HUP0100179A3 - Imidazopyrimidine and imidazopyridine derivatives and pharmaceutical compositions thereof - Google Patents
Imidazopyrimidine and imidazopyridine derivatives and pharmaceutical compositions thereofInfo
- Publication number
- HUP0100179A3 HUP0100179A3 HU0100179A HUP0100179A HUP0100179A3 HU P0100179 A3 HUP0100179 A3 HU P0100179A3 HU 0100179 A HU0100179 A HU 0100179A HU P0100179 A HUP0100179 A HU P0100179A HU P0100179 A3 HUP0100179 A3 HU P0100179A3
- Authority
- HU
- Hungary
- Prior art keywords
- imidazopyrimidine
- pharmaceutical compositions
- imidazopyridine derivatives
- imidazopyridine
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Addiction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US5162897P | 1997-07-03 | 1997-07-03 | |
US8066598P | 1998-04-03 | 1998-04-03 | |
PCT/US1998/013913 WO1999001454A1 (en) | 1997-07-03 | 1998-07-02 | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP0100179A2 HUP0100179A2 (hu) | 2001-11-28 |
HUP0100179A3 true HUP0100179A3 (en) | 2002-12-28 |
Family
ID=26729655
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU0100179A HUP0100179A3 (en) | 1997-07-03 | 1998-07-02 | Imidazopyrimidine and imidazopyridine derivatives and pharmaceutical compositions thereof |
Country Status (20)
Country | Link |
---|---|
US (3) | US6143743A (hu) |
EP (1) | EP0994877A1 (hu) |
JP (1) | JP2002507996A (hu) |
KR (1) | KR20010014431A (hu) |
CN (1) | CN1268137A (hu) |
AR (1) | AR016307A1 (hu) |
AU (1) | AU746706B2 (hu) |
BR (1) | BR9810508A (hu) |
CA (1) | CA2294117A1 (hu) |
EE (1) | EE04280B1 (hu) |
HR (1) | HRP980375A2 (hu) |
HU (1) | HUP0100179A3 (hu) |
IL (1) | IL133800A0 (hu) |
MY (1) | MY132871A (hu) |
NO (1) | NO316119B1 (hu) |
NZ (1) | NZ502642A (hu) |
PL (1) | PL337888A1 (hu) |
SK (1) | SK179899A3 (hu) |
TW (1) | TW589309B (hu) |
WO (1) | WO1999001454A1 (hu) |
Families Citing this family (75)
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AP1063A (en) * | 1996-12-11 | 2002-04-26 | Aventis Pharmaceuticals Products Inc | Preparation of [1s-[1a, 2b, 3b, 4a(S*)]-4-[7-[[1-3-chloro-2-thienyl) metthyl]propyl]amino]-3h-imidazo[4, 5-b]pyridin-3-YL]-N-ethyl-2,3-dihydroxycypentanecarboxamide. |
US6124463A (en) * | 1998-07-02 | 2000-09-26 | Dupont Pharmaceuticals | Benzimidazoles as corticotropin release factor antagonists |
US6365589B1 (en) * | 1998-07-02 | 2002-04-02 | Bristol-Myers Squibb Pharma Company | Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists |
EP1140941B1 (en) * | 1998-12-23 | 2004-10-20 | Bristol-Myers Squibb Pharma Company | Nitrogen containing heterobicycles as factor xa inhibitors |
US6271380B1 (en) * | 1998-12-30 | 2001-08-07 | Dupont Pharmaceuticals Company | 1H-imidazo[4,5-d]pyridazin-7-ones, 3H-imidazo-[4,5-c]pyridin-4-ones and corresponding thiones as corticotropin releasing factor (CRF) receptor ligands |
WO2000059908A2 (en) | 1999-04-06 | 2000-10-12 | Du Pont Pharmaceuticals Company | Pyrazolopyrimidines as crf antagonists |
AU4331500A (en) | 1999-04-06 | 2000-10-23 | Du Pont Pharmaceuticals Company | Pyrazolotriazines as crf antagonists |
US6432989B1 (en) | 1999-08-27 | 2002-08-13 | Pfizer Inc | Use of CRF antagonists to treat circadian rhythm disorders |
