IE47271B1 - Process for the preparation of 1-n-acyl-aminoglycosides - Google Patents

Process for the preparation of 1-n-acyl-aminoglycosides

Info

Publication number: IE47271B1
Authority: IE; Ireland
Prior art keywords: amino; groups; aminoglycoside; polysilylated; formula
Prior art date: 1977-04-28

Application number

IE842/78A

Other languages

English (en)

Other versions

IE780842L (en

Inventor

Martin John Cron

John Gerard Keil

Jeng Shyong Lin

Mariano Vecchio Ruggeri

Derek Walker

Original Assignee

Bristol Myers Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-04-28

Filing date

1978-04-27

Publication date

1984-02-08

1978-04-27 Application filed by Bristol Myers Co filed Critical Bristol Myers Co

1978-10-28 Publication of IE780842L publication Critical patent/IE780842L/xx

1984-02-08 Publication of IE47271B1 publication Critical patent/IE47271B1/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Health & Medical Sciences (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Life Sciences & Earth Sciences (AREA)
Saccharide Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

IE842/78A 1977-04-28 1978-04-27 Process for the preparation of 1-n-acyl-aminoglycosides IE47271B1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US79180677A	1977-04-28	1977-04-28
US88858578A	1978-03-20	1978-03-20

Publications (2)

Publication Number	Publication Date
IE780842L IE780842L (en)	1978-10-28
IE47271B1 true IE47271B1 (en)	1984-02-08

Family

ID=27121201

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
IE842/78A IE47271B1 (en)	1977-04-28	1978-04-27	Process for the preparation of 1-n-acyl-aminoglycosides
IE841/78A IE46945B1 (en)	1977-04-28	1978-04-27	Process for the preparation of kanamycin derivatives

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
IE841/78A IE46945B1 (en)	1977-04-28	1978-04-27	Process for the preparation of kanamycin derivatives

Country Status (27)

Country	Link
JP (1)	JPS53149951A (xx)
AR (1)	AR218910A1 (xx)
AT (1)	AT357675B (xx)
CA (2)	CA1105454A (xx)
CH (1)	CH639104A5 (xx)
CS (1)	CS207607B2 (xx)
CY (1)	CY1241A (xx)
DE (2)	DE2818822A1 (xx)
DK (2)	DK172543B1 (xx)
EG (1)	EG13710A (xx)
ES (1)	ES469303A1 (xx)
FI (1)	FI781288A (xx)
FR (2)	FR2388827A1 (xx)
GB (1)	GB1598294A (xx)
HK (1)	HK51484A (xx)
IE (2)	IE47271B1 (xx)
IT (2)	IT1156718B (xx)
KE (1)	KE3398A (xx)
LU (1)	LU79541A1 (xx)
MY (1)	MY8500528A (xx)
NL (1)	NL178790C (xx)
NO (2)	NO149635C (xx)
PL (1)	PL117307B1 (xx)
PT (1)	PT67959B (xx)
SE (2)	SE447259B (xx)
SG (1)	SG22884G (xx)
YU (2)	YU102578A (xx)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS55306A (en) *	1978-04-28	1980-01-05	Bristol Myers Co	Manufacture of 11nnomegaaaminooalphaahydroxy alkanoyl*aminoglycoside antibiotic
JP4621429B2 (ja) *	2002-02-19	2011-01-26	学校法人東海大学	乳酸誘導体
EP3150617B1 (en)	2007-11-21	2020-04-08	Cipla USA, Inc.	Antibacterial aminoglycoside analogs
WO2010132759A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of dibekacin
WO2010132757A2 (en) *	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial aminoglycoside analogs
WO2010132768A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of sisomicin
WO2010132765A2 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial aminoglycoside analogs
WO2010132760A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of tobramycin

