DISORDERS, SLEEP APNEA, SEXUAL DYSFUNCTIONS , Emese and motion sickness |
PCT/EP1996/005736 WO1997021439A1 (en) | 1995-12-12 | 1996-12-11 | Medicament intended to the treatment of obsessive compulsive troubles, sleep apnoea, sexual dysfunctions, emesa and transport sickness |
Publications (1)
Publication Number | Publication Date |
---|---|
IL121461A0 true IL121461A0 (en) | 1998-02-08 |
Family
ID=9485400
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL12146196A IL121461A0 (en) | 1995-12-12 | 1996-12-11 | Use of 1-[4-[4-aryl (or heteroaryl)-1-piperazinyl]butyl]-1H-azole derivatives |
Country Status (16)
Country | Link |
---|---|
EP (1) | EP0808166A1 (en) |
JP (1) | JPH11501051A (en) |
CN (1) | CN1177297A (en) |
AR (1) | AR004378A1 (en) |
AU (1) | AU716665B2 (en) |
CA (1) | CA2211161A1 (en) |
CZ (1) | CZ255197A3 (en) |
ES (1) | ES2134709B1 (en) |
FR (1) | FR2742052B1 (en) |
HU (1) | HUP9800198A2 (en) |
IL (1) | IL121461A0 (en) |
NO (1) | NO973589L (en) |
PL (1) | PL321779A1 (en) |
TR (1) | TR199700794T1 (en) |
WO (1) | WO1997021439A1 (en) |
ZA (1) | ZA9610457B (en) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2763950B1 (en) * | 1997-06-02 | 2002-09-20 | Esteve Labor Dr | 2- {4- [4- (4,5-DICHLORO-2-METHYLIMIDAZOL-1-YL) BUTYL] -1- PIPERAZINYL} -5-FLUOROPYRIMIDINE, ITS PREPARATION AND THERAPEUTIC USE |
TW526202B (en) * | 1998-11-27 | 2003-04-01 | Shionogi & Amp Co | Broad spectrum cephem having benzo[4,5-b]pyridium methyl group of antibiotic activity |
US6046331A (en) * | 1998-12-17 | 2000-04-04 | Synaptic Pharmaceutical Corporation | Imidazolones and their use in treating benign prostatic hyperplasia and other disorders |
US7309703B2 (en) | 2000-08-14 | 2007-12-18 | Ortho Mcneil Pharmaceutical, Inc. | Substituted pyrazoles |
CA2419550A1 (en) | 2000-08-14 | 2002-02-21 | Ortho-Mcneil Pharmaceutical, Inc. | Substituted pyrazoles |
US7332494B2 (en) | 2000-08-14 | 2008-02-19 | Janssen Pharmaceutica, N.V. | Method for treating allergies using substituted pyrazoles |
CZ307185B6 (en) | 2000-08-14 | 2018-03-07 | Ortho Mcneil Pharmaceutical, Inc. | Substituted pyrazole, a pharmaceutical composition containing it and their medical applications |
RU2290179C2 (en) | 2000-09-06 | 2006-12-27 | Орто-Макнейл Фармасьютикал, Инк. | Method for treatment of allergy by using substituted pyrazoles |
EP1715921B1 (en) | 2003-09-25 | 2013-04-24 | Abraxis BioScience, Inc. | Tetrahydroindolone derivatives for treatment of neurological conditions |
WO2005094827A1 (en) * | 2004-03-30 | 2005-10-13 | Kestrel Pharmaceuticals Inc. | Methods for treating sexual dysfunction |
ES2340066T3 (en) | 2005-04-26 | 2010-05-28 | Hypnion, Inc. | BENZISOXAZOL PIPERIDINE COMPOUNDS AND PROCEDURE FOR THE SAME USE. |
WO2006116615A1 (en) | 2005-04-26 | 2006-11-02 | Hypnion, Inc. | Benzisoxazole piperazine compounds and methods of use thereof |
GB2435827A (en) * | 2006-03-09 | 2007-09-12 | Del Dr Esteve S A Spain Lab | Use of substituted piperazine compounds for the treatment of food related disorders |
CN115304590B (en) * | 2022-09-19 | 2024-05-28 | 皮摩尔新药(辽宁)有限公司 | 2H-benzotriazole derivatives, preparation method thereof and pharmaceutical composition containing same |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2672052B1 (en) * | 1991-01-28 | 1995-05-24 | Esteve Labor Dr | DERIVATIVES OF ARYL (OR HETEROARYL) -PIPERAZINYL-ALKYL-AZOLES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICAMENTS. |
FR2723091B1 (en) * | 1994-07-29 | 1996-11-08 | Esteve Labor Dr | TETRAHYDROPYRIDINE- (6,4-HYDROXYPIPERIDINE) ALKYLAZOLES |
-
1995
- 1995-12-12 FR FR9514690A patent/FR2742052B1/en not_active Expired - Fee Related
-
1996
- 1996-12-11 WO PCT/EP1996/005736 patent/WO1997021439A1/en not_active Application Discontinuation