CA2392992A1 (en) * | 1999-12-17 | 2001-06-21 | Dupont Pharmaceuticals Company | Imidazopyrimidinyl and imidazopyridinyl derivatives |
KR20030016222A (ko) * | 2000-02-14 | 2003-02-26 | 니뽄 다바코 산교 가부시키가이샤 | 수술후 스트레스 예방ㆍ치료제 |
US20040077605A1 (en) * | 2001-06-20 | 2004-04-22 | Salvati Mark E. | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
AR028782A1 (es) | 2000-07-05 | 2003-05-21 | Taisho Pharmaceutical Co Ltd | Derivados heterociclicos tetrahidropiridino o piperidino |
EP1301511A2 (en) | 2000-07-14 | 2003-04-16 | Bristol-Myers Squibb Pharma Company | IMIDAZO 1,2-a]PYRAZINES FOR THE TREATMENT OF NEUROLOGICAL DISORDERS |
EP1854798A3 (en) | 2000-09-19 | 2007-11-28 | Bristol-Myers Squibb Company | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
GB0100623D0 (en) | 2001-01-10 | 2001-02-21 | Vernalis Res Ltd | Chemical compounds IV |
JP2004531475A (ja) | 2001-01-26 | 2004-10-14 | ブリストル−マイヤーズ スクイブ カンパニー | コルチコトロピン放出因子阻害剤としてのイミダゾリル誘導体 |
TWI312347B (en) | 2001-02-08 | 2009-07-21 | Eisai R&D Man Co Ltd | Bicyclic nitrogen-containing condensed ring compounds |
US20040087548A1 (en) | 2001-02-27 | 2004-05-06 | Salvati Mark E. | Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
NZ528207A (en) | 2001-03-13 | 2006-02-24 | Bristol Myers Squibb Pharma Co | 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-A]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands |
AU2002251546B2 (en) | 2001-04-27 | 2007-01-18 | Eisai R & D Management Co., Ltd. | Pyrazolo[1,5-A]pyridines and medicines containing the same |
DE60217669D1 (de) | 2001-05-14 | 2007-03-08 | Bristol Myers Squibb Co | Substitutierte pyrazinone, pyridine und pyrimidine als corticotropin-releasing-factor liganden |
AU2002354575A1 (en) | 2001-07-12 | 2003-01-29 | Bristol-Myers Squibb Pharma Company | Tetrahydropurinones as corticotropin releasing factor |
US7276526B2 (en) | 2001-07-13 | 2007-10-02 | Bristol-Myers Squibb Pharma Company | Substituted thiazoles and oxazoles as corticotropin releasing hormone ligands |
US20070129334A1 (en) * | 2001-10-30 | 2007-06-07 | Conforma Therapeutics Corporation | Orally Active Purine-Based Inhibitors of Heat Shock Protein 90 |
WO2003037860A2 (en) | 2001-10-30 | 2003-05-08 | Conforma Therapeutics Corporation | Purine analogs having hsp90-inhibiting activity |
WO2003043637A1 (en) | 2001-11-20 | 2003-05-30 | Bristol-Myers Squibb Pharma Company | 3,7-dihydro-purine-2,6-dione derivatives as crf receptor ligands |
JP4434740B2 (ja) | 2001-12-19 | 2010-03-17 | ブリストル−マイヤーズ スクイブ カンパニー | 核ホルモン受容体機能の調節剤である、縮合ヘテロ環化合物およびその類似体 |
CN100503608C (zh) * | 2002-01-07 | 2009-06-24 | 卫材R&D管理株式会社 | 脱氮嘌呤及其用途 |
AU2003220190A1 (en) | 2002-03-13 | 2003-09-29 | Pharmacia & Upjohn Company Llc | Pyrazolo(1,5-a)pyridine derivatives as neurotransmitter modulators |
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US7176216B2 (en) | 2002-10-22 | 2007-02-13 | Eisai Co., Ltd. | 7-phenylpyrazolopyridine compounds |
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US7332508B2 (en) | 2002-12-18 | 2008-02-19 | Novo Nordisk A/S | Substituted homopiperidine, piperidine or pyrrolidine derivatives |