1978
- 1978-04-21 AR AR271852A patent/AR218910A1/es active
- 1978-04-25 NO NO781437A patent/NO149635C/no unknown
- 1978-04-25 CA CA301,968A patent/CA1105454A/en not_active Expired
- 1978-04-25 FI FI781288A patent/FI781288A/fi not_active Application Discontinuation
- 1978-04-25 CA CA301,962A patent/CA1100953A/en not_active Expired
- 1978-04-26 CY CY1241A patent/CY1241A/en unknown
- 1978-04-26 NL NLAANVRAGE7804503,A patent/NL178790C/xx not_active IP Right Cessation
- 1978-04-26 GB GB16571/78A patent/GB1598294A/en not_active Expired
- 1978-04-26 DK DK197801830A patent/DK172543B1/da not_active IP Right Cessation
- 1978-04-26 DK DK182978A patent/DK165450C/da not_active IP Right Cessation
- 1978-04-27 IE IE842/78A patent/IE47271B1/en not_active IP Right Cessation
- 1978-04-27 CS CS782729A patent/CS207607B2/cs unknown
- 1978-04-27 FR FR7812591A patent/FR2388827A1/fr active Granted
- 1978-04-27 YU YU01025/78A patent/YU102578A/xx unknown
- 1978-04-27 IE IE841/78A patent/IE46945B1/en not_active IP Right Cessation
- 1978-04-27 LU LU79541A patent/LU79541A1/xx unknown
- 1978-04-27 PT PT67959A patent/PT67959B/pt unknown
- 1978-04-27 FR FR7812589A patent/FR2388826A1/fr active Granted
- 1978-04-27 YU YU1024/78A patent/YU41590B/xx unknown
- 1978-04-28 DE DE19782818822 patent/DE2818822A1/de active Granted
- 1978-04-28 AT AT312778A patent/AT357675B/de not_active IP Right Cessation
- 1978-04-28 JP JP5016078A patent/JPS53149951A/ja active Granted
- 1978-04-28 ES ES469303A patent/ES469303A1/es not_active Expired
- 1978-04-28 CH CH470278A patent/CH639104A5/de not_active IP Right Cessation
- 1978-04-28 DE DE19782818992 patent/DE2818992A1/de active Granted
- 1978-04-28 PL PL1978206457A patent/PL117307B1/pl unknown
- 1978-04-28 IT IT49136/78A patent/IT1156718B/it active
- 1978-04-28 SE SE7804973A patent/SE447259B/sv not_active IP Right Cessation
- 1978-04-28 IT IT49137/78A patent/IT1105500B/it active
- 1978-04-29 EG EG283/78A patent/EG13710A/xx active
1983
- 1983-04-05 NO NO83831197A patent/NO154697C/no unknown
- 1983-10-07 SE SE8305538A patent/SE461148B/sv not_active IP Right Cessation
1984
- 1984-03-12 SG SG228/84A patent/SG22884G/en unknown
- 1984-04-12 KE KE3398A patent/KE3398A/xx unknown
- 1984-06-22 HK HK514/84A patent/HK51484A/xx not_active IP Right Cessation
1985
- 1985-12-30 MY MY528/85A patent/MY8500528A/xx unknown

Also Published As

Publication number	Publication date
YU102578A (en)	1983-01-21
CA1100953A (en)	1981-05-12
GB1598294A (en)	1981-09-16
FR2388827B1 (xx)	1982-07-09
YU41590B (en)	1987-12-31
DE2818992A1 (de)	1978-11-23
PL117307B1 (en)	1981-07-31
SE461148B (sv)	1990-01-15
SE8305538D0 (sv)	1983-10-07
AR218910A1 (es)	1980-07-15
IT7849136A0 (it)	1978-04-28
NL178790B (nl)	1985-12-16
DE2818822A1 (de)	1978-11-09
AT357675B (de)	1980-07-25
IT7849137A0 (it)	1978-04-28
NO831197L (no)	1978-10-31
DK182978A (da)	1978-10-29
PL206457A1 (xx)	1980-03-24
IE780842L (en)	1978-10-28
DK165450B (da)	1992-11-30
FI781288A (fi)	1978-10-29
IE780841L (en)	1978-10-28
NO154697C (no)	1986-12-03
NL178790C (nl)	1986-05-16
PT67959A (en)	1978-05-01
LU79541A1 (fr)	1978-11-28
IT1156718B (it)	1987-02-04
NO149635C (no)	1984-05-23
DK183078A (da)	1978-10-29
CY1241A (en)	1984-06-29
IE46945B1 (en)	1983-11-16
JPS53149951A (en)	1978-12-27
HK51484A (en)	1984-06-22
FR2388827A1 (fr)	1978-11-24
MY8500528A (en)	1985-12-31
NO781437L (no)	1978-10-31
DK165450C (da)	1993-04-13
FR2388826A1 (fr)	1978-11-24
CS207607B2 (en)	1981-08-31
SG22884G (en)	1985-01-04
IT1105500B (it)	1985-11-04
YU102478A (en)	1982-10-31
DE2818822C2 (xx)	1989-01-26
DE2818992C2 (xx)	1988-03-17
EG13710A (en)	1982-09-30
ATA312778A (de)	1979-12-15
NO149635B (no)	1984-02-13
SE8305538L (sv)	1983-10-07
KE3398A (en)	1984-06-08
NO154697B (no)	1986-08-25
SE447259B (sv)	1986-11-03
CA1105454A (en)	1981-07-21
FR2388826B1 (xx)	1982-12-10
SE7804973L (sv)	1978-10-29
DK172543B1 (da)	1998-12-07
CH639104A5 (en)	1983-10-31
JPS5721277B2 (xx)	1982-05-06
NL7804503A (nl)	1978-10-31
PT67959B (en)	1980-03-05
ES469303A1 (es)	1979-09-16

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Legal Events

Date	Code	Title	Description
1998-06-03	MK9A	Patent expired