- 1996-12-11 IL IL12146196A patent/IL121461A0/en unknown
- 1996-12-11 CZ CZ972551A patent/CZ255197A3/en unknown
- 1996-12-11 TR TR97/00794T patent/TR199700794T1/en unknown
- 1996-12-11 EP EP96944029A patent/EP0808166A1/en not_active Withdrawn
- 1996-12-11 JP JP9521756A patent/JPH11501051A/en active Pending
- 1996-12-11 HU HU9800198A patent/HUP9800198A2/en unknown
- 1996-12-11 CN CN96192286A patent/CN1177297A/en active Pending
- 1996-12-11 PL PL96321779A patent/PL321779A1/en unknown
- 1996-12-11 AU AU13764/97A patent/AU716665B2/en not_active Ceased
- 1996-12-11 CA CA002211161A patent/CA2211161A1/en not_active Abandoned
- 1996-12-12 AR ARP960105644A patent/AR004378A1/en unknown
- 1996-12-12 ZA ZA9610457A patent/ZA9610457B/en unknown
- 1996-12-12 ES ES009602700A patent/ES2134709B1/en not_active Expired - Lifetime
-
1997
- 1997-08-04 NO NO973589A patent/NO973589L/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
FR2742052A1 (en) | 1997-06-13 |
ES2134709B1 (en) | 2000-05-16 |
MX9706133A (en) | 1997-11-29 |
TR199700794T1 (en) | 1997-11-21 |
AU1376497A (en) | 1997-07-03 |
NO973589L (en) | 1997-10-08 |
CN1177297A (en) | 1998-03-25 |
NO973589D0 (en) | 1997-08-04 |
PL321779A1 (en) | 1997-12-22 |
EP0808166A1 (en) | 1997-11-26 |
CZ255197A3 (en) | 1998-01-14 |
CA2211161A1 (en) | 1997-06-19 |
WO1997021439A1 (en) | 1997-06-19 |
AU716665B2 (en) | 2000-03-02 |
JPH11501051A (en) | 1999-01-26 |
FR2742052B1 (en) | 1998-04-10 |
HUP9800198A2 (en) | 1999-09-28 |
AR004378A1 (en) | 1998-11-04 |
ES2134709A1 (en) | 1999-10-01 |
ZA9610457B (en) | 1997-06-24 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PL327406A1 (en) | 1-(1,2-disubstituted-piperidinyl)-4-substituted derivatives of piperazine | |
NZ328387A (en) | 4-[2-(n-(heteroaryl)-hydrazonoethyloxy)]benzoyl-2-benzyloxy-carbonylamino-alanine derivatives and medicaments containing them | |
PL331431A1 (en) | Fluorine containing 1,4-substituted derivatives of piperidine | |
IL121461A0 (en) | Use of 1-[4-[4-aryl (or heteroaryl)-1-piperazinyl]butyl]-1H-azole derivatives | |
HUP9601328A2 (en) | 4-(aryl-amino-methylene)-2,4-dihydro-pyrazol-3-one derivatives and pharmaceutical compositions containing them | |
AU7692696A (en) | Heteroaryl derivatives | |
AU4620397A (en) | Piperazine derivatives | |
AU1619400A (en) | Modified adp-glucose pyrophosphorylase for improvement and optimization of plantphenotypes | |
AP9901458A0 (en) | Crystalline form of 4-[5-methyl-3-phenylsoxanol-4-yl] benzenesulfonamide | |
IL112249A0 (en) | Heterocyclic pyrimidine derivatives and pharmaceutical compositions containing them | |
NZ325845A (en) | 1-(1,2-disubstituted piperidinyl)-4-(fused imidazole)-piperidine derivatives, preparation and pharmaceutical use thereof | |
AU3039995A (en) | Heterocyclic derivatives of N-phenylamides | |
AU1824199A (en) | Folding window rack | |
PL338947A1 (en) | Derivatives of 2-(4-aryl or heteroaryl piperazin-1-ylmethyl)-1h-indole | |
AUPO735997A0 (en) | Piperazine derivatives | |
GB9515412D0 (en) | 2-(4-substituted)-benzylamino-2-methyl-propanamide derivatives | |
PL316382A1 (en) | Novel derivatives of piperidine | |
HU9802129D0 (en) | New piperazine and piperidine derivatives | |
ZA948520B (en) | 1-[2H-1-benzopyran-2one-8-yl]-piperazine derivatives | |
AU4664596A (en) | Antipsychotic 4-(1h-indolyl-1-yl)-1-substituted piperidine derivatives | |
AU7580796A (en) | Piperidine and tetrahydropyridine derivatives | |
AU7578296A (en) | Piperazine, piperidine and tetrahydropyridine derivatives | |
AU1018801A (en) | Use of 3,4-substituted piperidines | |
HU9202914D0 (en) | 4-(4-(4-hydroxiphenyl)-1-piperazinyl)-5-methyl-3h-1,2,4-triazole-3-one derivatives | |
GB9517381D0 (en) | Aryl and heteroaryl piperazine derivatives |