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DE102004037554A1 (de) * | 2004-08-03 | 2006-03-16 | Sanofi-Aventis Deutschland Gmbh | Substituierte 8-Aminoalkylthio-xanthine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
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BRPI0911659B8 (pt) | 2008-04-15 | 2021-05-25 | Eisai R&D Man Co Ltd | composto 3-fenilpirazolo[5,1-b]tiazol e composição farmacêutica compreendendo o mesmo |
WO2009152584A1 (en) * | 2008-06-20 | 2009-12-23 | Macquarie University | Synthesis of ageladine a and analogs thereof |
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JP2024500919A (ja) | 2020-12-23 | 2024-01-10 | ジェンザイム・コーポレーション | 重水素化コロニー刺激因子-1受容体(csf-1r)阻害剤 |
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-
1998
- 1998-07-02 EP EP98931795A patent/EP0994877A1/en not_active Withdrawn
- 1998-07-02 IL IL13380098A patent/IL133800A0/xx unknown
- 1998-07-02 AU AU81819/98A patent/AU746706B2/en not_active Ceased
- 1998-07-02 KR KR1019997012619A patent/KR20010014431A/ko not_active Application Discontinuation
- 1998-07-02 JP JP50744099A patent/JP2002507996A/ja active Pending
- 1998-07-02 US US09/109,877 patent/US6143743A/en not_active Expired - Lifetime
- 1998-07-02 CN CN98808584A patent/CN1268137A/zh active Pending
- 1998-07-02 PL PL98337888A patent/PL337888A1/xx unknown
- 1998-07-02 HR HR60/080,665A patent/HRP980375A2/hr not_active Application Discontinuation
- 1998-07-02 NZ NZ502642A patent/NZ502642A/en unknown
- 1998-07-02 SK SK1798-99A patent/SK179899A3/sk unknown
- 1998-07-02 MY MYPI98003027A patent/MY132871A/en unknown
- 1998-07-02 HU HU0100179A patent/HUP0100179A3/hu unknown
- 1998-07-02 CA CA002294117A patent/CA2294117A1/en not_active Abandoned
- 1998-07-02 WO PCT/US1998/013913 patent/WO1999001454A1/en not_active Application Discontinuation
- 1998-07-02 TW TW087110857A patent/TW589309B/zh active
- 1998-07-02 BR BR9810508-6A patent/BR9810508A/pt not_active IP Right Cessation
- 1998-07-02 EE EEP199900607A patent/EE04280B1/xx not_active IP Right Cessation
- 1998-07-03 AR ARP980103234A patent/AR016307A1/es not_active Application Discontinuation
- 1998-12-10 US US09/208,778 patent/US6362180B1/en not_active Expired - Lifetime
-
1999
- 1999-12-27 NO NO19996483A patent/NO316119B1/no not_active IP Right Cessation
-
2001
- 2001-11-07 US US10/053,475 patent/US6642230B2/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
US6143743A (en) | 2000-11-07 |
IL133800A0 (en) | 2001-04-30 |
SK179899A3 (en) | 2001-12-03 |
CA2294117A1 (en) | 1999-01-14 |
HUP0100179A2 (hu) | 2001-11-28 |
AR016307A1 (es) | 2001-07-04 |
PL337888A1 (en) | 2000-09-11 |
WO1999001454A1 (en) | 1999-01-14 |
US6642230B2 (en) | 2003-11-04 |
AU8181998A (en) | 1999-01-25 |
NO996483L (no) | 2000-03-02 |
NO996483D0 (no) | 1999-12-27 |
US20030114468A1 (en) | 2003-06-19 |
MY132871A (en) | 2007-10-31 |
US6362180B1 (en) | 2002-03-26 |
HRP980375A2 (en) | 1999-04-30 |
BR9810508A (pt) | 2000-09-05 |
EE04280B1 (et) | 2004-04-15 |
KR20010014431A (ko) | 2001-02-26 |
JP2002507996A (ja) | 2002-03-12 |
AU746706B2 (en) | 2002-05-02 |
CN1268137A (zh) | 2000-09-27 |
TW589309B (en) | 2004-06-01 |
EP0994877A1 (en) | 2000-04-26 |
NO316119B1 (no) | 2003-12-15 |
NZ502642A (en) | 2002-06-28 |
EE9900607A (et) | 2000-08-15 |
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