[go: up one dir, main page]

IL115585A0 - Dipeptide derivatives, processes for the preparation thereof and pharmaceutical compositions containing them - Google Patents

Dipeptide derivatives, processes for the preparation thereof and pharmaceutical compositions containing them

Info

Publication number
IL115585A0
IL115585A0 IL11558595A IL11558595A IL115585A0 IL 115585 A0 IL115585 A0 IL 115585A0 IL 11558595 A IL11558595 A IL 11558595A IL 11558595 A IL11558595 A IL 11558595A IL 115585 A0 IL115585 A0 IL 115585A0
Authority
IL
Israel
Prior art keywords
processes
preparation
pharmaceutical compositions
compositions containing
dipeptide derivatives
Prior art date
Application number
IL11558595A
Other versions
IL115585A (en
Original Assignee
Boehringer Mannheim Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Mannheim Gmbh filed Critical Boehringer Mannheim Gmbh
Publication of IL115585A0 publication Critical patent/IL115585A0/en
Publication of IL115585A publication Critical patent/IL115585A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Compounds of formula (I) in which R<1> and R<2> are hydroxy or an acyloxy group and R<3> is hydrogen, where R<2> and R<3> together may also signify a valency line. Process for their production from cyanobacteria of the Oscillatoria agardhii genus, and medicaments containing said compounds with a thrombin and trypsin inhibiting action.
IL11558595A 1994-10-14 1995-10-12 Dipeptide derivatives processes for the preparation thereof and pharmaceutical compositions containing them IL115585A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4436772A DE4436772A1 (en) 1994-10-14 1994-10-14 New dipeptide derivative, process for its preparation and medicinal products containing this compound

Publications (2)

Publication Number Publication Date
IL115585A0 true IL115585A0 (en) 1996-01-19
IL115585A IL115585A (en) 1999-09-22

Family

ID=6530791

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11558595A IL115585A (en) 1994-10-14 1995-10-12 Dipeptide derivatives processes for the preparation thereof and pharmaceutical compositions containing them

Country Status (9)

Country Link
EP (1) EP0788510B1 (en)
JP (1) JPH10507191A (en)
AT (1) ATE189229T1 (en)
AU (1) AU3804795A (en)
CA (1) CA2202379A1 (en)
DE (2) DE4436772A1 (en)
IL (1) IL115585A (en)
WO (1) WO1996011941A1 (en)
ZA (1) ZA958644B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6716869B2 (en) 2001-12-17 2004-04-06 Pharmacia Corporation Protease inhibitors of the coagulation cascade isolated from Dysidea sponges
KR101086259B1 (en) 2004-12-22 2011-11-24 에스케이케미칼주식회사 A composition for the treatment and prevention of cancer comprising an oscillatoria agardihi extract and a method of preparing the extract

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3505555A1 (en) * 1985-02-18 1986-09-11 Behringwerke Ag, 3550 Marburg NEW OLIGOPEPTIDYLARGININOL DERIVATIVES AND THEIR HOMOLOGOLOGY, METHOD FOR THE PRODUCTION THEREOF, THE USE THEREOF AND MEANS CONTAINING THEM
SE9103612D0 (en) * 1991-12-04 1991-12-04 Astra Ab NEW PEPTIDE DERIVATIVES

Also Published As

Publication number Publication date
JPH10507191A (en) 1998-07-14
CA2202379A1 (en) 1996-04-25
DE4436772A1 (en) 1996-04-18
EP0788510B1 (en) 2000-01-26
WO1996011941A1 (en) 1996-04-25
DE59507710D1 (en) 2000-03-02
EP0788510A1 (en) 1997-08-13
ATE189229T1 (en) 2000-02-15
ZA958644B (en) 1997-04-14
AU3804795A (en) 1996-05-06
IL115585A (en) 1999-09-22

Similar Documents

Publication Publication Date Title
TW289757B (en)
ZA962694B (en) Carbonyl piperazinyl and piperidinyl compounds
MX9604020A (en) Arylalkyldiazinones.
MY132115A (en) Novel thrombin inhibitors
MY106280A (en) Novel benzopyrido piperidine, piperidylidene and piperazine compounds, compositions, methods of manufacture and methods of use.
IL112622A (en) Iminoalkylamino or aminoalkylideneamino camptothecin derivatives, process for their preparation and pharmaceutical compositions containing them
CA2019404A1 (en) 11 beta-aryl-4-estrenes, process for their production as well as their use as pharmaceutical agents
AP9701041A0 (en) Pyridylpyrrole compounds.
IL117091A0 (en) Methylphenyloxazolidinone derivatives pharmaceutical compositions containing the same and processes for the preparation thereof
MX9503529A (en) Glycinamide derivatives, process for their preparation and medicaments containing them.
GR3021789T3 (en) 17-Aryl and 17-heterocyclyl-14beta-5alpha-androstane, androstene and androstadiene derivatives active on the cardiovascular system, processes for their preparation and pharmaceutical compositions containing same
AU1306795A (en) Anticonvulsant pseudofructopyranose sulfamates
MY120683A (en) New phenylamidine derivatives, processes for their preparation and their use as pharmaceuticals.
MY114282A (en) Anthracycline derivatives
IL115585A (en) Dipeptide derivatives processes for the preparation thereof and pharmaceutical compositions containing them
MY114693A (en) Substituted benzenesulfonylureas and thioureas,processes for their preparation,their use for the production of pharmaceutical preparations, and pharmaceutical preparation containing them
MY115795A (en) Substituted benzenesulfonylureas and -thioureas, processes for their preparation and use of pharmaceutical preparations based on these compounds, and medicaments containing them
AU2067592A (en) New n-(isoquinolin-5-ylsulphonyl)azacycloalkanes, process for the preparation thereof, and pharmaceutical compositions containing them
AU6970394A (en) Desoxyazaphospholipid derivatives having inhibiting activity on phospholipase a2
ZA986730B (en) Streptogramin derivatives their preparation and compositions containing them
AU5522794A (en) New angiopeptin cyclopeptide compounds, process for the preparation thereof, and pharmaceutical compositios containing them
TW344650B (en) Fungicidal compositions and the process for the preparation thereof
MY113432A (en) Substituted benzenesulfonylureas and -thioureas, processes for their preparation, their use for the production of pharmaceutical preparations, and medicaments containing them
AU4154993A (en) New peptide compounds active in cell adhesion processes, a process for the preparation thereof, and pharmaceutical compositions containing them
AU1192097A (en) 3-aminoethyl-n-amidino-2,5-dihydropyrrole derivatives having arginine mimetic properties

Legal Events

Date Code Title Description
FF Patent granted
MM9K Patent not in force due to non-payment of renewal fees