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HUP1100241A3 - Oxetane substituted pyrimidones - Google Patents

Oxetane substituted pyrimidones

Info

Publication number
HUP1100241A3
HUP1100241A3 HU1100241A HUP1100241A HUP1100241A3 HU P1100241 A3 HUP1100241 A3 HU P1100241A3 HU 1100241 A HU1100241 A HU 1100241A HU P1100241 A HUP1100241 A HU P1100241A HU P1100241 A3 HUP1100241 A3 HU P1100241A3
Authority
HU
Hungary
Prior art keywords
oxetane substituted
substituted pyrimidones
pyrimidones
oxetane
substituted
Prior art date
Application number
HU1100241A
Other languages
Hungarian (hu)
Original Assignee
Richter Gedeon Nyrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Nyrt filed Critical Richter Gedeon Nyrt
Priority to HU1100241A priority Critical patent/HUP1100241A3/en
Priority to PCT/HU2012/000032 priority patent/WO2012153154A1/en
Publication of HUP1100241A2 publication Critical patent/HUP1100241A2/en
Publication of HUP1100241A3 publication Critical patent/HUP1100241A3/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
HU1100241A 2011-05-06 2011-05-06 Oxetane substituted pyrimidones HUP1100241A3 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
HU1100241A HUP1100241A3 (en) 2011-05-06 2011-05-06 Oxetane substituted pyrimidones
PCT/HU2012/000032 WO2012153154A1 (en) 2011-05-06 2012-05-04 Oxetane substituted thieno pyrimidinones

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU1100241A HUP1100241A3 (en) 2011-05-06 2011-05-06 Oxetane substituted pyrimidones

Publications (2)

Publication Number Publication Date
HUP1100241A2 HUP1100241A2 (en) 2012-12-28
HUP1100241A3 true HUP1100241A3 (en) 2013-12-30

Family

ID=89990277

Family Applications (1)

Application Number Title Priority Date Filing Date
HU1100241A HUP1100241A3 (en) 2011-05-06 2011-05-06 Oxetane substituted pyrimidones

Country Status (2)

Country Link
HU (1) HUP1100241A3 (en)
WO (1) WO2012153154A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6669499B2 (en) * 2013-02-15 2020-03-18 カラ ファーマシューティカルズ インコーポレイテッド Therapeutic compounds
MX379159B (en) 2016-02-12 2025-03-10 Astellas Pharma Inc TETRAHYDROISOQUINOLINE DERIVATIVES.
CN113045523B (en) * 2019-12-27 2022-09-23 上海泓博智源医药股份有限公司 Preparation method of imidazoline pyridine compound intermediate

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1169027A (en) 1966-11-19 1969-10-29 Beecham Group Ltd Azetidine Derivatives
GB0124627D0 (en) 2001-10-15 2001-12-05 Smithkline Beecham Plc Novel compounds
EP1618112A1 (en) 2003-04-11 2006-01-25 SmithKline Beecham Corporation Heterocyclic mchr1 antagonists
US20070078125A1 (en) 2003-10-23 2007-04-05 Glaxo Group Limited Arylamine mch r1 antagonists
US20050176738A1 (en) 2003-11-07 2005-08-11 Neurocrine Biosciences, Inc. Melanin-concentrating hormone receptor antagonists and compositions and methods related thereto
EP1876179B1 (en) 2005-04-28 2015-03-25 Takeda Pharmaceutical Company Limited Thienopyrimidone compounds
JP2009501217A (en) 2005-07-15 2009-01-15 アストラゼネカ アクチボラグ Remedy
WO2007011286A1 (en) 2005-07-15 2007-01-25 Astrazeneca Ab Therapeutic agents
US7745447B2 (en) 2005-10-26 2010-06-29 Bristol-Myers Squibb Company Substituted thieno[3,2-D]pyrimidines as non-basic melanin concentrating hormone receptor-1 antagonists
US8618115B2 (en) 2005-10-26 2013-12-31 Bristol-Myers Squibb Company Substituted thieno[3,2-d]pyrimidinones as MCHR1 antagonists and methods for using them
CA2636879A1 (en) 2006-02-15 2007-08-23 Sanofi-Aventis Novel amino alcohol-substituted arylthienopyrimidinones, process for their preparation and their use as medicaments
CA2636605A1 (en) 2006-02-15 2007-08-23 Lothar Schwink Novel azacycly-substituted arylthienopyrimidinones, process for their preparation and their use as medicaments
WO2008002575A1 (en) 2006-06-26 2008-01-03 The Procter & Gamble Company Melanin concentrating hormone antagonists
WO2008020799A1 (en) 2006-08-18 2008-02-21 Astrazeneca Ab Thienopyrimidin-4-one and thienopyridazin-7-one derivatives as mch rl antagonists
WO2008131103A2 (en) 2007-04-17 2008-10-30 Vertex Pharmaceuticals Incorporated Drug discovery methods for aurora kinase inhibitors

Also Published As

Publication number Publication date
WO2012153154A1 (en) 2012-11-15
HUP1100241A2 (en) 2012-12-28

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Legal Events

Date Code Title Description
FA9A Lapse of provisional patent protection due to relinquishment or protection considered relinquished